JP2010510987A - ヘテロアリールアミド誘導体 - Google Patents
ヘテロアリールアミド誘導体 Download PDFInfo
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- JP2010510987A JP2010510987A JP2009538419A JP2009538419A JP2010510987A JP 2010510987 A JP2010510987 A JP 2010510987A JP 2009538419 A JP2009538419 A JP 2009538419A JP 2009538419 A JP2009538419 A JP 2009538419A JP 2010510987 A JP2010510987 A JP 2010510987A
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- Prior art keywords
- alkyl
- mono
- amino
- substituted
- aminocarbonyl
- Prior art date
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Classifications
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| US86724806P | 2006-11-27 | 2006-11-27 | |
| PCT/US2007/024396 WO2008066789A2 (en) | 2006-11-27 | 2007-11-27 | Heteroaryl amide derivatives |
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- 2007-11-27 JP JP2009538419A patent/JP2010510987A/ja active Pending
- 2007-11-27 US US12/516,480 patent/US8431593B2/en not_active Expired - Fee Related
- 2007-11-27 CA CA002670636A patent/CA2670636A1/en not_active Abandoned
- 2007-11-27 NZ NZ577814A patent/NZ577814A/en not_active IP Right Cessation
- 2007-11-27 WO PCT/US2007/024396 patent/WO2008066789A2/en not_active Ceased
- 2007-11-27 BR BRPI0719280-0A patent/BRPI0719280A2/pt not_active IP Right Cessation
- 2007-11-27 CN CN200780049692A patent/CN101621931A/zh active Pending
- 2007-11-27 EP EP13150025.8A patent/EP2591675A1/en not_active Withdrawn
- 2007-11-27 ZA ZA200904477A patent/ZA200904477B/xx unknown
- 2007-11-27 EA EA201300152A patent/EA201300152A1/ru unknown
- 2007-11-27 EP EP07862234.7A patent/EP2096923B1/en active Active
- 2007-11-27 MX MX2009005478A patent/MX2009005478A/es active IP Right Grant
- 2007-11-27 MY MYPI20092150 patent/MY150731A/en unknown
- 2007-11-27 UA UAA200906538A patent/UA99448C2/ru unknown
- 2007-11-27 EA EA200970516A patent/EA018036B1/ru not_active IP Right Cessation
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2013
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| JP2009542595A (ja) * | 2006-07-06 | 2009-12-03 | グラクソ グループ リミテッド | Ｐ２ｘ７受容体アンタゴニストとしての置換ｎ−フェニルメチル−５−オキソ−プロリン−２−アミドおよびそれらの使用方法 |
| JP2016508967A (ja) * | 2012-12-12 | 2016-03-24 | アクテリオン ファーマシューティカルズ リミテッドＡｃｔｅｌｉｏｎ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｌｔｄ | Ｐ２ｘ７受容体アンタゴニストとしてのインドールカルボキサミド誘導体 |
| JP2016504995A (ja) * | 2012-12-18 | 2016-02-18 | アクテリオン ファーマシューティカルズ リミテッドＡｃｔｅｌｉｏｎ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｌｔｄ | Ｐ２ｘ７受容体アンタゴニストとしてのインドールカルボキサミド誘導体 |
| JP2016506915A (ja) * | 2013-01-22 | 2016-03-07 | アクテリオン ファーマシューティカルズ リミテッドＡｃｔｅｌｉｏｎ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｌｔｄ | Ｐ２ｘ７受容体アンタゴニストとしての複素環アミド誘導体 |
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| EA037989B1 (ru) * | 2016-09-26 | 2021-06-21 | Тюгай Сэяку Кабусики Кайся | Производные пиразолопиридина, обладающие эффектом агониста рецептора glp-1 |
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| JP7280929B2 (ja) | 2016-09-26 | 2023-05-24 | 中外製薬株式会社 | Ｇｌｐ－１受容体アゴニスト作用を持つピラゾロピリジン誘導体 |
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| JP7602573B2 (ja) | 2016-09-26 | 2024-12-18 | 中外製薬株式会社 | Ｇｌｐ－１受容体アゴニスト作用を持つピラゾロピリジン誘導体 |
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| JP2019099571A (ja) * | 2017-11-29 | 2019-06-24 | 中外製薬株式会社 | Ｇｌｐ−１受容体アゴニスト作用を持つピラゾロピリジン誘導体を含有する医薬組成物 |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2008066789A2 (en) | 2008-06-05 |
| BRPI0719280A2 (pt) | 2014-03-11 |
| CO6190582A2 (es) | 2010-08-19 |
| NZ577814A (en) | 2012-03-30 |
| AU2007325780B9 (en) | 2013-09-12 |
| CA2670636A1 (en) | 2008-06-05 |
| EP2096923A4 (en) | 2011-01-12 |
| EA201300152A1 (ru) | 2013-07-30 |
| MX2009005478A (es) | 2009-08-12 |
| CN101621931A (zh) | 2010-01-06 |
| EA200970516A1 (ru) | 2009-12-30 |
| ZA200904477B (en) | 2010-09-29 |
| NO20092444L (no) | 2009-08-27 |
| EP2591675A1 (en) | 2013-05-15 |
| EP2096923B1 (en) | 2014-01-22 |
| US20130172549A1 (en) | 2013-07-04 |
| UA99448C2 (en) | 2012-08-27 |
| US8431593B2 (en) | 2013-04-30 |
| US20100216763A1 (en) | 2010-08-26 |
| EA018036B1 (ru) | 2013-05-30 |
| AU2007325780A1 (en) | 2008-06-05 |
| MY150731A (en) | 2014-02-28 |
| WO2008066789A3 (en) | 2008-08-21 |
| AU2007325780B2 (en) | 2013-05-02 |
| EP2096923A2 (en) | 2009-09-09 |
| KR20090094336A (ko) | 2009-09-04 |
| IL198827A0 (en) | 2010-02-17 |
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