JP2006508161A - 炭素−ヘテロ原子二重結合の接触水素化 - Google Patents
炭素−ヘテロ原子二重結合の接触水素化 Download PDFInfo
- Publication number
- JP2006508161A JP2006508161A JP2004556337A JP2004556337A JP2006508161A JP 2006508161 A JP2006508161 A JP 2006508161A JP 2004556337 A JP2004556337 A JP 2004556337A JP 2004556337 A JP2004556337 A JP 2004556337A JP 2006508161 A JP2006508161 A JP 2006508161A
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- group
- formula
- aryl
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 0 CC(CCC(C)C(C(C)(C)C1)C11C=*C(C)C2C1C2)C1CC1 Chemical compound CC(CCC(C)C(C(C)(C)C1)C11C=*C(C)C2C1C2)C1CC1 0.000 description 3
- KRAKYLMUCDNEGV-ARJAWSKDSA-N C/C=C\CCC=[N]=C Chemical compound C/C=C\CCC=[N]=C KRAKYLMUCDNEGV-ARJAWSKDSA-N 0.000 description 1
- KIYZXQSCKFYJAH-VCJLRHCSSA-N CC(C)C1=[N]=C([C@@](C2)(C2CC2)C2P)OC1 Chemical compound CC(C)C1=[N]=C([C@@](C2)(C2CC2)C2P)OC1 KIYZXQSCKFYJAH-VCJLRHCSSA-N 0.000 description 1
- QELBUFHMTAOBRH-HSOILSAZSA-N CC(C)C1N=C([C@H]2C(C)CCC2)OC1 Chemical compound CC(C)C1N=C([C@H]2C(C)CCC2)OC1 QELBUFHMTAOBRH-HSOILSAZSA-N 0.000 description 1
- RKOBLTQPGMADLU-ORFBVSJDSA-N CC(C)[C@H]1N=C(C(CCC2)C2P(c2ccccc2)c2ccccc2)OC1 Chemical compound CC(C)[C@H]1N=C(C(CCC2)C2P(c2ccccc2)c2ccccc2)OC1 RKOBLTQPGMADLU-ORFBVSJDSA-N 0.000 description 1
- NFWSQSCIDYBUOU-UHFFFAOYSA-N CC1=CC=CC1 Chemical compound CC1=CC=CC1 NFWSQSCIDYBUOU-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B41/00—Formation or introduction of functional groups containing oxygen
- C07B41/02—Formation or introduction of functional groups containing oxygen of hydroxy or O-metal groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B43/00—Formation or introduction of functional groups containing nitrogen
- C07B43/04—Formation or introduction of functional groups containing nitrogen of amino groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B53/00—Asymmetric syntheses
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
- C07D333/16—Radicals substituted by singly bound hetero atoms other than halogen by oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Catalysts (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Production Of Liquid Hydrocarbon Mixture For Refining Petroleum (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH20332002 | 2002-12-02 | ||
| PCT/EP2003/050902 WO2004050585A1 (en) | 2002-12-02 | 2003-11-27 | Catalytic hydrogeneration of carbon-heteroatom double bonds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2006508161A true JP2006508161A (ja) | 2006-03-09 |
| JP2006508161A5 JP2006508161A5 (enExample) | 2006-11-02 |
Family
ID=32399972
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004556337A Pending JP2006508161A (ja) | 2002-12-02 | 2003-11-27 | 炭素−ヘテロ原子二重結合の接触水素化 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US7446236B2 (enExample) |
| EP (1) | EP1567464B1 (enExample) |
| JP (1) | JP2006508161A (enExample) |
| CN (1) | CN100384791C (enExample) |
| AT (1) | ATE359986T1 (enExample) |
| AU (1) | AU2003298328A1 (enExample) |
| CA (1) | CA2507908A1 (enExample) |
| DE (1) | DE60313357T2 (enExample) |
| ES (1) | ES2283867T3 (enExample) |
| WO (1) | WO2004050585A1 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2017507924A (ja) * | 2014-01-24 | 2017-03-23 | ジボダン エス エー | 有機化合物における、または有機化合物に関する改良 |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7326784B2 (en) | 2003-12-19 | 2008-02-05 | Altana Pharma Ag | Intermediates for the preparation of tricyclic dihydropyrano-imidazo-pyridines derivatives |
| US7767657B2 (en) | 2005-02-16 | 2010-08-03 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| JP5038912B2 (ja) | 2005-02-16 | 2012-10-03 | アナコール ファーマシューティカルズ,インコーポレイテッド | ホウ素含有小分子 |
| NZ570257A (en) | 2006-02-16 | 2011-11-25 | Anacor Pharmaceuticals Inc | Boron-containing small molecules as anti-inflammatory agents |
| CA2645107A1 (en) * | 2006-03-10 | 2007-09-20 | Solvias Ag | Asymmetric catalytic hydrogenation of prochiral ketones and aldehydes |
| BRPI0908565A2 (pt) | 2008-03-06 | 2017-05-23 | Anacor Pharmaceuticals Inc | composto, formulação farmacêutica, métodos para reduzir a liberação de uma citocina ou de uma quimiocina, para tratar uma condição em um animal e para inibir uma fosfodiesterase |
| EP2348863A4 (en) | 2008-09-04 | 2012-03-07 | Anacor Pharmaceuticals Inc | BORN SMALL MOLECULES |
| US8461336B2 (en) * | 2008-09-04 | 2013-06-11 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| US9416100B2 (en) * | 2009-03-17 | 2016-08-16 | Johnson Matthey Public Limited Company | Process for hydrogenating ketones in the presence of Ru(II) catalysts |
| AP4039A (en) | 2009-08-14 | 2017-02-28 | Daitao Chen | Boron-containing small molecules as antiprotozoal agents |
| WO2011049971A1 (en) | 2009-10-20 | 2011-04-28 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules as antiprotozoal agents |
| US20110212918A1 (en) * | 2009-11-11 | 2011-09-01 | Anacor Pharmaceuticals, Inc. | Boron-containing small molecules |
| WO2011094450A1 (en) | 2010-01-27 | 2011-08-04 | Anacor Pharmaceuticals, Inc | Boron-containing small molecules |
| AP2012006482A0 (en) | 2010-03-19 | 2012-10-31 | Anacor Pharmacueticals Inc | Boron-containing small molecules as anti-protozoalagent |
| JP5603998B2 (ja) * | 2010-04-07 | 2014-10-08 | グラクソスミスクライン エルエルシー | ベンゾオキサボロールの調製方法 |
| SG10201507032YA (en) | 2010-09-07 | 2015-10-29 | Anacor Pharmaceuticals Inc | Benzoxaborole derivatives for treating bacterial infections |
| CN105492388B (zh) | 2013-08-09 | 2018-12-21 | 葛兰素史克知识产权第二有限公司 | 三环苯并氧杂硼杂环戊烯化合物及其用途 |
| MA41495A (fr) | 2015-02-12 | 2017-12-19 | Anacor Pharmaceuticals Inc | Composés benzoxaborole et leurs utilisations |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2002004466A2 (en) * | 2000-07-07 | 2002-01-17 | Dsm N.V. | Catalyst for asymmetric (transfer) hydrogenation |
| WO2002022526A2 (en) * | 2000-09-13 | 2002-03-21 | Firmenich S.A. | Catalytic hydrogenation processes |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2693190B1 (fr) * | 1992-07-02 | 1994-09-23 | Elf Aquitaine | Procédé d'hydrogénation énantiosélectif de la double liaison C=O OXO. |
| US6476233B1 (en) * | 1998-11-12 | 2002-11-05 | The Penn State Research Foundation | Transition metal-catalyzed reactions based on chiral amine oxazolinyl ligands and related compounds |
-
2003
- 2003-11-27 CA CA002507908A patent/CA2507908A1/en not_active Abandoned
- 2003-11-27 CN CNB2003801045565A patent/CN100384791C/zh not_active Expired - Lifetime
- 2003-11-27 DE DE60313357T patent/DE60313357T2/de not_active Expired - Lifetime
- 2003-11-27 EP EP03796062A patent/EP1567464B1/en not_active Expired - Lifetime
- 2003-11-27 AU AU2003298328A patent/AU2003298328A1/en not_active Abandoned
- 2003-11-27 US US10/536,883 patent/US7446236B2/en not_active Expired - Lifetime
- 2003-11-27 AT AT03796062T patent/ATE359986T1/de not_active IP Right Cessation
- 2003-11-27 WO PCT/EP2003/050902 patent/WO2004050585A1/en not_active Ceased
- 2003-11-27 JP JP2004556337A patent/JP2006508161A/ja active Pending
- 2003-11-27 ES ES03796062T patent/ES2283867T3/es not_active Expired - Lifetime
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2002004466A2 (en) * | 2000-07-07 | 2002-01-17 | Dsm N.V. | Catalyst for asymmetric (transfer) hydrogenation |
| WO2002022526A2 (en) * | 2000-09-13 | 2002-03-21 | Firmenich S.A. | Catalytic hydrogenation processes |
Non-Patent Citations (3)
| Title |
|---|
| ACC. CHEM. RES., vol. 33, JPN6010011795, 2000, pages 336 - 345, ISSN: 0001555915 * |
| JOURNAL OF ORGANOMETALLIC CHEMISTRY, vol. 572, JPN6010011797, 1999, pages 163 - 168, ISSN: 0001555914 * |
| ORGANOMETALLICS, vol. 18, JPN6010011799, 1999, pages 2291 - 2293, ISSN: 0001555913 * |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2017507924A (ja) * | 2014-01-24 | 2017-03-23 | ジボダン エス エー | 有機化合物における、または有機化合物に関する改良 |
Also Published As
| Publication number | Publication date |
|---|---|
| DE60313357D1 (de) | 2007-05-31 |
| EP1567464A1 (en) | 2005-08-31 |
| ES2283867T3 (es) | 2007-11-01 |
| DE60313357T2 (de) | 2008-01-03 |
| ATE359986T1 (de) | 2007-05-15 |
| CA2507908A1 (en) | 2004-06-17 |
| US20060106247A1 (en) | 2006-05-18 |
| EP1567464B1 (en) | 2007-04-18 |
| CN100384791C (zh) | 2008-04-30 |
| AU2003298328A1 (en) | 2004-06-23 |
| CN1717376A (zh) | 2006-01-04 |
| US7446236B2 (en) | 2008-11-04 |
| WO2004050585A1 (en) | 2004-06-17 |
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