CN100384791C - 碳-杂原子双键的催化氢化 - Google Patents

碳-杂原子双键的催化氢化 Download PDF

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Publication number
CN100384791C
CN100384791C CNB2003801045565A CN200380104556A CN100384791C CN 100384791 C CN100384791 C CN 100384791C CN B2003801045565 A CNB2003801045565 A CN B2003801045565A CN 200380104556 A CN200380104556 A CN 200380104556A CN 100384791 C CN100384791 C CN 100384791C
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CN1717376A (zh
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F·M·诺德
U·皮特尔科夫
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Solvias AG
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Solvias AG
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B41/00—Formation or introduction of functional groups containing oxygen
    • C07B41/02—Formation or introduction of functional groups containing oxygen of hydroxy or O-metal groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B43/00—Formation or introduction of functional groups containing nitrogen
    • C07B43/04—Formation or introduction of functional groups containing nitrogen of amino groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B53/00—Asymmetric syntheses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/16—Radicals substituted by singly bound hetero atoms other than halogen by oxygen atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Production Of Liquid Hydrocarbon Mixture For Refining Petroleum (AREA)
CNB2003801045565A 2002-12-02 2003-11-27 碳-杂原子双键的催化氢化 Expired - Lifetime CN100384791C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH2033/02 2002-12-02
CH20332002 2002-12-02

Publications (2)

Publication Number Publication Date
CN1717376A CN1717376A (zh) 2006-01-04
CN100384791C true CN100384791C (zh) 2008-04-30

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ID=32399972

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CNB2003801045565A Expired - Lifetime CN100384791C (zh) 2002-12-02 2003-11-27 碳-杂原子双键的催化氢化

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US (1) US7446236B2 (enExample)
EP (1) EP1567464B1 (enExample)
JP (1) JP2006508161A (enExample)
CN (1) CN100384791C (enExample)
AT (1) ATE359986T1 (enExample)
AU (1) AU2003298328A1 (enExample)
CA (1) CA2507908A1 (enExample)
DE (1) DE60313357T2 (enExample)
ES (1) ES2283867T3 (enExample)
WO (1) WO2004050585A1 (enExample)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7326784B2 (en) 2003-12-19 2008-02-05 Altana Pharma Ag Intermediates for the preparation of tricyclic dihydropyrano-imidazo-pyridines derivatives
US7767657B2 (en) 2005-02-16 2010-08-03 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
JP5038912B2 (ja) 2005-02-16 2012-10-03 アナコール ファーマシューティカルズ，インコーポレイテッド ホウ素含有小分子
NZ570257A (en) 2006-02-16 2011-11-25 Anacor Pharmaceuticals Inc Boron-containing small molecules as anti-inflammatory agents
CA2645107A1 (en) * 2006-03-10 2007-09-20 Solvias Ag Asymmetric catalytic hydrogenation of prochiral ketones and aldehydes
BRPI0908565A2 (pt) 2008-03-06 2017-05-23 Anacor Pharmaceuticals Inc composto, formulação farmacêutica, métodos para reduzir a liberação de uma citocina ou de uma quimiocina, para tratar uma condição em um animal e para inibir uma fosfodiesterase
EP2348863A4 (en) 2008-09-04 2012-03-07 Anacor Pharmaceuticals Inc BORN SMALL MOLECULES
US8461336B2 (en) * 2008-09-04 2013-06-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
US9416100B2 (en) * 2009-03-17 2016-08-16 Johnson Matthey Public Limited Company Process for hydrogenating ketones in the presence of Ru(II) catalysts
AP4039A (en) 2009-08-14 2017-02-28 Daitao Chen Boron-containing small molecules as antiprotozoal agents
WO2011049971A1 (en) 2009-10-20 2011-04-28 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
US20110212918A1 (en) * 2009-11-11 2011-09-01 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2011094450A1 (en) 2010-01-27 2011-08-04 Anacor Pharmaceuticals, Inc Boron-containing small molecules
AP2012006482A0 (en) 2010-03-19 2012-10-31 Anacor Pharmacueticals Inc Boron-containing small molecules as anti-protozoalagent
JP5603998B2 (ja) * 2010-04-07 2014-10-08 グラクソスミスクライン エルエルシー ベンゾオキサボロールの調製方法
SG10201507032YA (en) 2010-09-07 2015-10-29 Anacor Pharmaceuticals Inc Benzoxaborole derivatives for treating bacterial infections
CN105492388B (zh) 2013-08-09 2018-12-21 葛兰素史克知识产权第二有限公司 三环苯并氧杂硼杂环戊烯化合物及其用途
GB201401230D0 (en) * 2014-01-24 2014-03-12 Givaudan Sa Improvements in or relating to organic compounds
MA41495A (fr) 2015-02-12 2017-12-19 Anacor Pharmaceuticals Inc Composés benzoxaborole et leurs utilisations

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002004466A2 (en) * 2000-07-07 2002-01-17 Dsm N.V. Catalyst for asymmetric (transfer) hydrogenation
WO2002022526A2 (en) * 2000-09-13 2002-03-21 Firmenich S.A. Catalytic hydrogenation processes

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2693190B1 (fr) * 1992-07-02 1994-09-23 Elf Aquitaine Procédé d'hydrogénation énantiosélectif de la double liaison C=O OXO.
US6476233B1 (en) * 1998-11-12 2002-11-05 The Penn State Research Foundation Transition metal-catalyzed reactions based on chiral amine oxazolinyl ligands and related compounds

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002004466A2 (en) * 2000-07-07 2002-01-17 Dsm N.V. Catalyst for asymmetric (transfer) hydrogenation
WO2002022526A2 (en) * 2000-09-13 2002-03-21 Firmenich S.A. Catalytic hydrogenation processes

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
extremely high enantioselectvie redox reaction of ketones ansalcohols catalyzed by RuCl2(PPh3)3(oxazolinylferrocenylphosphine). Yoshiaki Nishibayashi et al.Organometallics,Vol.18 . 1999 *
Ruthenium(II)-catalyzed asymmetric transfer hydrogention ofketones using chiral oxazolinylferrocenylphosphines and oneof their Ru(II) complex. Yasuyoshi Arikawa et al.Journal of Organometallic Chemistry,Vol.572 No.2. 1999 *

Also Published As

Publication number Publication date
DE60313357D1 (de) 2007-05-31
EP1567464A1 (en) 2005-08-31
ES2283867T3 (es) 2007-11-01
DE60313357T2 (de) 2008-01-03
ATE359986T1 (de) 2007-05-15
CA2507908A1 (en) 2004-06-17
US20060106247A1 (en) 2006-05-18
EP1567464B1 (en) 2007-04-18
AU2003298328A1 (en) 2004-06-23
CN1717376A (zh) 2006-01-04
JP2006508161A (ja) 2006-03-09
US7446236B2 (en) 2008-11-04
WO2004050585A1 (en) 2004-06-17

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