JP2009538327A5 - - Google Patents

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Publication number
JP2009538327A5
JP2009538327A5 JP2009512222A JP2009512222A JP2009538327A5 JP 2009538327 A5 JP2009538327 A5 JP 2009538327A5 JP 2009512222 A JP2009512222 A JP 2009512222A JP 2009512222 A JP2009512222 A JP 2009512222A JP 2009538327 A5 JP2009538327 A5 JP 2009538327A5
Authority
JP
Japan
Prior art keywords
compound
optionally substituted
alkyl
piperidinyl
activating protease
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2009512222A
Other languages
English (en)
Japanese (ja)
Other versions
JP2009538327A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2007/069059 external-priority patent/WO2007137080A2/en
Publication of JP2009538327A publication Critical patent/JP2009538327A/ja
Publication of JP2009538327A5 publication Critical patent/JP2009538327A5/ja
Pending legal-status Critical Current

Links

JP2009512222A 2006-05-23 2007-05-16 チャネル活性化プロテアーゼ阻害剤である化合物および組成物 Pending JP2009538327A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US80298306P 2006-05-23 2006-05-23
US86060406P 2006-11-22 2006-11-22
PCT/US2007/069059 WO2007137080A2 (en) 2006-05-23 2007-05-16 Compounds and compositions as channel activating protease inhibitors

Publications (2)

Publication Number Publication Date
JP2009538327A JP2009538327A (ja) 2009-11-05
JP2009538327A5 true JP2009538327A5 (enExample) 2010-07-01

Family

ID=38565503

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009512222A Pending JP2009538327A (ja) 2006-05-23 2007-05-16 チャネル活性化プロテアーゼ阻害剤である化合物および組成物

Country Status (14)

Country Link
US (2) US7951823B2 (enExample)
EP (1) EP2027143A2 (enExample)
JP (1) JP2009538327A (enExample)
KR (1) KR101069051B1 (enExample)
AR (1) AR061109A1 (enExample)
AU (1) AU2007253819B2 (enExample)
BR (1) BRPI0712021A2 (enExample)
CA (1) CA2651762A1 (enExample)
CL (1) CL2007001481A1 (enExample)
MX (1) MX2008014839A (enExample)
PE (1) PE20080708A1 (enExample)
RU (1) RU2419626C2 (enExample)
TW (1) TW200813094A (enExample)
WO (1) WO2007137080A2 (enExample)

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CA2677485A1 (en) * 2007-02-09 2008-08-14 Irm Llc Compounds and compositions as channel activating protease inhibitors
CA2677487A1 (en) 2007-02-09 2008-08-14 Irm Llc Compounds and compositions as channel activating protease inhibitors
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JP2013518897A (ja) * 2010-02-03 2013-05-23 エムイーエイチ アソシエイツ，インコーポレイテッド 選択的および生体活性的等配電子体としての多重置換フルオロメタン
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EP3204352B1 (en) * 2014-10-06 2020-07-01 Cortexyme, Inc. Inhibitors of lysine gingipain
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AU2020349353A1 (en) 2019-09-17 2022-04-14 Duke University Alvelestat for use in the treatment of graft rejection, bronchiolitis obliterans syndrome and graft versus host disease
HUE064089T2 (hu) 2020-04-16 2024-02-28 Mereo Biopharma 4 Ltd Alvelesztat neutrofil elasztáz inhibitort alkalmazó módszerek alfa-1-antitripszin hiány által közvetített légzõszervi megbetegedés kezelésére
AU2022373971A1 (en) 2021-10-20 2024-04-04 Mereo Biopharma 4 Limited Neutrophil elastase inhibitors for use in the treatment of fibrosis

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