JP2010513531A5 - - Google Patents
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- Publication number
- JP2010513531A5 JP2010513531A5 JP2009542959A JP2009542959A JP2010513531A5 JP 2010513531 A5 JP2010513531 A5 JP 2010513531A5 JP 2009542959 A JP2009542959 A JP 2009542959A JP 2009542959 A JP2009542959 A JP 2009542959A JP 2010513531 A5 JP2010513531 A5 JP 2010513531A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- mixture
- reaction
- compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 0 CC(CC1)(C=C1C(OC)=O)c1ccc(*=C)cc1 Chemical compound CC(CC1)(C=C1C(OC)=O)c1ccc(*=C)cc1 0.000 description 4
- IOAMXHPKIUMBMD-NHYWBVRUSA-N C=C[C@](CC1)(C[C@H]1c(cc1)ccc1Br)C(NC(N)=O)=O Chemical compound C=C[C@](CC1)(C[C@H]1c(cc1)ccc1Br)C(NC(N)=O)=O IOAMXHPKIUMBMD-NHYWBVRUSA-N 0.000 description 2
- GFOKSKMVRLJJNR-IINYFYTJSA-N CN(C([C@@](CC1)(C[C@H]1c(cc1)ccc1Br)N1)=O)C1=O Chemical compound CN(C([C@@](CC1)(C[C@H]1c(cc1)ccc1Br)N1)=O)C1=O GFOKSKMVRLJJNR-IINYFYTJSA-N 0.000 description 1
- GFOKSKMVRLJJNR-HZMBPMFUSA-N CN(C([C@](CC1)(C[C@H]1c(cc1)ccc1Br)N1)=O)C1=O Chemical compound CN(C([C@](CC1)(C[C@H]1c(cc1)ccc1Br)N1)=O)C1=O GFOKSKMVRLJJNR-HZMBPMFUSA-N 0.000 description 1
- OVMPLGZIMNITFL-DGCLKSJQSA-N COc1ccc([C@H](CC2)C[C@]2(C#N)N)cc1 Chemical compound COc1ccc([C@H](CC2)C[C@]2(C#N)N)cc1 OVMPLGZIMNITFL-DGCLKSJQSA-N 0.000 description 1
- YYWBOYFAACOYTR-ZWNOBZJWSA-N COc1ccc([C@H](CC2)C[C@]2(C(O)=O)N)cc1 Chemical compound COc1ccc([C@H](CC2)C[C@]2(C(O)=O)N)cc1 YYWBOYFAACOYTR-ZWNOBZJWSA-N 0.000 description 1
- PKGWZXNPDCYMSH-SECBINFHSA-N C[C@H](CCNC(NC=O)=O)c(cc1)ccc1Br Chemical compound C[C@H](CCNC(NC=O)=O)c(cc1)ccc1Br PKGWZXNPDCYMSH-SECBINFHSA-N 0.000 description 1
- DRUFIZLVYAZXGE-JDRUZZMFSA-N O=C([C@](CC1)(C[C@H]1C1C=CC(Br)=CC1)N1)NC1=O Chemical compound O=C([C@](CC1)(C[C@H]1C1C=CC(Br)=CC1)N1)NC1=O DRUFIZLVYAZXGE-JDRUZZMFSA-N 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US87625106P | 2006-12-21 | 2006-12-21 | |
| PCT/US2007/026257 WO2008079380A1 (en) | 2006-12-21 | 2007-12-21 | Process for the preparation and isolation of the individual stereoisomers of 1-amino, 3-substituted phenylcyclopentane carboxylates |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010513531A JP2010513531A (ja) | 2010-04-30 |
| JP2010513531A5 true JP2010513531A5 (https=) | 2011-03-24 |
Family
ID=39562855
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009542959A Withdrawn JP2010513531A (ja) | 2006-12-21 | 2007-12-21 | １−アミノ、３−置換フェニルシクロペンタンカルボン酸エステルの個々の立体異性体の製造および単離方法 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7956195B2 (https=) |
| EP (1) | EP2102145A4 (https=) |
| JP (1) | JP2010513531A (https=) |
| CN (1) | CN101563316A (https=) |
| CA (1) | CA2673076A1 (https=) |
| MX (1) | MX2009006748A (https=) |
| RU (1) | RU2009128063A (https=) |
| WO (1) | WO2008079380A1 (https=) |
| ZA (1) | ZA200903874B (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2013006867A (es) * | 2010-12-22 | 2013-07-05 | Bayer Ip Gmbh | Procedimiento para la preparacion de sales de cis-1-amonio-4-alcoxiciclohexanocarbonitrilo. |
| CN107759483B (zh) * | 2016-08-16 | 2022-03-11 | 浙江瑞博制药有限公司 | 一种甲氨基取代的环戊烷甲酸烷基酯的制备方法 |
| CN115847629B (zh) * | 2022-11-30 | 2023-09-29 | 江苏富乐徳石英科技有限公司 | 一种高效节能环保的石英环制备工艺 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4841079A (en) * | 1987-08-07 | 1989-06-20 | Pfizer, Inc. | Process for the production of asymmetric hydantoins |
| JP3333510B2 (ja) * | 1991-10-02 | 2002-10-15 | スミスクライン・ビーチャム・コーポレイション | 抗アレルギー、抗炎症および腫瘍壊死因子抑制活性を有するシクロペンタンおよびシクロペンテン誘導体 |
| US5314896A (en) | 1991-11-20 | 1994-05-24 | Warner-Lambert Company | 1,3-substituted cycloalkenes and cycloalkanes as central nervous system agents |
| US20020052370A1 (en) * | 2000-07-06 | 2002-05-02 | Barber Christopher Gordon | Cyclopentyl-substituted glutaramide derivatives as inhibitors of neutral endopeptidase |
| EP1188826B1 (en) * | 2000-09-13 | 2011-06-08 | Ajinomoto Co., Inc. | 5-substituted hydantoin racemase, DNA coding for the same, and process for producing optically active amino acids |
| AU2003261774A1 (en) * | 2002-09-06 | 2004-03-29 | Kaneka Corporation | PROCESS FOR PRODUCING L-Alpha-METHYLCYSTEINE DERIVATIVE |
| TW200420573A (en) * | 2002-09-26 | 2004-10-16 | Rib X Pharmaceuticals Inc | Bifunctional heterocyclic compounds and methods of making and using same |
| US7256198B2 (en) * | 2004-02-18 | 2007-08-14 | Wyeth | Pyrimidoindolones and methods for using same |
| BRPI0519058A2 (pt) * | 2004-12-14 | 2008-12-23 | Astrazeneca Ab | composto ou um sal prà-droga farmaceuticamente aceitÁvel do mesmo, mÉtodos para produzir uma inibiÇço da atividade de dgat1 e para tratar diabete melito e/ou obesidade em um animal de sangue quente, uso de um composto, composiÇço farmacÊutica, e, processo para preparar um composto |
| US7754703B2 (en) | 2005-02-14 | 2010-07-13 | University Of Virginia Patent Foundation | Cycloalkane-containing sphingosine 1-phosphate agonists |
| US7521557B2 (en) * | 2005-05-20 | 2009-04-21 | Bristol-Myers Squibb Company | Pyrrolopyridine-based inhibitors of dipeptidyl peptidase IV and methods |
| JP2009528274A (ja) | 2006-01-27 | 2009-08-06 | ユニバーシティ オブ バージニア パテント ファンデーション | 神経因性疼痛の治療法 |
| KR20080096780A (ko) * | 2006-02-21 | 2008-11-03 | 유니버시티 오브 버지니아 페이턴트 파운데이션 | Ｓ１ｐ 수용체 효능제로서의 페닐-시클로알킬 및 페닐-헤테로시클릭 유도체 |
| BRPI0720478A2 (pt) * | 2006-12-21 | 2014-01-14 | Abbott Laboratoires | Compostos agonistas e antagonistas do receptor esfingosina-1-fosfato |
-
2007
- 2007-12-21 CA CA002673076A patent/CA2673076A1/en not_active Abandoned
- 2007-12-21 WO PCT/US2007/026257 patent/WO2008079380A1/en not_active Ceased
- 2007-12-21 CN CNA2007800467996A patent/CN101563316A/zh active Pending
- 2007-12-21 US US12/004,582 patent/US7956195B2/en not_active Expired - Fee Related
- 2007-12-21 EP EP07863231.2A patent/EP2102145A4/en not_active Withdrawn
- 2007-12-21 JP JP2009542959A patent/JP2010513531A/ja not_active Withdrawn
- 2007-12-21 MX MX2009006748A patent/MX2009006748A/es active IP Right Grant
- 2007-12-21 RU RU2009128063/04A patent/RU2009128063A/ru not_active Application Discontinuation
-
2009
- 2009-06-03 ZA ZA200903874A patent/ZA200903874B/xx unknown
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