JP2009518301A5 - - Google Patents

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Publication number
JP2009518301A5
JP2009518301A5 JP2008543496A JP2008543496A JP2009518301A5 JP 2009518301 A5 JP2009518301 A5 JP 2009518301A5 JP 2008543496 A JP2008543496 A JP 2008543496A JP 2008543496 A JP2008543496 A JP 2008543496A JP 2009518301 A5 JP2009518301 A5 JP 2009518301A5
Authority
JP
Japan
Prior art keywords
alkyl
pyrazolo
chlorophenylsulfonyl
tetrahydro
pyridine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2008543496A
Other languages
English (en)
Japanese (ja)
Other versions
JP2009518301A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2006/046039 external-priority patent/WO2007064914A2/en
Publication of JP2009518301A publication Critical patent/JP2009518301A/ja
Publication of JP2009518301A5 publication Critical patent/JP2009518301A5/ja
Pending legal-status Critical Current

Links

JP2008543496A 2005-12-01 2006-12-01 5−(アリールスルホニル)−ピラゾロピペリジン Pending JP2009518301A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US74136605P 2005-12-01 2005-12-01
PCT/US2006/046039 WO2007064914A2 (en) 2005-12-01 2006-12-01 5-(arylsulfonyl)-pyrazolopiperidines

Publications (2)

Publication Number Publication Date
JP2009518301A JP2009518301A (ja) 2009-05-07
JP2009518301A5 true JP2009518301A5 (https=) 2010-01-21

Family

ID=38092841

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008543496A Pending JP2009518301A (ja) 2005-12-01 2006-12-01 5−(アリールスルホニル)−ピラゾロピペリジン

Country Status (18)

Country Link
US (2) US7732609B2 (https=)
EP (1) EP1957458A2 (https=)
JP (1) JP2009518301A (https=)
KR (1) KR20080073359A (https=)
CN (1) CN101370776A (https=)
AR (1) AR057959A1 (https=)
AU (1) AU2006320423B2 (https=)
BR (1) BRPI0619633A2 (https=)
CA (1) CA2632227A1 (https=)
EA (1) EA014906B1 (https=)
EC (1) ECSP088593A (https=)
IL (1) IL190608A0 (https=)
MA (1) MA30089B1 (https=)
MY (1) MY149422A (https=)
NZ (1) NZ568109A (https=)
PE (1) PE20071090A1 (https=)
TW (1) TW200736255A (https=)
WO (1) WO2007064914A2 (https=)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT2029602E (pt) * 2006-05-31 2010-07-08 Galapagos Nv Compostos de triazolopirazina uteis para o tratamento de doenãas degenerativas e inflamatërias
JP2010528036A (ja) * 2007-05-25 2010-08-19 エラン ファーマシューティカルズ,インコーポレイテッド γセクレターゼの阻害剤としてのピラゾロピロリジン
MX2010010773A (es) 2008-04-01 2011-04-11 Abbott Gmbh & Co Kg Tetrahidroisoquinolinas, composiciones farmaceuticas que las contienen y su uso en terapia.
TW201038569A (en) * 2009-02-16 2010-11-01 Abbott Gmbh & Co Kg Heterocyclic compounds, pharmaceutical compositions containing them, and their use in therapy
AR075442A1 (es) 2009-02-16 2011-03-30 Abbott Gmbh & Co Kg Derivados de aminotetralina, composiciones farmaceuticas que las contienen y sus usos en terapia
JP2012521993A (ja) * 2009-03-25 2012-09-20 エラン ファーマシューティカルズ,インコーポレイテッド 縮合三環式スルホンアミドの製造プロセス
US8883839B2 (en) 2010-08-13 2014-11-11 Abbott Laboratories Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy
US9051280B2 (en) 2010-08-13 2015-06-09 AbbVie Deutschland GmbH & Co. KG Tetraline and indane derivatives, pharmaceutical compositions containing them, and their use in therapy
US8846743B2 (en) 2010-08-13 2014-09-30 Abbott Laboratories Aminoindane derivatives, pharmaceutical compositions containing them, and their use in therapy
US9045459B2 (en) 2010-08-13 2015-06-02 AbbVie Deutschland GmbH & Co. KG Phenalkylamine derivatives, pharmaceutical compositions containing them, and their use in therapy
US8877794B2 (en) 2010-08-13 2014-11-04 Abbott Laboratories Phenalkylamine derivatives, pharmaceutical compositions containing them, and their use in therapy
US9309200B2 (en) 2011-05-12 2016-04-12 AbbVie Deutschland GmbH & Co. KG Benzazepine derivatives, pharmaceutical compositions containing them, and their use in therapy
CA2844275A1 (en) 2011-08-05 2013-02-14 AbbVie Deutschland GmbH & Co. KG Aminochromane, aminothiochromane and amino-1,2,3,4-tetrahydroquinoline derivatives, pharmaceutical compositions containing them, and their use in therapy
MX2014006004A (es) 2011-11-18 2015-04-16 Abbvie Deutschland Derivados de aminobenzociclohepteno, aminotetralina, aminoindano y fenalcilamina n-sustituidas, composiciones farmaceuticas que los contienen, y su uso en terapia.
US9365512B2 (en) 2012-02-13 2016-06-14 AbbVie Deutschland GmbH & Co. KG Isoindoline derivatives, pharmaceutical compositions containing them, and their use in therapy
US9656955B2 (en) 2013-03-15 2017-05-23 Abbvie Inc. Pyrrolidine derivatives, pharmaceutical compositions containing them, and their use in therapy
US9650334B2 (en) 2013-03-15 2017-05-16 Abbvie Inc. Pyrrolidine derivatives, pharmaceutical compositions containing them, and their use in therapy
CA2924689A1 (en) 2013-10-17 2015-04-23 AbbVie Deutschland GmbH & Co. KG Aminochromane, aminothiochromane and amino-1,2,3,4-tetrahydroquinoline derivatives, pharmaceutical compositions containing them, and their use in therapy
MX2016004934A (es) 2013-10-17 2016-12-20 Abbvie Deutschland Derivados de aminotetralina y aminoindano, composiciones farmaceuticas que los contienen, y su uso en terapia.
CN104059063A (zh) * 2014-04-03 2014-09-24 丽水绿氟科技有限公司 7,7-二氟-4,5,6,7-四氢吡唑并[4,3-c]吡啶及其衍生物的制备方法
BR112020018094A2 (pt) 2018-03-08 2020-12-22 Incyte Corporation Compostos de aminopirazina diol como inibidores de pi3k-¿
US11046658B2 (en) 2018-07-02 2021-06-29 Incyte Corporation Aminopyrazine derivatives as PI3K-γ inhibitors

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL319758A1 (en) * 1994-10-20 1997-08-18 Pfizer Bicyclic tetrahydropyrasole pyridines and their application as medicines
ES2349762T3 (es) * 2000-08-10 2011-01-11 Pfizer Italia S.R.L. Biciclo-pirazoles activos como inhibidores de quinasas, procedimientos para su preparación y composiciones farmacéuticas que los comprenden.
US7375115B2 (en) * 2001-10-09 2008-05-20 Kyorin Pharmaceutical Co., Ltd. 4-(2-furoyl) aminopiperidines, intermediates in synthesizing the same, process for producing the same and medicinal use of the same
AU2003292724A1 (en) * 2002-12-27 2004-07-29 Japan Tobacco Inc. Fused n-containing heterocyclic compounds and medicinal use thereof
CA2567343A1 (en) * 2004-05-20 2005-12-01 Elan Pharmaceuticals, Inc. N-cyclic sulfonamido inhibitors of gamma secretase
US20060089378A1 (en) * 2004-10-27 2006-04-27 Mingde Xia Tetrahydro-pyridinyl pyrazole cannabinoid modulators
DE102005002500A1 (de) * 2005-01-19 2006-07-27 Sanofi-Aventis Deutschland Gmbh Tetrahydrofuranderivate als Inhibitoren von Matrix-Metalloproteinasen
TW200716628A (en) * 2005-03-22 2007-05-01 Astrazeneca Ab Novel compounds
DE102005016170A1 (de) * 2005-04-07 2006-10-12 Grünenthal GmbH 4,5,6,7- Tetrahydro-isoxazolo(4,5c)pyridin-Verbindungen und deren Verwendung zur Herstellung von Arzneimitteln
BRPI0614944A2 (pt) 2005-08-19 2011-04-26 Elan Pharm Inc inibidores sulfonamido n-bicìclicos ponte de gama-secretase

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