JP2009536147A - 経口経粘膜送達用の生体接着性薬調合物 - Google Patents
経口経粘膜送達用の生体接着性薬調合物 Download PDFInfo
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- A—HUMAN NECESSITIES
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61J—CONTAINERS SPECIALLY ADAPTED FOR MEDICAL OR PHARMACEUTICAL PURPOSES; DEVICES OR METHODS SPECIALLY ADAPTED FOR BRINGING PHARMACEUTICAL PRODUCTS INTO PARTICULAR PHYSICAL OR ADMINISTERING FORMS; DEVICES FOR ADMINISTERING FOOD OR MEDICINES ORALLY; BABY COMFORTERS; DEVICES FOR RECEIVING SPITTLE
- A61J3/00—Devices or methods specially adapted for bringing pharmaceutical products into particular physical or administering forms
- A61J3/005—Coating of tablets or the like
Landscapes
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- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
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| PCT/US2007/000528 WO2007081948A2 (en) | 2006-01-06 | 2007-01-08 | Bioadhesive drug formulations for oral transmucosal delivery |
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2010518086A (ja) * | 2007-02-09 | 2010-05-27 | デュレクト コーポレーション | スフェンタニルおよびナロキソンを含む経口腔投与製剤 |
| JP2013527846A (ja) * | 2010-04-30 | 2013-07-04 | アロヴェイト・エルエルシー | 口腔粘膜を介してアレルギーを減感作するための方法、物品及びキット |
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| US20020119187A1 (en) * | 2000-09-29 | 2002-08-29 | Cantor Adam S. | Composition for the transdermal delivery of fentanyl |
| DE02715112T1 (de) * | 2001-03-16 | 2007-04-19 | Alza Corp., Mountain View | Transdermales pflaster zur verabreichung von fentanyl |
| US20050208117A1 (en) * | 2001-03-16 | 2005-09-22 | Venkatraman Subramanian S | Transdermal administration of fentanyl and analogs thereof |
| US8753308B2 (en) | 2006-01-06 | 2014-06-17 | Acelrx Pharmaceuticals, Inc. | Methods for administering small volume oral transmucosal dosage forms using a dispensing device |
| US8865743B2 (en) | 2006-01-06 | 2014-10-21 | Acelrx Pharmaceuticals, Inc. | Small volume oral transmucosal dosage forms containing sufentanil for treatment of pain |
| US8202535B2 (en) | 2006-01-06 | 2012-06-19 | Acelrx Pharmaceuticals, Inc. | Small-volume oral transmucosal dosage forms |
| US8357114B2 (en) | 2006-01-06 | 2013-01-22 | Acelrx Pharmaceuticals, Inc. | Drug dispensing device with flexible push rod |
| US9289583B2 (en) | 2006-01-06 | 2016-03-22 | Acelrx Pharmaceuticals, Inc. | Methods for administering small volume oral transmucosal dosage forms using a dispensing device |
| US9066847B2 (en) | 2007-01-05 | 2015-06-30 | Aceirx Pharmaceuticals, Inc. | Storage and dispensing devices for administration of oral transmucosal dosage forms |
| US8535714B2 (en) | 2006-01-06 | 2013-09-17 | Acelrx Pharmaceuticals, Inc. | Small volume oral transmucosal dosage forms containing sufentanil for treatment of pain |
| US8252329B2 (en) | 2007-01-05 | 2012-08-28 | Acelrx Pharmaceuticals, Inc. | Bioadhesive drug formulations for oral transmucosal delivery |
| US20110008431A1 (en) * | 2007-04-02 | 2011-01-13 | Toyo Boseki Kabushiki Kaisha | Therapeutic tablet for postherpetic neuralgia and method of treating postherpetic neuralgia |
| CA2704929C (en) | 2007-08-07 | 2018-05-15 | Pamela Palmer | Compositions and methods for procedural sedation and analgesia using oral transmucosal dosage forms |
| NZ584190A (en) * | 2007-10-15 | 2012-09-28 | Alza Corp | Once-a-day replacement transdermal administration of fentanyl |
| DE102008014533A1 (de) * | 2008-03-15 | 2009-09-17 | Lts Lohmann Therapie-Systeme Ag | Gingival-Wafer |
| US20090286832A1 (en) * | 2008-05-15 | 2009-11-19 | Kiichiro Nabeta | Narcotic emulsion formulations for treatment of surgical pain |
| US8807070B2 (en) * | 2008-08-07 | 2014-08-19 | Vector Corporation | Rotor processor for dry powders |
| US20100034968A1 (en) * | 2008-08-07 | 2010-02-11 | Vector Corporation | Polymer coating process using dry glidant in a rotor processor |
| US20100034967A1 (en) * | 2008-08-07 | 2010-02-11 | Vector Corporation | Dry polymer layering using a rotor processor |
| US8945592B2 (en) * | 2008-11-21 | 2015-02-03 | Acelrx Pharmaceuticals, Inc. | Sufentanil solid dosage forms comprising oxygen scavengers and methods of using the same |
| KR20110099747A (ko) | 2009-02-26 | 2011-09-08 | 테이코쿠 팔마 유에스에이, 인코포레이티드 | 암 통증 치료용 마취 유상액 제제 |
| US8548623B2 (en) | 2009-03-18 | 2013-10-01 | Acelrx Pharmaceuticals, Inc. | Storage and dispensing devices for administration of oral transmucosal dosage forms |
| US20110091544A1 (en) * | 2009-10-16 | 2011-04-21 | Acelrx Pharmaceuticals, Inc. | Compositions and Methods for Mild Sedation, Anxiolysis and Analgesia in the Procedural Setting |
| WO2011137422A2 (en) | 2010-04-30 | 2011-11-03 | Apellis Pharmaceuticals, Inc. | Methods and articles for preventing or reducing risk of developing a hyperallergenic immune system |
| US20110288128A1 (en) | 2010-05-21 | 2011-11-24 | Acelrx Pharmaceuticals, Inc. | Oral Transmucosal Administration of Sufentanil |
| PH12014500316B1 (en) | 2011-09-19 | 2018-10-03 | Orexo Ab | New abuse-resistant pharmaceutical composition for the treatment of opioid dependence |
| TR201815935T4 (tr) | 2012-05-02 | 2018-11-21 | Orexo Ab | Akut ağrının tedavisi için yeni alfentanil bileşimi. |
| US9770514B2 (en) | 2013-09-03 | 2017-09-26 | ExxPharma Therapeutics LLC | Tamper-resistant pharmaceutical dosage forms |
| US11058856B2 (en) | 2014-12-23 | 2021-07-13 | Acelrx Pharmaceuticals, Inc. | Systems, devices and methods for dispensing oral transmucosal dosage forms |
| NZ741171A (en) | 2015-09-10 | 2022-01-28 | Impel Neuropharma Inc | In-line nasal delivery device |
| PT3682915T (pt) | 2015-10-30 | 2023-06-26 | Acelrx Pharmaceuticals Inc | Aparelho e métodos para dispensar formas de dosagem trasnmucosa oral |
| JP7317020B2 (ja) | 2018-01-05 | 2023-07-28 | インペル ファーマシューティカルズ インコーポレイテッド | 精密嗅覚デバイスによるジヒドロエルゴタミンの鼻腔内送達 |
| WO2025097068A1 (en) * | 2023-11-01 | 2025-05-08 | Entrega Inc. | Oral dosage form with ionically chargeable hydrogel for delivery of active agent and permeation enhancer |
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Also Published As
| Publication number | Publication date |
|---|---|
| WO2007081948A2 (en) | 2007-07-19 |
| US20070207207A1 (en) | 2007-09-06 |
| CA2636119A1 (en) | 2007-07-19 |
| EP1968554A2 (en) | 2008-09-17 |
| US8252328B2 (en) | 2012-08-28 |
| KR20080084858A (ko) | 2008-09-19 |
| WO2007081948A3 (en) | 2008-04-03 |
| EP1968554A4 (en) | 2013-01-23 |
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