JP2007508347A5 - - Google Patents

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Publication number
JP2007508347A5
JP2007508347A5 JP2006534704A JP2006534704A JP2007508347A5 JP 2007508347 A5 JP2007508347 A5 JP 2007508347A5 JP 2006534704 A JP2006534704 A JP 2006534704A JP 2006534704 A JP2006534704 A JP 2006534704A JP 2007508347 A5 JP2007508347 A5 JP 2007508347A5
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JP
Japan
Prior art keywords
pro
ile
pyrrolidine
inhibitor
valinyl
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JP2006534704A
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English (en)
Japanese (ja)
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JP5707014B2 (ja
JP2007508347A (ja
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Priority claimed from PCT/EP2004/011630 external-priority patent/WO2005039548A2/en
Publication of JP2007508347A publication Critical patent/JP2007508347A/ja
Publication of JP2007508347A5 publication Critical patent/JP2007508347A5/ja
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Publication of JP5707014B2 publication Critical patent/JP5707014B2/ja
Anticipated expiration legal-status Critical
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JP2006534704A 2003-10-15 2004-10-15 グルタミニル、及びグルタミン酸シクラーゼのエフェクターの使用 Expired - Fee Related JP5707014B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US51203803P 2003-10-15 2003-10-15
US60/512,038 2003-10-15
PCT/EP2004/011630 WO2005039548A2 (en) 2003-10-15 2004-10-15 Use of effectors of glutaminyl and glutamate cyclases

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2014213807A Division JP2015057400A (ja) 2003-10-15 2014-10-20 グルタミニル、及びグルタミン酸シクラーゼのエフェクターの使用

Publications (3)

Publication Number Publication Date
JP2007508347A JP2007508347A (ja) 2007-04-05
JP2007508347A5 true JP2007508347A5 (enExample) 2007-12-06
JP5707014B2 JP5707014B2 (ja) 2015-04-22

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JP2006534704A Expired - Fee Related JP5707014B2 (ja) 2003-10-15 2004-10-15 グルタミニル、及びグルタミン酸シクラーゼのエフェクターの使用
JP2014213807A Withdrawn JP2015057400A (ja) 2003-10-15 2014-10-20 グルタミニル、及びグルタミン酸シクラーゼのエフェクターの使用

Family Applications After (1)

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JP2014213807A Withdrawn JP2015057400A (ja) 2003-10-15 2014-10-20 グルタミニル、及びグルタミン酸シクラーゼのエフェクターの使用

Country Status (14)

Country Link
US (2) US7462599B2 (enExample)
EP (2) EP1675578B9 (enExample)
JP (2) JP5707014B2 (enExample)
KR (3) KR101313975B1 (enExample)
CN (2) CN1867324A (enExample)
AU (1) AU2004283461B2 (enExample)
BR (1) BRPI0415409A (enExample)
CA (1) CA2542419C (enExample)
DK (1) DK1675578T3 (enExample)
EA (1) EA010108B1 (enExample)
IL (1) IL174372A (enExample)
MX (1) MXPA06003998A (enExample)
NZ (1) NZ546322A (enExample)
WO (1) WO2005039548A2 (enExample)

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JP5675343B2 (ja) 2007-04-18 2015-02-25 プロビオドルグ エージー グルタミニルシクラーゼ阻害剤としての尿素誘導体
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US8541596B2 (en) 2010-04-21 2013-09-24 Probiodrug Ag Inhibitors
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RU2766579C2 (ru) 2015-07-02 2022-03-15 ХОРАЙЗОН ОРФАН ЭлЭлСи Цистеаминдиоксигеназа-резистентные аналоги цистеамина и их применение
WO2019022600A1 (en) 2017-07-24 2019-01-31 Stichting Het Nederlands Kanker Instituut-Antoni van Leeuwenhoek Ziekenhuis TREATMENT OF PATHOLOGICAL CONDITIONS BY DIRECT AND INDIRECT TARGETING OF SIRPA INTERACTION - CD47
PL3461819T3 (pl) 2017-09-29 2020-11-30 Probiodrug Ag Inhibitory cyklazy glutaminylowej
CN112107568B (zh) * 2019-06-19 2022-03-25 北京龙嘉博创医药科技有限公司 二芳基酰胺类化合物及其应用
CN112816581A (zh) * 2020-12-30 2021-05-18 浙江大学 衍生化-固相萃取-液相色谱串联质谱检测饮用水中卤代醌亚胺的方法
CN112898286A (zh) * 2021-01-28 2021-06-04 中国药科大学 苯并噻吩类化合物或其可药用的盐、异构体及其制备方法、药物组合物和用途
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JP2005523288A (ja) 2002-02-19 2005-08-04 ファルマシア・アンド・アップジョン・カンパニー・エルエルシー 疾病治療用の縮合した二環式−ｎ−架橋−複素環式芳香族カルボキサミド
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PL1620082T3 (pl) * 2003-05-05 2010-10-29 Probiodrug Ag Medyczne zastosowanie inhibitorów cyklazy glutaminylowej i glutaminianowej do leczenia choroby Alzheimera i zespołu Downa
US7732162B2 (en) * 2003-05-05 2010-06-08 Probiodrug Ag Inhibitors of glutaminyl cyclase for treating neurodegenerative diseases
KR20060009902A (ko) * 2003-05-05 2006-02-01 프로비오드룩 아게 글루타미닐 및 글루타메이트 사이클라제의 이펙터의 용도
AU2004283461B2 (en) 2003-10-15 2010-02-11 Probiodrug Ag Use of effectors of glutaminyl and glutamate cyclases
WO2005059100A2 (en) * 2003-12-12 2005-06-30 New York University Methods and compositions relating to cystatin c
GB0704100D0 (en) 2006-03-17 2007-04-11 Vodafone Plc Improvements in an ehspa architecture

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