JP2010518173A5 - - Google Patents

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Publication number
JP2010518173A5
JP2010518173A5 JP2009549760A JP2009549760A JP2010518173A5 JP 2010518173 A5 JP2010518173 A5 JP 2010518173A5 JP 2009549760 A JP2009549760 A JP 2009549760A JP 2009549760 A JP2009549760 A JP 2009549760A JP 2010518173 A5 JP2010518173 A5 JP 2010518173A5
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JP
Japan
Prior art keywords
salt
cancer
salts
group
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2009549760A
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English (en)
Japanese (ja)
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JP2010518173A (ja
JP5504460B2 (ja
Filing date
Publication date
Priority claimed from CNA2007100375572A external-priority patent/CN101245050A/zh
Application filed filed Critical
Publication of JP2010518173A publication Critical patent/JP2010518173A/ja
Publication of JP2010518173A5 publication Critical patent/JP2010518173A5/ja
Application granted granted Critical
Publication of JP5504460B2 publication Critical patent/JP5504460B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2009549760A 2007-02-14 2008-02-04 4−フェニルアミノキナゾリン誘導体の塩形態 Active JP5504460B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CNA2007100375572A CN101245050A (zh) 2007-02-14 2007-02-14 4-苯胺喹唑啉衍生物的盐
CN200710037557.2 2007-02-14
PCT/CN2008/000318 WO2008098485A1 (en) 2007-02-14 2008-02-04 The salts of 4-aniline quinazoline derivative

Publications (3)

Publication Number Publication Date
JP2010518173A JP2010518173A (ja) 2010-05-27
JP2010518173A5 true JP2010518173A5 (OSRAM) 2011-04-07
JP5504460B2 JP5504460B2 (ja) 2014-05-28

Family

ID=39689656

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009549760A Active JP5504460B2 (ja) 2007-02-14 2008-02-04 4−フェニルアミノキナゾリン誘導体の塩形態

Country Status (8)

Country Link
US (1) US8349854B2 (OSRAM)
EP (1) EP2116540B1 (OSRAM)
JP (1) JP5504460B2 (OSRAM)
KR (1) KR20100014947A (OSRAM)
CN (3) CN101245050A (OSRAM)
AU (1) AU2008215053B2 (OSRAM)
CA (1) CA2677978C (OSRAM)
WO (1) WO2008098485A1 (OSRAM)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101347433B (zh) * 2007-07-20 2012-05-02 江苏艾力斯生物医药有限公司 4-苯胺喹唑啉衍生物的制药用途
CN101544609A (zh) * 2008-03-25 2009-09-30 上海艾力斯医药科技有限公司 4-苯胺喹唑啉衍生物的结晶形式
CN101584696A (zh) 2008-05-21 2009-11-25 上海艾力斯医药科技有限公司 包含喹唑啉衍生物的组合物及制备方法、用途
CN108430972B (zh) 2015-12-24 2022-12-27 协和麒麟株式会社 α,β不饱和酰胺化合物
CN106117182B (zh) * 2016-06-20 2019-08-30 中国药科大学 喹唑啉-n-苯乙基四氢异喹啉类化合物及其制备方法和应用
CN112225679A (zh) * 2020-10-13 2021-01-15 苏州亚科科技股份有限公司 一种3-(环己胺)-2-羟基-1-丙磺酸的制备方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ243082A (en) 1991-06-28 1995-02-24 Ici Plc 4-anilino-quinazoline derivatives; pharmaceutical compositions, preparatory processes, and use thereof
AU661533B2 (en) 1992-01-20 1995-07-27 Astrazeneca Ab Quinazoline derivatives
GB9314893D0 (en) 1993-07-19 1993-09-01 Zeneca Ltd Quinazoline derivatives
GB9510757D0 (en) * 1994-09-19 1995-07-19 Wellcome Found Therapeuticaly active compounds
EP1110953B1 (en) 1995-03-30 2009-10-28 Pfizer Products Inc. Quinazoline derivatives
RO121900B1 (ro) 1996-04-12 2008-07-30 Warner-Lambert Company Compuşi inhibitori, ireversibili, ai tirozin kinazelor, compoziţie farmaceutică care îi conţine şi utilizarea acestora
GB9800575D0 (en) * 1998-01-12 1998-03-11 Glaxo Group Ltd Heterocyclic compounds
GB9800569D0 (en) 1998-01-12 1998-03-11 Glaxo Group Ltd Heterocyclic compounds
TW533204B (en) 1998-07-30 2003-05-21 Wyeth Corp A process for preparing substituted quinazoline derivatives
CZ300945B6 (cs) * 2000-06-30 2009-09-23 Glaxo Group Limited Zpusob prípravy 5-(6-chinazolinyl)-furan-2-karbaldehydu
KR100735639B1 (ko) * 2004-12-29 2007-07-04 한미약품 주식회사 암세포 성장 억제 효과를 갖는 퀴나졸린 유도체 및 이의제조방법
CN101003514A (zh) * 2006-01-20 2007-07-25 上海艾力斯医药科技有限公司 喹唑啉衍生物、其制备方法及用途

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