JP2006508161A5 - - Google Patents

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Publication number
JP2006508161A5
JP2006508161A5 JP2004556337A JP2004556337A JP2006508161A5 JP 2006508161 A5 JP2006508161 A5 JP 2006508161A5 JP 2004556337 A JP2004556337 A JP 2004556337A JP 2004556337 A JP2004556337 A JP 2004556337A JP 2006508161 A5 JP2006508161 A5 JP 2006508161A5
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JP
Japan
Prior art keywords
alkyl
formula
group
aryl
optionally substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2004556337A
Other languages
English (en)
Japanese (ja)
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JP2006508161A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/EP2003/050902 external-priority patent/WO2004050585A1/en
Publication of JP2006508161A publication Critical patent/JP2006508161A/ja
Publication of JP2006508161A5 publication Critical patent/JP2006508161A5/ja
Pending legal-status Critical Current

Links

JP2004556337A 2002-12-02 2003-11-27 炭素−ヘテロ原子二重結合の接触水素化 Pending JP2006508161A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH20332002 2002-12-02
PCT/EP2003/050902 WO2004050585A1 (en) 2002-12-02 2003-11-27 Catalytic hydrogeneration of carbon-heteroatom double bonds

Publications (2)

Publication Number Publication Date
JP2006508161A JP2006508161A (ja) 2006-03-09
JP2006508161A5 true JP2006508161A5 (enExample) 2006-11-02

Family

ID=32399972

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2004556337A Pending JP2006508161A (ja) 2002-12-02 2003-11-27 炭素−ヘテロ原子二重結合の接触水素化

Country Status (10)

Country Link
US (1) US7446236B2 (enExample)
EP (1) EP1567464B1 (enExample)
JP (1) JP2006508161A (enExample)
CN (1) CN100384791C (enExample)
AT (1) ATE359986T1 (enExample)
AU (1) AU2003298328A1 (enExample)
CA (1) CA2507908A1 (enExample)
DE (1) DE60313357T2 (enExample)
ES (1) ES2283867T3 (enExample)
WO (1) WO2004050585A1 (enExample)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005058894A1 (en) 2003-12-19 2005-06-30 Altana Pharma Ag Intermediates for the preparation of tricyclic dihydropyrano -imidazo -pyridines derivatives
US7767657B2 (en) 2005-02-16 2010-08-03 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
ES2872962T3 (es) 2005-02-16 2021-11-03 Anacor Pharmaceuticals Inc Boronoftalidas para uso terapéutico
RU2642628C2 (ru) 2006-02-16 2018-01-25 Анакор Фармасьютикалз, Инк. Бор-содержащие малые молекулы в качестве противовоспалительных средств
CA2645107A1 (en) * 2006-03-10 2007-09-20 Solvias Ag Asymmetric catalytic hydrogenation of prochiral ketones and aldehydes
EP3246034A1 (en) 2008-03-06 2017-11-22 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-inflammatory agents
WO2010027975A1 (en) 2008-09-04 2010-03-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
US8461336B2 (en) * 2008-09-04 2013-06-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
ES2863542T3 (es) * 2009-03-17 2021-10-11 Johnson Matthey Plc Proceso para la hidrogenación de cetonas en presencia de catalizadores de Ru (II)
AP4039A (en) * 2009-08-14 2017-02-28 Daitao Chen Boron-containing small molecules as antiprotozoal agents
WO2011049971A1 (en) 2009-10-20 2011-04-28 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
US8461134B2 (en) * 2009-11-11 2013-06-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
US8716478B2 (en) 2010-01-27 2014-05-06 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2011116348A1 (en) 2010-03-19 2011-09-22 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agent
AU2011237681B2 (en) * 2010-04-07 2015-01-22 Glaxosmithkline Llc Process for preparing benzoxaboroles
DK2613788T3 (en) 2010-09-07 2017-08-07 Anacor Pharmaceuticals Inc BENZOXABOROLD DERIVATIVES FOR TREATMENT OF BACTERIA INFECTIONS
US20160251380A1 (en) 2013-08-09 2016-09-01 Glaxosmithkline Intellectual Property (No.2) Limited Tricyclic benzoxaborole compounds and uses thereof
GB201401230D0 (en) * 2014-01-24 2014-03-12 Givaudan Sa Improvements in or relating to organic compounds
MA41495A (fr) 2015-02-12 2017-12-19 Anacor Pharmaceuticals Inc Composés benzoxaborole et leurs utilisations

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2693190B1 (fr) * 1992-07-02 1994-09-23 Elf Aquitaine Procédé d'hydrogénation énantiosélectif de la double liaison C=O OXO.
US6476233B1 (en) * 1998-11-12 2002-11-05 The Penn State Research Foundation Transition metal-catalyzed reactions based on chiral amine oxazolinyl ligands and related compounds
NL1015655C2 (nl) * 2000-07-07 2002-01-08 Dsm Nv Katalysator voor de asymmetrische hydrogenering.
ES2305095T3 (es) 2000-09-13 2008-11-01 Firmenich S.A. Procesos de hidrogenacion catalitica.

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