JP2009542785A5 - - Google Patents

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Publication number
JP2009542785A5
JP2009542785A5 JP2009518952A JP2009518952A JP2009542785A5 JP 2009542785 A5 JP2009542785 A5 JP 2009542785A5 JP 2009518952 A JP2009518952 A JP 2009518952A JP 2009518952 A JP2009518952 A JP 2009518952A JP 2009542785 A5 JP2009542785 A5 JP 2009542785A5
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JP
Japan
Prior art keywords
besylate
salt
salt according
formula
compound
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JP2009518952A
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English (en)
Japanese (ja)
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JP2009542785A (ja
JP5433413B2 (ja
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Priority claimed from GB0613694A external-priority patent/GB0613694D0/en
Priority claimed from GB0613692A external-priority patent/GB0613692D0/en
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Priority claimed from PCT/GB2007/002565 external-priority patent/WO2008007071A1/en
Publication of JP2009542785A publication Critical patent/JP2009542785A/ja
Publication of JP2009542785A5 publication Critical patent/JP2009542785A5/ja
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Publication of JP5433413B2 publication Critical patent/JP5433413B2/ja
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JP2009518952A 2006-07-10 2007-07-10 短時間作用型ベンゾジアゼピンの塩およびそれらの多形形態 Active JP5433413B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB0613692.3 2006-07-10
GB0613694A GB0613694D0 (en) 2006-07-10 2006-07-10 Benzodiazepine salts
GB0613694.9 2006-07-10
GB0613692A GB0613692D0 (en) 2006-07-10 2006-07-10 Benzodiazepine salts
PCT/GB2007/002565 WO2008007071A1 (en) 2006-07-10 2007-07-10 Short-acting benzodiazepine salts and their polymorphic forms

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2012235328A Division JP5785923B2 (ja) 2006-07-10 2012-10-25 短時間作用型ベンゾジアゼピンの塩およびそれらの多形形態

Publications (3)

Publication Number Publication Date
JP2009542785A JP2009542785A (ja) 2009-12-03
JP2009542785A5 true JP2009542785A5 (https=) 2011-07-28
JP5433413B2 JP5433413B2 (ja) 2014-03-05

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ID=38535381

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2009518952A Active JP5433413B2 (ja) 2006-07-10 2007-07-10 短時間作用型ベンゾジアゼピンの塩およびそれらの多形形態
JP2012235328A Active JP5785923B2 (ja) 2006-07-10 2012-10-25 短時間作用型ベンゾジアゼピンの塩およびそれらの多形形態

Family Applications After (1)

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JP2012235328A Active JP5785923B2 (ja) 2006-07-10 2012-10-25 短時間作用型ベンゾジアゼピンの塩およびそれらの多形形態

Country Status (17)

Country Link
US (7) US9193730B2 (https=)
EP (1) EP2081921B1 (https=)
JP (2) JP5433413B2 (https=)
KR (3) KR20150081370A (https=)
CN (3) CN103288834B (https=)
AT (1) ATE480532T1 (https=)
AU (1) AU2007274054B2 (https=)
BR (1) BRPI0714886B8 (https=)
CA (1) CA2657347C (https=)
DE (1) DE602007009128D1 (https=)
DK (1) DK2081921T3 (https=)
MX (1) MX2009000404A (https=)
PL (1) PL2081921T3 (https=)
PT (1) PT2081921E (https=)
RU (1) RU2470935C2 (https=)
SI (1) SI2081921T1 (https=)
WO (1) WO2008007071A1 (https=)

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GB0613693D0 (en) 2006-07-10 2006-08-16 Cenes Ltd Benzodiazepine salts (3)
CA2657347C (en) 2006-07-10 2014-11-18 Paion Uk Limited Short-acting benzodiazepine salts and their polymorphic forms
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EP2450039A1 (en) 2010-11-08 2012-05-09 PAION UK Ltd. Dosing regimen for sedation with CNS 7056 (Remimazolam)
NZ702063A (en) * 2012-05-22 2016-11-25 Paion Uk Ltd Compositions comprising short-acting benzodiazepines
UA116452C2 (uk) * 2012-08-31 2018-03-26 ПАЙОН ЮКей ЛІМІТЕД Режим дозування седативного засобу
AR094963A1 (es) 2013-03-04 2015-09-09 Ono Pharmaceutical Co Reacción de oxidación excelente en el índice de conversión
HUE047450T2 (hu) 2014-07-23 2020-04-28 Jiangsu Nhwaluokang Pharmaceutical Res And Development Co Ltd Új benzodiazepin származék és alkalmazása
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CN110511224A (zh) * 2016-04-08 2019-11-29 四川科伦药物研究院有限公司 苯并二氮杂*衍生物的盐及其晶体形式、制备方法和用途
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CN108503644B (zh) * 2016-12-09 2019-06-14 成都倍特药业有限公司 一种苯并二氮杂*衍生物的氢溴酸盐及其制备方法和用途
WO2018148361A1 (en) 2017-02-09 2018-08-16 Watson Laboratories Inc. Process for the preparation of remimazolam and solid state forms of remimazolam salts
CN108948018B (zh) * 2017-05-17 2021-03-30 四川科伦博泰生物医药股份有限公司 苯并二氮*衍生物及其盐和相关晶体形式、制备方法和用途
EA202091927A1 (ru) 2018-02-13 2020-12-07 Цзянсу Нхвалокан Фармасьютикал Рисерч Энд Дивелопмент Ко., Лтд. Гидрохлорид производного бензодиазепина и кристаллическая форма, способ их получения и применения
CN110398514B (zh) * 2018-04-24 2023-04-28 恒天纤维集团有限公司 一种快速判断纤维素胶液中金属杂质含量的方法
ES2803099B2 (es) * 2019-07-22 2021-11-08 Moehs Iberica Sl Procedimiento de obtención de besilato de remimazolam amorfo
CN114478535B (zh) * 2020-10-23 2024-02-09 成都苑东生物制药股份有限公司 一种苯磺酸瑞马唑仑ii晶型的制备方法
WO2023037237A1 (en) * 2021-09-09 2023-03-16 Wavelength Enterprises Ltd Process for the preparation of remimazolam
US12540140B2 (en) 2022-04-08 2026-02-03 Fresenius Kabi Oncology Ltd. Process for the preparation of remimazolam
CN115448927A (zh) * 2022-10-20 2022-12-09 重庆瑞泊莱医药科技有限公司 一种氢溴酸依匹斯汀晶型ii及其制备方法
WO2025052259A1 (en) 2023-09-05 2025-03-13 Reena Patel Ready to use compositions of remimazolam

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AR094963A1 (es) 2013-03-04 2015-09-09 Ono Pharmaceutical Co Reacción de oxidación excelente en el índice de conversión

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