JP2007537258A - １７−ａａｇを含む医薬溶液製剤 - Google Patents
１７−ａａｇを含む医薬溶液製剤 Download PDFInfo
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- JP2007537258A JP2007537258A JP2007513239A JP2007513239A JP2007537258A JP 2007537258 A JP2007537258 A JP 2007537258A JP 2007513239 A JP2007513239 A JP 2007513239A JP 2007513239 A JP2007513239 A JP 2007513239A JP 2007537258 A JP2007537258 A JP 2007537258A
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- OGWKCGZFUXNPDA-UHFFFAOYSA-N vincristine Natural products C1C(CC)(O)CC(CC2(C(=O)OC)C=3C(=CC4=C(C56C(C(C(OC(C)=O)C7(CC)C=CCN(C67)CC5)(O)C(=O)OC)N4C=O)C=3)OC)CN1CCC1=C2NC2=CC=CC=C12 OGWKCGZFUXNPDA-UHFFFAOYSA-N 0.000 description 1
- OGWKCGZFUXNPDA-XQKSVPLYSA-N vincristine Chemical compound C([N@]1C[C@@H](C[C@]2(C(=O)OC)C=3C(=CC4=C([C@]56[C@H]([C@@]([C@H](OC(C)=O)[C@]7(CC)C=CCN([C@H]67)CC5)(O)C(=O)OC)N4C=O)C=3)OC)C[C@@](C1)(O)CC)CC1=C2NC2=CC=CC=C12 OGWKCGZFUXNPDA-XQKSVPLYSA-N 0.000 description 1
- 229960004355 vindesine Drugs 0.000 description 1
- UGGWPQSBPIFKDZ-KOTLKJBCSA-N vindesine Chemical compound C([C@@H](C[C@]1(C(=O)OC)C=2C(=CC3=C([C@]45[C@H]([C@@]([C@H](O)[C@]6(CC)C=CCN([C@H]56)CC4)(O)C(N)=O)N3C)C=2)OC)C[C@@](C2)(O)CC)N2CCC2=C1N=C1[C]2C=CC=C1 UGGWPQSBPIFKDZ-KOTLKJBCSA-N 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/20—Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US57021504P | 2004-05-11 | 2004-05-11 | |
| US11/123,570 US20050256097A1 (en) | 2004-05-11 | 2005-05-05 | Pharmaceutical solution formulations containing 17-AAG |
| PCT/US2005/016010 WO2005110398A2 (en) | 2004-05-11 | 2005-05-06 | Pharmaceutical solution formulations containing 17-aag |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2007537258A true JP2007537258A (ja) | 2007-12-20 |
| JP2007537258A5 JP2007537258A5 (https=) | 2008-06-19 |
Family
ID=35310196
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007513239A Abandoned JP2007537258A (ja) | 2004-05-11 | 2005-05-06 | １７−ａａｇを含む医薬溶液製剤 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20050256097A1 (https=) |
| EP (1) | EP1744743A2 (https=) |
| JP (1) | JP2007537258A (https=) |
| AU (1) | AU2005244115A1 (https=) |
| BR (1) | BRPI0511036A (https=) |
| CA (1) | CA2565583A1 (https=) |
| IL (1) | IL178689A0 (https=) |
| MX (1) | MXPA06012935A (https=) |
| RU (1) | RU2382643C2 (https=) |
| WO (1) | WO2005110398A2 (https=) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2018008922A (ja) * | 2015-08-04 | 2018-01-18 | わかもと製薬株式会社 | ステロイド白内障の予防及び治療 |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20090197852A9 (en) * | 2001-08-06 | 2009-08-06 | Johnson Robert G Jr | Method of treating breast cancer using 17-AAG or 17-AG or a prodrug of either in combination with a HER2 inhibitor |
| US8241670B2 (en) | 2004-04-15 | 2012-08-14 | Chiasma Inc. | Compositions capable of facilitating penetration across a biological barrier |
| EP1874296A4 (en) * | 2005-04-29 | 2010-06-30 | Kosan Biosciences Inc | METHOD FOR THE TREATMENT OF SEVERAL MYELOMES USING 17-AAG OR 17-AG OR PRODRUGS OR ALL |
| BRPI0609861A2 (pt) * | 2005-04-29 | 2010-05-11 | Kosan Biosciences Inc | uso de 17-aag ou 17-ag ou um pró-fármaco de ambos em combinação com um inibidor de proteassoma na preparação de formulações farmacêuticas para tratar mieloma múltiplo |
| US7648976B2 (en) * | 2005-11-23 | 2010-01-19 | Bristol-Myers Squibb Company | 17-allylamino-17-demethoxygeldanamycin polymorphs and formulations |
| US20090042847A1 (en) * | 2005-11-23 | 2009-02-12 | Kosan Biosciences Incorporated | 17-allylamino-17-demethoxygeldanamycin polymorphs and formulations |
| US20070167422A1 (en) * | 2006-01-18 | 2007-07-19 | Yu Kwok S | Pharmaceutical compositions comprising 17-allylamino-17-demethoxygeldanamycin |
| WO2008044041A1 (en) | 2006-10-12 | 2008-04-17 | Astex Therapeutics Limited | Pharmaceutical combinations |
| JP5528807B2 (ja) | 2006-10-12 | 2014-06-25 | アステックス、セラピューティックス、リミテッド | 複合薬剤 |
| WO2008055386A1 (fr) * | 2006-11-10 | 2008-05-15 | Shenzhen Shengeryimei Biotech Co., Ltd. | Composition pharmaceutique hydrosoluble pour injection de 17-allyl amino-17-déméthoxy geldanamycine (17-aag) |
| PE20081506A1 (es) * | 2006-12-12 | 2008-12-09 | Infinity Discovery Inc | Formulaciones de ansamicina |
| CN101688227B (zh) | 2007-01-26 | 2013-07-24 | 科森生物科学公司 | 通过工程化生物合成制备的大环内酰胺 |
| EP2180880A2 (en) * | 2007-07-09 | 2010-05-05 | Glen S. Kwon | Micelle encapsulation of therapeutic agents |
| NZ584275A (en) * | 2007-10-08 | 2012-06-29 | Fovea Pharmaceuticals | Aqueous cyclosporine ophthalmic formulations |
| US20090258869A1 (en) * | 2008-02-08 | 2009-10-15 | The Regents Of The University Of California | Methods and compounds for treatment or prevention of substance-related disorders |
| CN102176900B (zh) | 2008-09-17 | 2017-09-26 | 克艾思马有限公司 | 药物组合物和相关的给药方法 |
| US8236329B2 (en) | 2009-09-25 | 2012-08-07 | Wisconsin Alumni Research Foundation | Micelle encapsulation of therapeutic agents |
| NZ602392A (en) * | 2010-03-18 | 2014-03-28 | Innopharma Inc | Stable bortezomib formulations |
| WO2012151544A1 (en) | 2011-05-05 | 2012-11-08 | Wisconsin Alumni Research Foundation | Micelles for the solubilization of gossypol |
| US10682415B2 (en) | 2013-07-22 | 2020-06-16 | Wisconsin Alumni Research Foundation | Thermogel formulation for combination drug delivery |
| WO2016094831A1 (en) * | 2014-12-11 | 2016-06-16 | University Of Utah Research Foundation | Bi-functional allosteric protein-drug molecules for targeted therapy |
| HUE071943T2 (hu) | 2015-02-03 | 2025-10-28 | Amryt Endo Inc | Akromegália kezelése oktreotid orális alkalmazásával |
| US11141457B1 (en) | 2020-12-28 | 2021-10-12 | Amryt Endo, Inc. | Oral octreotide therapy and contraceptive methods |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US553153A (en) * | 1896-01-14 | Type-writing machine | ||
| US4261989A (en) * | 1979-02-19 | 1981-04-14 | Kaken Chemical Co. Ltd. | Geldanamycin derivatives and antitumor drug |
| US6262022B1 (en) * | 1992-06-25 | 2001-07-17 | Novartis Ag | Pharmaceutical compositions containing cyclosporin as the active agent |
| US5932556A (en) * | 1995-09-17 | 1999-08-03 | Tam; Robert C | Methods and compositions for regulation of CD28 expression |
| JP4713698B2 (ja) * | 1997-03-05 | 2011-06-29 | スージェン， インク． | 疎水性薬剤の処方 |
| US20030044434A1 (en) * | 1997-07-29 | 2003-03-06 | Ping Gao | Self-emulsifying formulation for lipophilic compounds |
| US6121323A (en) * | 1997-12-03 | 2000-09-19 | 3M Innovative Properties Company | Bishydroxyureas |
| US5925776A (en) * | 1997-12-24 | 1999-07-20 | Schein Pharmacetical, Inc. | Polyethoxylated castor oil, process of making the same and formulations thereof |
| US6682758B1 (en) * | 1998-12-22 | 2004-01-27 | The United States Of America As Represented By The Department Of Health And Human Services | Water-insoluble drug delivery system |
| AU773618B2 (en) * | 1998-12-22 | 2004-05-27 | United States Of America, Represented By The Secretary, Department Of Health And Human Services, The | Water-insoluble drug delivery system |
| TW471968B (en) * | 1999-08-25 | 2002-01-11 | Committee On Chinese Medicine | Solamargine pharmaceutical composition for killing cancer cells |
| US20020037855A1 (en) * | 2000-05-05 | 2002-03-28 | Fritz Stanislaus | Stabilized medicament containing cysteinyl derivatives |
| AU2001292548B2 (en) * | 2000-07-28 | 2005-06-16 | Sloan-Kettering Institute For Cancer Research | Methods for treating cell proliferative disorders and viral infections |
| NZ526169A (en) * | 2000-10-31 | 2005-12-23 | Boehringer Ingelheim Pharma | Oral dosage self-emulsifying formulations of pyranone protease inhibitors |
| US7025992B2 (en) * | 2001-02-14 | 2006-04-11 | Gw Pharma Limited | Pharmaceutical formulations |
| EP1373215B1 (en) * | 2001-03-30 | 2006-07-26 | THE UNITED STATES OF AMERICA, represented by THE SECRETARY, DEPT. OF HEALTH AND HUMAN SERVICES NATIONAL INSTITUTES OF HEALTH | Geldanamycin derivatives useful for treating cancer |
| WO2002092076A1 (en) * | 2001-05-16 | 2002-11-21 | Cytovia, Inc. | Substituted coumarins and quinolines as caspases activators |
| US6962944B2 (en) * | 2001-07-31 | 2005-11-08 | Arqule, Inc. | Pharmaceutical compositions containing beta-lapachone, or derivatives or analogs thereof, and methods of using same |
| US6872715B2 (en) * | 2001-08-06 | 2005-03-29 | Kosan Biosciences, Inc. | Benzoquinone ansamycins |
| US6653319B1 (en) * | 2001-08-10 | 2003-11-25 | University Of Kentucky Research Foundation | Pharmaceutical formulation for poorly water soluble camptothecin analogues |
| US8071133B2 (en) * | 2001-08-20 | 2011-12-06 | Stiefel Laboratories, Inc. | Oral dosage forms of water insoluble drugs and methods of making the same |
| HRP20040354B1 (en) * | 2001-10-19 | 2012-10-31 | Isotechnika Inc. | Novel cyclosporin analog microemulsion preconcentrates |
| EP1465592A2 (en) * | 2001-12-19 | 2004-10-13 | Alza Corporation | Formulation and dosage form for increasing oral bioavailability of hydrophilic macromolecules |
| US20030232078A1 (en) * | 2001-12-19 | 2003-12-18 | Dong Liang C. | Formulation & dosage form for the controlled delivery of therapeutic agents |
| US6803046B2 (en) * | 2002-08-16 | 2004-10-12 | Bracco International B.V. | Sincalide formulations |
| US7649006B2 (en) * | 2002-08-23 | 2010-01-19 | Sloan-Kettering Institute For Cancer Research | Synthesis of epothilones, intermediates thereto and analogues thereof |
-
2005
- 2005-05-05 US US11/123,570 patent/US20050256097A1/en not_active Abandoned
- 2005-05-06 CA CA002565583A patent/CA2565583A1/en not_active Abandoned
- 2005-05-06 AU AU2005244115A patent/AU2005244115A1/en not_active Abandoned
- 2005-05-06 BR BRPI0511036-0A patent/BRPI0511036A/pt not_active IP Right Cessation
- 2005-05-06 MX MXPA06012935A patent/MXPA06012935A/es active IP Right Grant
- 2005-05-06 RU RU2006143666/15A patent/RU2382643C2/ru not_active IP Right Cessation
- 2005-05-06 JP JP2007513239A patent/JP2007537258A/ja not_active Abandoned
- 2005-05-06 WO PCT/US2005/016010 patent/WO2005110398A2/en not_active Ceased
- 2005-05-06 EP EP05779076A patent/EP1744743A2/en not_active Withdrawn
-
2006
- 2006-10-17 IL IL178689A patent/IL178689A0/en unknown
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2018008922A (ja) * | 2015-08-04 | 2018-01-18 | わかもと製薬株式会社 | ステロイド白内障の予防及び治療 |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2005110398A2 (en) | 2005-11-24 |
| US20050256097A1 (en) | 2005-11-17 |
| CA2565583A1 (en) | 2005-11-24 |
| IL178689A0 (en) | 2007-02-11 |
| AU2005244115A1 (en) | 2005-11-24 |
| WO2005110398A3 (en) | 2006-05-04 |
| RU2006143666A (ru) | 2008-06-20 |
| BRPI0511036A (pt) | 2007-11-27 |
| MXPA06012935A (es) | 2007-01-26 |
| EP1744743A2 (en) | 2007-01-24 |
| RU2382643C2 (ru) | 2010-02-27 |
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