JP2007509058A5 - - Google Patents

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Publication number
JP2007509058A5
JP2007509058A5 JP2006535367A JP2006535367A JP2007509058A5 JP 2007509058 A5 JP2007509058 A5 JP 2007509058A5 JP 2006535367 A JP2006535367 A JP 2006535367A JP 2006535367 A JP2006535367 A JP 2006535367A JP 2007509058 A5 JP2007509058 A5 JP 2007509058A5
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JP
Japan
Prior art keywords
lower alkyl
cancer
compound
halo
hydrogen
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2006535367A
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English (en)
Japanese (ja)
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JP4755991B2 (ja
JP2007509058A (ja
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Priority claimed from PCT/US2004/034179 external-priority patent/WO2005037273A1/en
Publication of JP2007509058A publication Critical patent/JP2007509058A/ja
Publication of JP2007509058A5 publication Critical patent/JP2007509058A5/ja
Application granted granted Critical
Publication of JP4755991B2 publication Critical patent/JP4755991B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2006535367A 2003-10-16 2004-10-15 Ｒａｆキナーゼインヒビターとしての置換ベンゾアゾールおよびその使用 Expired - Fee Related JP4755991B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US51196603P 2003-10-16 2003-10-16
US60/511,966 2003-10-16
PCT/US2004/034179 WO2005037273A1 (en) 2003-10-16 2004-10-15 Substituted benzazoles and use thereof as inhibitors of raf kinase

Publications (3)

Publication Number Publication Date
JP2007509058A JP2007509058A (ja) 2007-04-12
JP2007509058A5 true JP2007509058A5 (enExample) 2007-11-15
JP4755991B2 JP4755991B2 (ja) 2011-08-24

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ID=34465300

Family Applications (1)

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JP2006535367A Expired - Fee Related JP4755991B2 (ja) 2003-10-16 2004-10-15 Ｒａｆキナーゼインヒビターとしての置換ベンゾアゾールおよびその使用

Country Status (16)

Country Link
US (3) US7423150B2 (enExample)
EP (1) EP1682126B1 (enExample)
JP (1) JP4755991B2 (enExample)
KR (1) KR20060118472A (enExample)
CN (1) CN1889951A (enExample)
AT (1) ATE435015T1 (enExample)
AU (1) AU2004281151A1 (enExample)
CA (1) CA2542653A1 (enExample)
DE (1) DE602004021838D1 (enExample)
ES (1) ES2327418T3 (enExample)
IL (1) IL174965A0 (enExample)
MX (1) MXPA06004236A (enExample)
PL (1) PL1682126T3 (enExample)
PT (1) PT1682126E (enExample)
TW (1) TW200526208A (enExample)
WO (1) WO2005037273A1 (enExample)

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JO3101B1 (ar) 2008-12-02 2017-09-20 Takeda Pharmaceuticals Co مشتقات بنزوثيازول كعوامل مضادة للسرطان
AU2011224410B2 (en) * 2010-03-09 2015-05-28 Dana-Farber Cancer Institute, Inc. Methods of diagnosing and treating cancer in patients having or developing resistance to a first cancer therapy
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US9408885B2 (en) 2011-12-01 2016-08-09 Vib Vzw Combinations of therapeutic agents for treating melanoma
BR112015001528B1 (pt) * 2012-07-28 2020-12-22 Calitor Sciences, Llc E Sunshine Lake Pharma Co., Ltd. composto, composição farmacêutica, e, uso de um composto ou de uma composição farmacêutica
US9242969B2 (en) 2013-03-14 2016-01-26 Novartis Ag Biaryl amide compounds as kinase inhibitors
UY36294A (es) 2014-09-12 2016-04-29 Novartis Ag Compuestos y composiciones como inhibidores de quinasa
WO2016100184A1 (en) 2014-12-16 2016-06-23 Forum Pharmaceuticals, Inc. Geminal substituted quinuclidine amide compounds as agonists of alpha-7 nicotinic acetylcholine receptors
CN105949178B (zh) * 2015-03-09 2020-05-26 西格莱(苏州)生物医药有限公司 一种苯并咪唑类化合物、其制备方法、中间体及应用
JP2018516973A (ja) 2015-06-10 2018-06-28 フォーラム・ファーマシューティカルズ・インコーポレイテッドＦｏｒｕｍ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃ． α７−ニコチン性アセチルコリン受容体のアゴニストとしてのアミノベンゾイソオキサゾール化合物
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