JP2010514733A - 高眼圧症の治療のためのイソソルビドモノニトレート誘導体 - Google Patents
高眼圧症の治療のためのイソソルビドモノニトレート誘導体 Download PDFInfo
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- JP2010514733A JP2010514733A JP2009543471A JP2009543471A JP2010514733A JP 2010514733 A JP2010514733 A JP 2010514733A JP 2009543471 A JP2009543471 A JP 2009543471A JP 2009543471 A JP2009543471 A JP 2009543471A JP 2010514733 A JP2010514733 A JP 2010514733A
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- cycloalkenyl
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Ophthalmology & Optometry (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06380338A EP1941876A1 (en) | 2006-12-28 | 2006-12-28 | Isosorbide mononitrate derivatives for the treatment of Inflammation and ocular hypertension |
| PCT/EP2007/064570 WO2008080939A1 (en) | 2006-12-28 | 2007-12-27 | Isosorbide mononitrate derivatives for the treatment of ocular hypertension |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010514733A true JP2010514733A (ja) | 2010-05-06 |
| JP2010514733A5 JP2010514733A5 (ru) | 2011-02-17 |
Family
ID=38043051
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009543471A Pending JP2010514733A (ja) | 2006-12-28 | 2007-12-27 | 高眼圧症の治療のためのイソソルビドモノニトレート誘導体 |
| JP2009543474A Pending JP2010514734A (ja) | 2006-12-28 | 2007-12-27 | 腸障害の治療のためのイソソルビドモノニトレート誘導体 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009543474A Pending JP2010514734A (ja) | 2006-12-28 | 2007-12-27 | 腸障害の治療のためのイソソルビドモノニトレート誘導体 |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US20080161389A1 (ru) |
| EP (3) | EP1941876A1 (ru) |
| JP (2) | JP2010514733A (ru) |
| KR (2) | KR20090112673A (ru) |
| CN (2) | CN101600425A (ru) |
| AR (1) | AR064543A1 (ru) |
| AT (2) | ATE484279T1 (ru) |
| AU (2) | AU2007341218B2 (ru) |
| BR (2) | BRPI0720663A2 (ru) |
| CA (2) | CA2674144A1 (ru) |
| CL (2) | CL2007003836A1 (ru) |
| DE (2) | DE602007009877D1 (ru) |
| ES (3) | ES2324130B1 (ru) |
| IL (2) | IL198912A0 (ru) |
| MX (2) | MX2009007038A (ru) |
| NO (2) | NO20092763L (ru) |
| PL (2) | PL2124930T3 (ru) |
| RU (2) | RU2009128970A (ru) |
| UY (1) | UY30847A1 (ru) |
| WO (2) | WO2008080939A1 (ru) |
| ZA (2) | ZA200903567B (ru) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2149577B1 (en) * | 2008-07-22 | 2011-04-27 | Lacer, S.A. | New stereospecific method for the preparation of dioxa-bicyclooctane compounds |
| EP2149576A1 (en) * | 2008-07-22 | 2010-02-03 | Lacer, S.A. | Isosorbide Nitrates having vasodilating activity |
| EP2177216A1 (en) * | 2008-10-13 | 2010-04-21 | Lacer, S.A. | Use of dianhydrohexite mononitrate derivatives as healing agents |
| WO2010055138A1 (en) * | 2008-11-14 | 2010-05-20 | Lacer, S.A. | New stereospecific method for the preparation of dioxa-bicyclooctane compounds |
| EP2199294A1 (en) * | 2008-12-19 | 2010-06-23 | Lacer, S.A. | New stereospecific method for the preparation of dioxa bicyclooctane nitrate compounds |
| DK2515899T3 (en) * | 2009-12-23 | 2016-08-15 | Arca Biopharma Inc | METHODS AND COMPOSITIONS FOR CARDIOVASCULAR DISEASES AND CONDITIONS |
| US20160016969A1 (en) * | 2013-03-05 | 2016-01-21 | Archer Daniels Midland Company | Isohexide monotriflates and process for synthesis thereof |
| WO2018224419A1 (en) | 2017-06-06 | 2018-12-13 | Nicox S.A. | Nitric oxide donating isomannide derivatives |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS60149521A (ja) * | 1984-01-18 | 1985-08-07 | Eisai Co Ltd | 高眼圧・緑内障治療・予防用点眼剤 |
| JP2002526544A (ja) * | 1998-10-07 | 2002-08-20 | レイサー ソシエダッド アノニマ | イソソルビドモノニトレートの誘導体及び耐性が低下した血管拡張剤としてのその使用 |
| WO2005037842A1 (en) * | 2003-10-03 | 2005-04-28 | Lácer, S.A. | Disulfide, sulfide, sulfoxide, and sulfone derivatives of cyclic sugars and uses thereof |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2739689C2 (de) * | 1977-09-02 | 1986-10-16 | Euratom | Thermische Wärmepumpe |
| US5573758A (en) * | 1995-04-28 | 1996-11-12 | Allergan | Method for reducing intraocular pressure in the mammalian eye by administration of potassium channel blockers |
| US5925342A (en) * | 1996-11-13 | 1999-07-20 | Allergan | Method for reducing intraocular pressure in the mammalian eye by administration of potassium channel blockers |
| GB9720797D0 (en) * | 1997-09-30 | 1997-12-03 | Rhodes John | Pharmaceutical composition for the treatment of inflammatory bowel disease and irritable bowel syndrome |
| US20040077664A1 (en) * | 2001-01-31 | 2004-04-22 | Hans-Michael Eggenweiler | Pharmaceutical formulation comprising pyrazolo[4,3-d]pyrimidine and nitrates or thienopyrimidines and nitrates |
| AU2003222049B2 (en) * | 2002-03-21 | 2007-05-31 | Cayman Chemical Company, Incorporated | Prostaglandin F2 alpha analogs in combination with antimicrobials for treating glaucoma |
| JP2007504807A (ja) * | 2003-09-08 | 2007-03-08 | ボード オブ リージェンツ オブ ザ ユニバーシティー オブ テキサス システム | 培養培地にプロスタグランジン又はプロスタグランジン類似物を補足することによってインビトロ胚発生を高めるための方法及び組成 |
-
2006
- 2006-12-28 EP EP06380338A patent/EP1941876A1/en not_active Withdrawn
-
2007
- 2007-01-23 ES ES200700181A patent/ES2324130B1/es not_active Expired - Fee Related
- 2007-03-01 US US11/680,691 patent/US20080161389A1/en not_active Abandoned
- 2007-12-27 RU RU2009128970/15A patent/RU2009128970A/ru not_active Application Discontinuation
- 2007-12-27 ES ES07858167T patent/ES2348314T3/es active Active
- 2007-12-27 CN CNA2007800441623A patent/CN101600425A/zh active Pending
- 2007-12-27 MX MX2009007038A patent/MX2009007038A/es active IP Right Grant
- 2007-12-27 MX MX2009007040A patent/MX2009007040A/es active IP Right Grant
- 2007-12-27 UY UY30847A patent/UY30847A1/es not_active Application Discontinuation
- 2007-12-27 CA CA002674144A patent/CA2674144A1/en not_active Abandoned
- 2007-12-27 EP EP07858187A patent/EP2124930B1/en active Active
- 2007-12-27 AU AU2007341218A patent/AU2007341218B2/en not_active Ceased
- 2007-12-27 ES ES07858187T patent/ES2354317T3/es active Active
- 2007-12-27 KR KR1020097015821A patent/KR20090112673A/ko not_active Application Discontinuation
- 2007-12-27 BR BRPI0720663-1A patent/BRPI0720663A2/pt not_active IP Right Cessation
- 2007-12-27 EP EP07858167A patent/EP2114398B1/en active Active
- 2007-12-27 AU AU2007341289A patent/AU2007341289B2/en not_active Ceased
- 2007-12-27 ZA ZA200903567A patent/ZA200903567B/xx unknown
- 2007-12-27 ZA ZA200903566A patent/ZA200903566B/xx unknown
- 2007-12-27 CL CL200703836A patent/CL2007003836A1/es unknown
- 2007-12-27 AR ARP070105911A patent/AR064543A1/es unknown
- 2007-12-27 KR KR1020097015820A patent/KR20100100584A/ko not_active Application Discontinuation
- 2007-12-27 PL PL07858187T patent/PL2124930T3/pl unknown
- 2007-12-27 WO PCT/EP2007/064570 patent/WO2008080939A1/en active Application Filing
- 2007-12-27 AT AT07858187T patent/ATE484279T1/de not_active IP Right Cessation
- 2007-12-27 PL PL07858167T patent/PL2114398T3/pl unknown
- 2007-12-27 AT AT07858167T patent/ATE472324T1/de not_active IP Right Cessation
- 2007-12-27 DE DE602007009877T patent/DE602007009877D1/de active Active
- 2007-12-27 JP JP2009543471A patent/JP2010514733A/ja active Pending
- 2007-12-27 BR BRPI0720664-0A patent/BRPI0720664A2/pt not_active IP Right Cessation
- 2007-12-27 WO PCT/EP2007/064591 patent/WO2008080955A1/en active Application Filing
- 2007-12-27 CN CN2007800443012A patent/CN101600426B/zh not_active Expired - Fee Related
- 2007-12-27 JP JP2009543474A patent/JP2010514734A/ja active Pending
- 2007-12-27 CL CL200703837A patent/CL2007003837A1/es unknown
- 2007-12-27 DE DE602007007523T patent/DE602007007523D1/de active Active
- 2007-12-27 RU RU2009128968/15A patent/RU2009128968A/ru not_active Application Discontinuation
- 2007-12-27 CA CA002674550A patent/CA2674550A1/en not_active Abandoned
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2009
- 2009-05-24 IL IL198912A patent/IL198912A0/en unknown
- 2009-05-25 IL IL198941A patent/IL198941A0/en unknown
- 2009-07-27 NO NO20092763A patent/NO20092763L/no not_active Application Discontinuation
- 2009-07-27 NO NO20092764A patent/NO20092764L/no not_active Application Discontinuation
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS60149521A (ja) * | 1984-01-18 | 1985-08-07 | Eisai Co Ltd | 高眼圧・緑内障治療・予防用点眼剤 |
| JP2002526544A (ja) * | 1998-10-07 | 2002-08-20 | レイサー ソシエダッド アノニマ | イソソルビドモノニトレートの誘導体及び耐性が低下した血管拡張剤としてのその使用 |
| WO2005037842A1 (en) * | 2003-10-03 | 2005-04-28 | Lácer, S.A. | Disulfide, sulfide, sulfoxide, and sulfone derivatives of cyclic sugars and uses thereof |
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