JP2009502829A5 - - Google Patents

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Publication number
JP2009502829A5
JP2009502829A5 JP2008523188A JP2008523188A JP2009502829A5 JP 2009502829 A5 JP2009502829 A5 JP 2009502829A5 JP 2008523188 A JP2008523188 A JP 2008523188A JP 2008523188 A JP2008523188 A JP 2008523188A JP 2009502829 A5 JP2009502829 A5 JP 2009502829A5
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JP
Japan
Prior art keywords
alkylene
alkyl
halogen
aryl
compound according
Prior art date
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Application number
JP2008523188A
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English (en)
Japanese (ja)
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JP2009502829A (ja
JP5060478B2 (ja
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Priority claimed from PCT/EP2006/007139 external-priority patent/WO2007012421A1/en
Publication of JP2009502829A publication Critical patent/JP2009502829A/ja
Publication of JP2009502829A5 publication Critical patent/JP2009502829A5/ja
Application granted granted Critical
Publication of JP5060478B2 publication Critical patent/JP5060478B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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JP2008523188A 2005-07-26 2006-07-20 Rho−キナーゼ阻害剤としてのピペリジニル置換されたイソキノロン誘導体 Expired - Lifetime JP5060478B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP05016154.6 2005-07-26
EP05016154 2005-07-26
PCT/EP2006/007139 WO2007012421A1 (en) 2005-07-26 2006-07-20 Piperidinyl-substituted isoquinolone derivatives as rho-kinase inhibitors

Publications (3)

Publication Number Publication Date
JP2009502829A JP2009502829A (ja) 2009-01-29
JP2009502829A5 true JP2009502829A5 (enExample) 2009-09-03
JP5060478B2 JP5060478B2 (ja) 2012-10-31

Family

ID=34979095

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2008523188A Expired - Lifetime JP5060478B2 (ja) 2005-07-26 2006-07-20 Rho−キナーゼ阻害剤としてのピペリジニル置換されたイソキノロン誘導体

Country Status (31)

Country Link
US (1) US8188117B2 (enExample)
EP (2) EP2385047B1 (enExample)
JP (1) JP5060478B2 (enExample)
KR (1) KR101373535B1 (enExample)
CN (1) CN101228149B (enExample)
AR (1) AR054868A1 (enExample)
AU (1) AU2006274245B2 (enExample)
BR (1) BRPI0613861B8 (enExample)
CA (1) CA2615577C (enExample)
CR (1) CR9603A (enExample)
DK (1) DK1910333T3 (enExample)
DO (1) DOP2006000178A (enExample)
EC (1) ECSP088135A (enExample)
ES (1) ES2423006T3 (enExample)
GT (1) GT200600328A (enExample)
IL (1) IL188702A (enExample)
MA (1) MA29636B1 (enExample)
MX (1) MX2008001053A (enExample)
MY (1) MY148479A (enExample)
NI (1) NI200800025A (enExample)
NO (1) NO341888B1 (enExample)
NZ (1) NZ565668A (enExample)
PE (1) PE20070217A1 (enExample)
PT (1) PT1910333E (enExample)
RU (1) RU2414467C2 (enExample)
TN (1) TNSN08039A1 (enExample)
TW (1) TWI383979B (enExample)
UA (1) UA93882C2 (enExample)
UY (1) UY29697A1 (enExample)
WO (1) WO2007012421A1 (enExample)
ZA (1) ZA200710951B (enExample)

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ATE502027T1 (de) 2006-12-27 2011-04-15 Sanofi Aventis Substituierte isochinoline und ihre verwendung als rho-kinase-inhibitoren
JP5421783B2 (ja) 2006-12-27 2014-02-19 サノフイ Rhoキナーゼ阻害剤としての置換イソキノロン及びイソキノリノン誘導体
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BR122019007990B1 (pt) 2013-11-18 2021-05-04 Forma Therapeutics, Inc Composto, e, composição farmacêutica
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