JP2010513531A5 - - Google Patents
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- JP2010513531A5 JP2010513531A5 JP2009542959A JP2009542959A JP2010513531A5 JP 2010513531 A5 JP2010513531 A5 JP 2010513531A5 JP 2009542959 A JP2009542959 A JP 2009542959A JP 2009542959 A JP2009542959 A JP 2009542959A JP 2010513531 A5 JP2010513531 A5 JP 2010513531A5
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- JP
- Japan
- Prior art keywords
- formula
- compound
- mixture
- reaction
- compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 0 CC(CC1)(C=C1C(OC)=O)c1ccc(*=C)cc1 Chemical compound CC(CC1)(C=C1C(OC)=O)c1ccc(*=C)cc1 0.000 description 4
- IOAMXHPKIUMBMD-NHYWBVRUSA-N C=C[C@](CC1)(C[C@H]1c(cc1)ccc1Br)C(NC(N)=O)=O Chemical compound C=C[C@](CC1)(C[C@H]1c(cc1)ccc1Br)C(NC(N)=O)=O IOAMXHPKIUMBMD-NHYWBVRUSA-N 0.000 description 2
- GFOKSKMVRLJJNR-IINYFYTJSA-N CN(C([C@@](CC1)(C[C@H]1c(cc1)ccc1Br)N1)=O)C1=O Chemical compound CN(C([C@@](CC1)(C[C@H]1c(cc1)ccc1Br)N1)=O)C1=O GFOKSKMVRLJJNR-IINYFYTJSA-N 0.000 description 1
- GFOKSKMVRLJJNR-HZMBPMFUSA-N CN(C([C@](CC1)(C[C@H]1c(cc1)ccc1Br)N1)=O)C1=O Chemical compound CN(C([C@](CC1)(C[C@H]1c(cc1)ccc1Br)N1)=O)C1=O GFOKSKMVRLJJNR-HZMBPMFUSA-N 0.000 description 1
- OVMPLGZIMNITFL-DGCLKSJQSA-N COc1ccc([C@H](CC2)C[C@]2(C#N)N)cc1 Chemical compound COc1ccc([C@H](CC2)C[C@]2(C#N)N)cc1 OVMPLGZIMNITFL-DGCLKSJQSA-N 0.000 description 1
- YYWBOYFAACOYTR-ZWNOBZJWSA-N COc1ccc([C@H](CC2)C[C@]2(C(O)=O)N)cc1 Chemical compound COc1ccc([C@H](CC2)C[C@]2(C(O)=O)N)cc1 YYWBOYFAACOYTR-ZWNOBZJWSA-N 0.000 description 1
- PKGWZXNPDCYMSH-SECBINFHSA-N C[C@H](CCNC(NC=O)=O)c(cc1)ccc1Br Chemical compound C[C@H](CCNC(NC=O)=O)c(cc1)ccc1Br PKGWZXNPDCYMSH-SECBINFHSA-N 0.000 description 1
- DRUFIZLVYAZXGE-JDRUZZMFSA-N O=C([C@](CC1)(C[C@H]1C1C=CC(Br)=CC1)N1)NC1=O Chemical compound O=C([C@](CC1)(C[C@H]1C1C=CC(Br)=CC1)N1)NC1=O DRUFIZLVYAZXGE-JDRUZZMFSA-N 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US87625106P | 2006-12-21 | 2006-12-21 | |
| PCT/US2007/026257 WO2008079380A1 (en) | 2006-12-21 | 2007-12-21 | Process for the preparation and isolation of the individual stereoisomers of 1-amino, 3-substituted phenylcyclopentane carboxylates |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010513531A JP2010513531A (ja) | 2010-04-30 |
| JP2010513531A5 true JP2010513531A5 (https=) | 2011-03-24 |
Family
ID=39562855
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009542959A Withdrawn JP2010513531A (ja) | 2006-12-21 | 2007-12-21 | １−アミノ、３−置換フェニルシクロペンタンカルボン酸エステルの個々の立体異性体の製造および単離方法 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7956195B2 (https=) |
| EP (1) | EP2102145A4 (https=) |
| JP (1) | JP2010513531A (https=) |
| CN (1) | CN101563316A (https=) |
| CA (1) | CA2673076A1 (https=) |
| MX (1) | MX2009006748A (https=) |
| RU (1) | RU2009128063A (https=) |
| WO (1) | WO2008079380A1 (https=) |
| ZA (1) | ZA200903874B (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR101999937B1 (ko) * | 2010-12-22 | 2019-07-12 | 바이엘 인텔렉쳐 프로퍼티 게엠베하 | 시스-1-암모늄-4-알콕시시클로헥산카보니트릴 염의 제조 방법 |
| CN107759483B (zh) * | 2016-08-16 | 2022-03-11 | 浙江瑞博制药有限公司 | 一种甲氨基取代的环戊烷甲酸烷基酯的制备方法 |
| CN115847629B (zh) * | 2022-11-30 | 2023-09-29 | 江苏富乐徳石英科技有限公司 | 一种高效节能环保的石英环制备工艺 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4841079A (en) * | 1987-08-07 | 1989-06-20 | Pfizer, Inc. | Process for the production of asymmetric hydantoins |
| JP3333510B2 (ja) * | 1991-10-02 | 2002-10-15 | スミスクライン・ビーチャム・コーポレイション | 抗アレルギー、抗炎症および腫瘍壊死因子抑制活性を有するシクロペンタンおよびシクロペンテン誘導体 |
| US5314896A (en) | 1991-11-20 | 1994-05-24 | Warner-Lambert Company | 1,3-substituted cycloalkenes and cycloalkanes as central nervous system agents |
| US20020052370A1 (en) * | 2000-07-06 | 2002-05-02 | Barber Christopher Gordon | Cyclopentyl-substituted glutaramide derivatives as inhibitors of neutral endopeptidase |
| ATE512217T1 (de) * | 2000-09-13 | 2011-06-15 | Ajinomoto Kk | 5-substituerte hydantoin racemase, dafür kodierende dna, und verfahren zur herstellung optisch aktiver aminosäure |
| WO2004022766A1 (ja) * | 2002-09-06 | 2004-03-18 | Kaneka Corporation | Ｌ−αーメチルシステイン誘導体の製造方法 |
| AR043050A1 (es) * | 2002-09-26 | 2005-07-13 | Rib X Pharmaceuticals Inc | Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos |
| US7256198B2 (en) * | 2004-02-18 | 2007-08-14 | Wyeth | Pyrimidoindolones and methods for using same |
| US7795283B2 (en) * | 2004-12-14 | 2010-09-14 | Astrazeneca Ab | Oxadiazole derivative as DGAT inhibitors |
| AU2006214314B2 (en) | 2005-02-14 | 2012-02-09 | University Of Virginia Patent Foundation | Sphingosine 1- phos phate agonists comprising cycloalkanes and 5 -membered heterocycles substituted by amino and phenyl groups |
| US7521557B2 (en) * | 2005-05-20 | 2009-04-21 | Bristol-Myers Squibb Company | Pyrrolopyridine-based inhibitors of dipeptidyl peptidase IV and methods |
| KR20080086546A (ko) * | 2006-01-27 | 2008-09-25 | 유니버시티 오브 버지니아 페이턴트 파운데이션 | 신경병증성 통증의 치료 방법 |
| BRPI0707957A2 (pt) * | 2006-02-21 | 2011-05-17 | Univ Virginia Patent Found | composto, e, método para prevenção ou tratamento de uma condição ou sintoma patológico em um mamìfero |
| CL2007003784A1 (es) * | 2006-12-21 | 2008-06-27 | Abbott Lab | Compuestos derivados de 1-amino-3-fenilciclopentano, que son agonistas o antagonistas de uno o mas receptores de la familia s1p; composicion farmaceutica que comprende a dichos compuestos; y su uso para tratar la esclerosis multiple, artritis reumato |
-
2007
- 2007-12-21 CA CA002673076A patent/CA2673076A1/en not_active Abandoned
- 2007-12-21 JP JP2009542959A patent/JP2010513531A/ja not_active Withdrawn
- 2007-12-21 US US12/004,582 patent/US7956195B2/en not_active Expired - Fee Related
- 2007-12-21 WO PCT/US2007/026257 patent/WO2008079380A1/en not_active Ceased
- 2007-12-21 RU RU2009128063/04A patent/RU2009128063A/ru not_active Application Discontinuation
- 2007-12-21 MX MX2009006748A patent/MX2009006748A/es active IP Right Grant
- 2007-12-21 CN CNA2007800467996A patent/CN101563316A/zh active Pending
- 2007-12-21 EP EP07863231.2A patent/EP2102145A4/en not_active Withdrawn
-
2009
- 2009-06-03 ZA ZA200903874A patent/ZA200903874B/xx unknown
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