JP2009531465A5 - - Google Patents

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Publication number
JP2009531465A5
JP2009531465A5 JP2009503340A JP2009503340A JP2009531465A5 JP 2009531465 A5 JP2009531465 A5 JP 2009531465A5 JP 2009503340 A JP2009503340 A JP 2009503340A JP 2009503340 A JP2009503340 A JP 2009503340A JP 2009531465 A5 JP2009531465 A5 JP 2009531465A5
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JP
Japan
Prior art keywords
acetone
cooled
hours
polymorph
washed
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JP2009503340A
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English (en)
Japanese (ja)
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JP4477097B2 (ja
JP2009531465A (ja
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Priority claimed from PCT/US2007/068446 external-priority patent/WO2007134034A1/en
Publication of JP2009531465A publication Critical patent/JP2009531465A/ja
Publication of JP2009531465A5 publication Critical patent/JP2009531465A5/ja
Application granted granted Critical
Publication of JP4477097B2 publication Critical patent/JP4477097B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2009503340A 2006-05-09 2007-05-08 中枢神経系障害の治療のための(2s)−(4e)−n−メチル−5−[3−(5−イソプロポキシピリジン)イル]−4−ペンテン−2−アミンの多形形態 Expired - Fee Related JP4477097B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US74682106P 2006-05-09 2006-05-09
PCT/US2007/068446 WO2007134034A1 (en) 2006-05-09 2007-05-08 Polymorph forms of (2s) - (4e) -n-methyl-5- (3-isopropoxypyridin) yl] -4-penten-2-amine for the treatment of central nervous system disorders

Publications (3)

Publication Number Publication Date
JP2009531465A JP2009531465A (ja) 2009-09-03
JP2009531465A5 true JP2009531465A5 (https=) 2009-11-05
JP4477097B2 JP4477097B2 (ja) 2010-06-09

Family

ID=38441430

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009503340A Expired - Fee Related JP4477097B2 (ja) 2006-05-09 2007-05-08 中枢神経系障害の治療のための(2s)−(4e)−n−メチル−5−[3−(5−イソプロポキシピリジン)イル]−4−ペンテン−2−アミンの多形形態

Country Status (29)

Country Link
US (3) US8461344B2 (https=)
EP (2) EP2418201B1 (https=)
JP (1) JP4477097B2 (https=)
KR (1) KR20090005369A (https=)
CN (1) CN101472893A (https=)
AR (1) AR060786A1 (https=)
AU (1) AU2007249485B2 (https=)
BR (1) BRPI0709781A2 (https=)
CA (1) CA2649961A1 (https=)
DK (1) DK2418201T3 (https=)
EC (1) ECSP088876A (https=)
ES (1) ES2460919T3 (https=)
HR (1) HRP20140385T1 (https=)
IL (1) IL194833A0 (https=)
MX (1) MX2008013982A (https=)
MY (1) MY144132A (https=)
NO (1) NO20084567L (https=)
NZ (1) NZ597177A (https=)
PL (1) PL2418201T3 (https=)
PT (1) PT2418201E (https=)
RS (1) RS53286B (https=)
RU (1) RU2440984C2 (https=)
SA (1) SA07280230B1 (https=)
SI (1) SI2418201T1 (https=)
TW (1) TWI389889B (https=)
UA (1) UA96447C2 (https=)
UY (1) UY30330A1 (https=)
WO (1) WO2007134034A1 (https=)
ZA (1) ZA200809284B (https=)

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US7790757B2 (en) 1998-06-16 2010-09-07 Targacept, Inc. Compounds capable of activating cholinergic receptors
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US7459469B2 (en) 2004-11-10 2008-12-02 Targacept, Inc. Hydroxybenzoate salts of metanicotine compounds
TWI389889B (zh) * 2006-05-09 2013-03-21 Targacept Inc (2s)-(4e)-n-甲基-5-〔3-(5-異丙氧基吡啶)基〕-4-戊烯-2-胺之新穎多晶型
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WO2008091592A1 (en) * 2007-01-22 2008-07-31 Targacept, Inc. Intranasal, buccal, and sublingual administration of metanicotine analogs
KR20100052490A (ko) * 2007-07-31 2010-05-19 타가셉트 인코포레이티드 (2s)-(4e)-n-메틸-5-(3-(5-이소프로폭시피리딘)일)-4-펜텐-2-아민의 경피투여
JP2011522886A (ja) * 2008-06-11 2011-08-04 アストラゼネカ・アクチエボラーグ (2s)−(4e)−n−メチル−5−(3−(5−イソプロポキシピリジン)イル)−4−ペンテン−2−アミンを含む舌下組成物
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FR2959107B1 (fr) 2010-04-23 2015-03-27 Oreal Unite d'application d'un produit cosmetique
US8703802B2 (en) * 2010-05-20 2014-04-22 Targacept, Inc. Process for the preparation of aryl substituted olefinic amines
WO2013184732A1 (en) * 2012-06-06 2013-12-12 Targacept, Inc. Crystalline (2s)-(4e)-n-methyl-5-[3-(5-isopropoxypyridin)yl]4-penten-2-amine 1,5-naphthalenedisulfonate
KR101579904B1 (ko) 2014-09-05 2016-01-05 동신대학교산학협력단 마스카라

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