JP2008500284A5 - - Google Patents

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Publication number
JP2008500284A5
JP2008500284A5 JP2007513296A JP2007513296A JP2008500284A5 JP 2008500284 A5 JP2008500284 A5 JP 2008500284A5 JP 2007513296 A JP2007513296 A JP 2007513296A JP 2007513296 A JP2007513296 A JP 2007513296A JP 2008500284 A5 JP2008500284 A5 JP 2008500284A5
Authority
JP
Japan
Prior art keywords
pyridin
urea
tert
phenyl
butylphenoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2007513296A
Other languages
English (en)
Japanese (ja)
Other versions
JP2008500284A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2005/016422 external-priority patent/WO2005113511A1/en
Publication of JP2008500284A publication Critical patent/JP2008500284A/ja
Publication of JP2008500284A5 publication Critical patent/JP2008500284A5/ja
Pending legal-status Critical Current

Links

JP2007513296A 2004-05-12 2005-05-11 血栓症の治療に有用なp2y1レセプターのウレアアンタゴニスト Pending JP2008500284A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US57028804P 2004-05-12 2004-05-12
US66581705P 2005-03-28 2005-03-28
PCT/US2005/016422 WO2005113511A1 (en) 2004-05-12 2005-05-11 Urea antagonists of p2y1 receptor useful in the treatment of thrombotic conditions
US11/126,915 US7388021B2 (en) 2004-05-12 2005-05-11 Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions

Publications (2)

Publication Number Publication Date
JP2008500284A JP2008500284A (ja) 2008-01-10
JP2008500284A5 true JP2008500284A5 (https=) 2008-02-21

Family

ID=35456856

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007513296A Pending JP2008500284A (ja) 2004-05-12 2005-05-11 血栓症の治療に有用なp2y1レセプターのウレアアンタゴニスト

Country Status (11)

Country Link
US (2) US7388021B2 (https=)
EP (1) EP1751113B1 (https=)
JP (1) JP2008500284A (https=)
KR (1) KR20070032648A (https=)
AT (1) ATE460402T1 (https=)
AU (1) AU2005245389A1 (https=)
DE (1) DE602005019874D1 (https=)
ES (1) ES2340179T3 (https=)
MX (1) MXPA06013022A (https=)
NO (1) NO20065534L (https=)
WO (1) WO2005113511A1 (https=)

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US8912184B1 (en) 2010-03-01 2014-12-16 Alzheimer's Institute Of America, Inc. Therapeutic and diagnostic methods
AU2011223790A1 (en) * 2010-03-01 2012-08-30 Myrexis, Inc. Compounds and therapeutic uses thereof
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US9540323B2 (en) * 2012-08-01 2017-01-10 Bristol-Myers Squibb Company 7-hydroxy-indolinyl antagonists of P2Y1 receptor
US9428504B2 (en) * 2012-08-01 2016-08-30 Bristol-Myers Squibb Company 7-hydroxy-spiropipiperidine indolinyl antagonists of P2Y1 receptor
EP2970114B1 (en) * 2013-03-15 2019-05-15 Bristol-Myers Squibb Company Ido inhibitors
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US7550499B2 (en) * 2004-05-12 2009-06-23 Bristol-Myers Squibb Company Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
WO2006078621A2 (en) * 2005-01-19 2006-07-27 Bristol-Myers Squibb Company 2-phenoxy-n- (1, 3 , 4-thiadizol-2-yl) pyridin-3-amine derivatives and related compounds as p2y1 receptor inhibitors for the treatment of thromboembolic disorders
ATE502924T1 (de) * 2005-06-27 2011-04-15 Bristol Myers Squibb Co Lineare harnstoffmimetika-antagonisten des p2y1- rezeptors zur behandlung von thromboseleiden
WO2007002634A1 (en) * 2005-06-27 2007-01-04 Bristol-Myers Squibb Company Carbocycle and heterocycle antagonists of p2y1 receptor useful in the treatment of thrombotic conditions

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