JP2007513070A5 - - Google Patents
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- Publication number
- JP2007513070A5 JP2007513070A5 JP2006538449A JP2006538449A JP2007513070A5 JP 2007513070 A5 JP2007513070 A5 JP 2007513070A5 JP 2006538449 A JP2006538449 A JP 2006538449A JP 2006538449 A JP2006538449 A JP 2006538449A JP 2007513070 A5 JP2007513070 A5 JP 2007513070A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- unsubstituted
- alkyl group
- halogen
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 0 *C1OC(CC([C@]23)=O)([C@]2*3(*)*2=CC2)O[C@@]1* Chemical compound *C1OC(CC([C@]23)=O)([C@]2*3(*)*2=CC2)O[C@@]1* 0.000 description 5
- AHMNPWKULMPFME-WHXUTIOJSA-N CC[O](C)C[C@H](CC1)C(CC2)C1C2=O Chemical compound CC[O](C)C[C@H](CC1)C(CC2)C1C2=O AHMNPWKULMPFME-WHXUTIOJSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US51839103P | 2003-11-07 | 2003-11-07 | |
| US60/518,391 | 2003-11-07 | ||
| PCT/US2004/036574 WO2005047215A2 (en) | 2003-11-07 | 2004-11-03 | Processes for preparing bicyclo [3.1.0] hexane derivatives, and intermediates thereto |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2007513070A JP2007513070A (ja) | 2007-05-24 |
| JP2007513070A5 true JP2007513070A5 (https=) | 2007-12-27 |
| JP4742239B2 JP4742239B2 (ja) | 2011-08-10 |
Family
ID=34590258
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006538449A Expired - Fee Related JP4742239B2 (ja) | 2003-11-07 | 2004-11-03 | ビシクロ［３．１．０］ヘキサン誘導体およびその中間体の製造方法 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US7786314B2 (https=) |
| EP (1) | EP1689727A4 (https=) |
| JP (1) | JP4742239B2 (https=) |
| KR (1) | KR101204145B1 (https=) |
| CN (2) | CN100475800C (https=) |
| AU (1) | AU2004289652B8 (https=) |
| CA (1) | CA2544560C (https=) |
| RU (1) | RU2388747C2 (https=) |
| TW (1) | TWI347316B (https=) |
| WO (1) | WO2005047215A2 (https=) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5309680B2 (ja) * | 2008-05-09 | 2013-10-09 | 大正製薬株式会社 | フッ素化エステル化合物の製造方法及びその中間体 |
| WO2009142184A1 (ja) | 2008-05-21 | 2009-11-26 | 大正製薬株式会社 | 酵素を用いたビシクロ［３．１．０］ヘキサン誘導体の製造方法 |
| TW201129700A (en) * | 2009-11-18 | 2011-09-01 | Taisho Pharmaceutical Co Ltd | Method for producing optically active bicyclo [310] hexane derivative using oxygen |
| BR112020018094A2 (pt) | 2018-03-08 | 2020-12-22 | Incyte Corporation | Compostos de aminopirazina diol como inibidores de pi3k-¿ |
| US11046658B2 (en) | 2018-07-02 | 2021-06-29 | Incyte Corporation | Aminopyrazine derivatives as PI3K-γ inhibitors |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5750566A (en) | 1994-08-12 | 1998-05-12 | Eli Lilly And Company | Synthetic excitatory amino acids |
| RU2152925C1 (ru) * | 1994-08-12 | 2000-07-20 | Эли Лилли Энд Компани | Производные аминобицикло[3.1.0]гексан-2,6-дикарбоновой кислоты и фармацевтическая композиция |
| ZA983930B (en) * | 1997-05-14 | 1999-11-08 | Lilly Co Eli | Excitatory amino acid receptor modulators. |
| JP4194715B2 (ja) * | 1998-08-31 | 2008-12-10 | 大正製薬株式会社 | ６−フルオロビシクロ［３．１．０］ヘキサン誘導体 |
| JP2000072731A (ja) * | 1998-08-31 | 2000-03-07 | Taisho Pharmaceut Co Ltd | ４−置換−２−アミノビシクロ［３．１．０］ヘキサン−２，６−ジカルボン酸誘導体及び製薬用組成物 |
| ATE269293T1 (de) | 1998-08-31 | 2004-07-15 | Taisho Pharmaceutical Co Ltd | 6-fluoro(3.1.0)hexan-derivate |
| PE20001236A1 (es) * | 1998-11-13 | 2000-11-10 | Lilly Co Eli | Moduladores del receptor de aminoacidos excitadores |
| CA2368454C (en) * | 1999-03-25 | 2009-11-24 | Taisho Pharmaceutical Co., Ltd. | Novel carboxylic acid derivatives and process for producing the same |
| AU2001267855B2 (en) | 2000-06-28 | 2005-09-08 | Taisho Pharmaceutical Co., Ltd. | Intermediate and process for producing fluorinated carboxylic acid derivative from the same |
| CA2441127A1 (en) * | 2001-03-14 | 2002-09-19 | Taisho Pharmaceutical Co., Ltd. | Process for producing bicyclocarboxylic acid derivative |
-
2004
- 2004-11-03 RU RU2006119924/04A patent/RU2388747C2/ru not_active IP Right Cessation
- 2004-11-03 CN CNB2004800381879A patent/CN100475800C/zh not_active Expired - Fee Related
- 2004-11-03 AU AU2004289652A patent/AU2004289652B8/en not_active Ceased
- 2004-11-03 KR KR1020067011065A patent/KR101204145B1/ko not_active Expired - Fee Related
- 2004-11-03 JP JP2006538449A patent/JP4742239B2/ja not_active Expired - Fee Related
- 2004-11-03 WO PCT/US2004/036574 patent/WO2005047215A2/en not_active Ceased
- 2004-11-03 CA CA2544560A patent/CA2544560C/en not_active Expired - Fee Related
- 2004-11-03 CN CN2009100086868A patent/CN101654410B/zh not_active Expired - Fee Related
- 2004-11-03 EP EP04800646A patent/EP1689727A4/en not_active Withdrawn
- 2004-11-03 US US10/578,476 patent/US7786314B2/en not_active Expired - Fee Related
- 2004-11-05 TW TW093133900A patent/TWI347316B/zh not_active IP Right Cessation