JP2010513531A5 - - Google Patents
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- Publication number
- JP2010513531A5 JP2010513531A5 JP2009542959A JP2009542959A JP2010513531A5 JP 2010513531 A5 JP2010513531 A5 JP 2010513531A5 JP 2009542959 A JP2009542959 A JP 2009542959A JP 2009542959 A JP2009542959 A JP 2009542959A JP 2010513531 A5 JP2010513531 A5 JP 2010513531A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- mixture
- reaction
- compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 0 CC(CC1)(C=C1C(OC)=O)c1ccc(*=C)cc1 Chemical compound CC(CC1)(C=C1C(OC)=O)c1ccc(*=C)cc1 0.000 description 4
- IOAMXHPKIUMBMD-NHYWBVRUSA-N C=C[C@](CC1)(C[C@H]1c(cc1)ccc1Br)C(NC(N)=O)=O Chemical compound C=C[C@](CC1)(C[C@H]1c(cc1)ccc1Br)C(NC(N)=O)=O IOAMXHPKIUMBMD-NHYWBVRUSA-N 0.000 description 2
- GFOKSKMVRLJJNR-IINYFYTJSA-N CN(C([C@@](CC1)(C[C@H]1c(cc1)ccc1Br)N1)=O)C1=O Chemical compound CN(C([C@@](CC1)(C[C@H]1c(cc1)ccc1Br)N1)=O)C1=O GFOKSKMVRLJJNR-IINYFYTJSA-N 0.000 description 1
- GFOKSKMVRLJJNR-HZMBPMFUSA-N CN(C([C@](CC1)(C[C@H]1c(cc1)ccc1Br)N1)=O)C1=O Chemical compound CN(C([C@](CC1)(C[C@H]1c(cc1)ccc1Br)N1)=O)C1=O GFOKSKMVRLJJNR-HZMBPMFUSA-N 0.000 description 1
- OVMPLGZIMNITFL-DGCLKSJQSA-N COc1ccc([C@H](CC2)C[C@]2(C#N)N)cc1 Chemical compound COc1ccc([C@H](CC2)C[C@]2(C#N)N)cc1 OVMPLGZIMNITFL-DGCLKSJQSA-N 0.000 description 1
- YYWBOYFAACOYTR-ZWNOBZJWSA-N COc1ccc([C@H](CC2)C[C@]2(C(O)=O)N)cc1 Chemical compound COc1ccc([C@H](CC2)C[C@]2(C(O)=O)N)cc1 YYWBOYFAACOYTR-ZWNOBZJWSA-N 0.000 description 1
- PKGWZXNPDCYMSH-SECBINFHSA-N C[C@H](CCNC(NC=O)=O)c(cc1)ccc1Br Chemical compound C[C@H](CCNC(NC=O)=O)c(cc1)ccc1Br PKGWZXNPDCYMSH-SECBINFHSA-N 0.000 description 1
- DRUFIZLVYAZXGE-JDRUZZMFSA-N O=C([C@](CC1)(C[C@H]1C1C=CC(Br)=CC1)N1)NC1=O Chemical compound O=C([C@](CC1)(C[C@H]1C1C=CC(Br)=CC1)N1)NC1=O DRUFIZLVYAZXGE-JDRUZZMFSA-N 0.000 description 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US87625106P | 2006-12-21 | 2006-12-21 | |
| PCT/US2007/026257 WO2008079380A1 (en) | 2006-12-21 | 2007-12-21 | Process for the preparation and isolation of the individual stereoisomers of 1-amino, 3-substituted phenylcyclopentane carboxylates |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2010513531A JP2010513531A (ja) | 2010-04-30 |
| JP2010513531A5 true JP2010513531A5 (enExample) | 2011-03-24 |
Family
ID=39562855
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009542959A Withdrawn JP2010513531A (ja) | 2006-12-21 | 2007-12-21 | １−アミノ、３−置換フェニルシクロペンタンカルボン酸エステルの個々の立体異性体の製造および単離方法 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US7956195B2 (enExample) |
| EP (1) | EP2102145A4 (enExample) |
| JP (1) | JP2010513531A (enExample) |
| CN (1) | CN101563316A (enExample) |
| CA (1) | CA2673076A1 (enExample) |
| MX (1) | MX2009006748A (enExample) |
| RU (1) | RU2009128063A (enExample) |
| WO (1) | WO2008079380A1 (enExample) |
| ZA (1) | ZA200903874B (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN103270020B (zh) * | 2010-12-22 | 2016-01-20 | 拜耳知识产权有限责任公司 | 制备顺-1-铵-4-烷氧基环己甲腈盐的方法 |
| CN107759483B (zh) * | 2016-08-16 | 2022-03-11 | 浙江瑞博制药有限公司 | 一种甲氨基取代的环戊烷甲酸烷基酯的制备方法 |
| CN115847629B (zh) * | 2022-11-30 | 2023-09-29 | 江苏富乐徳石英科技有限公司 | 一种高效节能环保的石英环制备工艺 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4841079A (en) * | 1987-08-07 | 1989-06-20 | Pfizer, Inc. | Process for the production of asymmetric hydantoins |
| EP0642489A1 (en) * | 1991-10-02 | 1995-03-15 | Smithkline Beecham Corporation | Cyclopentane and cyclopentene derivatives with antiallergic antiinflammatory and tumor necrosis factor inhibiting activity |
| US5314896A (en) | 1991-11-20 | 1994-05-24 | Warner-Lambert Company | 1,3-substituted cycloalkenes and cycloalkanes as central nervous system agents |
| US20020052370A1 (en) * | 2000-07-06 | 2002-05-02 | Barber Christopher Gordon | Cyclopentyl-substituted glutaramide derivatives as inhibitors of neutral endopeptidase |
| EP1188826B1 (en) * | 2000-09-13 | 2011-06-08 | Ajinomoto Co., Inc. | 5-substituted hydantoin racemase, DNA coding for the same, and process for producing optically active amino acids |
| US20060051846A1 (en) * | 2002-09-06 | 2006-03-09 | Kaneka Corporation | Process for producing l-alpha-methylcysteine derivative |
| AR043050A1 (es) | 2002-09-26 | 2005-07-13 | Rib X Pharmaceuticals Inc | Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos |
| US7256198B2 (en) | 2004-02-18 | 2007-08-14 | Wyeth | Pyrimidoindolones and methods for using same |
| AU2005315430B2 (en) * | 2004-12-14 | 2010-05-27 | Astrazeneca Ab | Oxadiazole derivatives as DGAT inhibitors |
| MX2007009848A (es) | 2005-02-14 | 2008-03-10 | Univ Virginia | Agonistas de esfingosina 1-fosfato comprendiendo cicloalcanos y heterociclos de 5 miembros substituidos por grupos amino y fenilo. |
| US7521557B2 (en) | 2005-05-20 | 2009-04-21 | Bristol-Myers Squibb Company | Pyrrolopyridine-based inhibitors of dipeptidyl peptidase IV and methods |
| MX2008009579A (es) * | 2006-01-27 | 2008-09-25 | Univ Virginia | Metodo para el tratamiento de dolor neuropatico. |
| BRPI0707957A2 (pt) * | 2006-02-21 | 2011-05-17 | Univ Virginia Patent Found | composto, e, método para prevenção ou tratamento de uma condição ou sintoma patológico em um mamìfero |
| CA2672727A1 (en) * | 2006-12-21 | 2008-07-03 | Abbott Laboratories | Sphingosine-1-phosphate receptor agonist and antagonist compounds |
-
2007
- 2007-12-21 EP EP07863231.2A patent/EP2102145A4/en not_active Withdrawn
- 2007-12-21 CA CA002673076A patent/CA2673076A1/en not_active Abandoned
- 2007-12-21 WO PCT/US2007/026257 patent/WO2008079380A1/en not_active Ceased
- 2007-12-21 RU RU2009128063/04A patent/RU2009128063A/ru not_active Application Discontinuation
- 2007-12-21 US US12/004,582 patent/US7956195B2/en not_active Expired - Fee Related
- 2007-12-21 CN CNA2007800467996A patent/CN101563316A/zh active Pending
- 2007-12-21 JP JP2009542959A patent/JP2010513531A/ja not_active Withdrawn
- 2007-12-21 MX MX2009006748A patent/MX2009006748A/es active IP Right Grant
-
2009
- 2009-06-03 ZA ZA200903874A patent/ZA200903874B/xx unknown
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