JP2005539045A5 - - Google Patents

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Publication number
JP2005539045A5
JP2005539045A5 JP2004532233A JP2004532233A JP2005539045A5 JP 2005539045 A5 JP2005539045 A5 JP 2005539045A5 JP 2004532233 A JP2004532233 A JP 2004532233A JP 2004532233 A JP2004532233 A JP 2004532233A JP 2005539045 A5 JP2005539045 A5 JP 2005539045A5
Authority
JP
Japan
Prior art keywords
dioxan
propylcarbamate
trans
general formula
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2004532233A
Other languages
English (en)
Japanese (ja)
Other versions
JP4585854B2 (ja
JP2005539045A (ja
Filing date
Publication date
Priority claimed from FR0210707A external-priority patent/FR2843964B1/fr
Application filed filed Critical
Publication of JP2005539045A publication Critical patent/JP2005539045A/ja
Publication of JP2005539045A5 publication Critical patent/JP2005539045A5/ja
Application granted granted Critical
Publication of JP4585854B2 publication Critical patent/JP4585854B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

JP2004532233A 2002-08-29 2003-08-27 ジオキサン−2−アルキルカルバメート誘導体、その製造法および治療における適用 Expired - Fee Related JP4585854B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0210707A FR2843964B1 (fr) 2002-08-29 2002-08-29 Derives de dioxane-2-alkylcarbamates, leur preparation et leur application en therapeutique
PCT/FR2003/002590 WO2004020430A2 (fr) 2002-08-29 2003-08-27 Derives de dioxane-2-alkylcarbamates, leur preparation et leur application en therapeutique

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2010139427A Division JP5244863B2 (ja) 2002-08-29 2010-06-18 ジオキサン−2−アルキルカルバメート誘導体の製造法およびその中間体

Publications (3)

Publication Number Publication Date
JP2005539045A JP2005539045A (ja) 2005-12-22
JP2005539045A5 true JP2005539045A5 (https=) 2006-10-05
JP4585854B2 JP4585854B2 (ja) 2010-11-24

Family

ID=31502974

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2004532233A Expired - Fee Related JP4585854B2 (ja) 2002-08-29 2003-08-27 ジオキサン−2−アルキルカルバメート誘導体、その製造法および治療における適用
JP2010139427A Expired - Fee Related JP5244863B2 (ja) 2002-08-29 2010-06-18 ジオキサン−2−アルキルカルバメート誘導体の製造法およびその中間体

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2010139427A Expired - Fee Related JP5244863B2 (ja) 2002-08-29 2010-06-18 ジオキサン−2−アルキルカルバメート誘導体の製造法およびその中間体

Country Status (34)

Country Link
US (4) US7119116B2 (https=)
EP (2) EP1840125B1 (https=)
JP (2) JP4585854B2 (https=)
KR (2) KR101139160B1 (https=)
CN (3) CN101906071A (https=)
AR (1) AR041053A1 (https=)
AT (2) ATE409184T1 (https=)
AU (1) AU2003274292B2 (https=)
BR (1) BR0313846A (https=)
CA (2) CA2700319C (https=)
CO (1) CO5700820A2 (https=)
CY (2) CY1108792T1 (https=)
DE (2) DE60323754D1 (https=)
DK (2) DK1537096T3 (https=)
EA (1) EA008218B1 (https=)
ES (2) ES2312808T3 (https=)
FR (1) FR2843964B1 (https=)
HR (2) HRP20090270B1 (https=)
IL (1) IL166882A (https=)
IS (1) IS2733B (https=)
MA (1) MA27390A1 (https=)
ME (2) MEP24208A (https=)
MX (1) MXPA05002319A (https=)
NO (2) NO331165B1 (https=)
NZ (1) NZ538404A (https=)
PL (1) PL209339B1 (https=)
PT (2) PT1537096E (https=)
RS (2) RS51085B (https=)
SI (2) SI1537096T1 (https=)
TN (1) TNSN05057A1 (https=)
TW (2) TWI294878B (https=)
UA (1) UA82847C2 (https=)
WO (1) WO2004020430A2 (https=)
ZA (1) ZA200501537B (https=)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2843964B1 (fr) * 2002-08-29 2004-10-01 Sanofi Synthelabo Derives de dioxane-2-alkylcarbamates, leur preparation et leur application en therapeutique
EP1558591B1 (en) * 2002-10-07 2014-05-07 The Regents of The University of California Modulation of anxiety through blockade of anandamide hydrolysis
FR2854633B1 (fr) * 2003-05-07 2005-06-24 Sanofi Synthelabo Derives de piperidinyl-et piperazinyl-alkylcarbamates, leur preparation et leur application en therapeutique
FR2865205B1 (fr) * 2004-01-16 2006-02-24 Sanofi Synthelabo Derives de type aryloxyalkylcarbamates, leur preparation et leur application en therapeutique
FR2866886B1 (fr) * 2004-02-26 2007-08-31 Sanofi Synthelabo Derives d'aryl-et d'heteroaryl-akylcarbamates, leur preparation et leur application en therapeutique
FR2866884B1 (fr) * 2004-02-26 2007-08-31 Sanofi Synthelabo Derives d'aryl-et d'heteroaryl-piperidinecarboxylates, leur preparation et leur application en therapeutique
FR2866888B1 (fr) * 2004-02-26 2006-05-05 Sanofi Synthelabo Derives de alkylpiperazine- et alkylhomopiperazine- carboxylates, leur preparation et leur application en therapeutique
FR2866885B1 (fr) 2004-02-26 2007-08-31 Sanofi Synthelabo Derives de piperidinylalkylcarbamates, leur prepation et leur application en therapeutique
US7269708B2 (en) * 2004-04-20 2007-09-11 Rambus Inc. Memory controller for non-homogenous memory system
US20080103209A1 (en) * 2004-04-23 2008-05-01 The Regents Of The University Of California Compounds And Methods For Treating Non-Inflammatory Pain Using Ppar Alpha Agonists
DE102004039326A1 (de) * 2004-08-12 2006-02-16 Abbott Gmbh & Co. Kg Neue medizinische Verwendungen und Verfahren
ES2528674T3 (es) 2005-02-17 2015-02-11 Astellas Pharma Inc. Piperidina y carboxilatos de piperacina como inhibidores de FAAH
FR2885364B1 (fr) * 2005-05-03 2007-06-29 Sanofi Aventis Sa Derives d'alkyl-, alkenyl-et alkynylcarbamates, leur preparation et leur application en therapeutique
WO2008021625A2 (en) * 2006-08-18 2008-02-21 N.V. Organon Combination faah inhibitor and analgesic, anti-inflammatory or anti-pyretic agent
WO2008030752A2 (en) * 2006-09-07 2008-03-13 N.V. Organon Methods for determining effective doses of fatty acid amide hydrolase inhibitors in vivo
US20090099240A1 (en) * 2006-10-02 2009-04-16 N.V. Organon Methods for treating energy metabolism disorders by inhibiting fatty acid amide hydrolase activity
US20080119549A1 (en) * 2006-11-20 2008-05-22 N.V. Organon Metabolically-stabilized inhibitors of fatty acid amide hydrolase
US8207226B1 (en) 2008-06-03 2012-06-26 Alcon Research, Ltd. Use of FAAH antagonists for treating dry eye and ocular pain
FR2941696B1 (fr) * 2009-02-05 2011-04-15 Sanofi Aventis Derives d'azaspiranyl-alkylcarbamates d'heterocycles a 5 chainons, leur preparation et leur application en therapeutique
TW201044234A (en) * 2009-06-08 2010-12-16 Chunghwa Picture Tubes Ltd Method of scanning touch panel
ES2626246T3 (es) 2009-09-09 2017-07-24 Sumitomo Dainippon Pharma Co., Ltd. Derivado de 8-oxodihidropurina
US8274566B2 (en) * 2009-10-09 2012-09-25 John Mezzalingua Associates, Inc. Modulation analyzer and level measurement device
EP2545914A1 (en) 2011-07-11 2013-01-16 Sanofi 2-amino-2-oxoethyl trans-3-[5-(6-methoxy-naphtalen-1-yl)-1,3-dioxan-2-yl]propyl-carbamate for use in the treatment of persistent cancer pain
EP2545915A1 (en) 2011-07-11 2013-01-16 Sanofi 2-amino-2-oxoethyl trans-3-[5-(6-methoxy-naphtalen-1-yl)-1,3-dioxan-2-yl]propyl-carbamate for use in the treatment of persistent cancer pain
PE20141702A1 (es) * 2012-01-06 2014-11-19 Abide Therapeutics Inc Compuestos de carbamato y preparacion y uso de los mismos
CN114835726B (zh) * 2022-03-24 2024-01-26 上海诺精生物科技有限公司 一类抑制肿瘤细胞干性的化合物及用途

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK0461958T3 (da) * 1990-06-15 1995-02-20 Synthelabo 2-(aminoalkyl)-5-(arylalkyl)-1,3-dioxanderivater, fremgangsmåde til fremstilling deraf og anvendelse deraf i terapien
US5173506A (en) * 1990-08-16 1992-12-22 Schering Corporation N-(mercaptoalkyl)ureas and carbamates
FR2742152B1 (fr) * 1995-12-06 1998-01-16 Synthelabo Derives de 5-naphtalen-1-yl-1,3-dioxanes, leur preparation et leur application en therapeutique
AT403579B (de) * 1995-12-07 1998-03-25 Agrolinz Melamin Gmbh Verfahren zur herstellung von hochreinem melamin
AU8025198A (en) 1997-06-05 1998-12-21 Sanofi-Synthelabo 5-naphthalen-1-yl-1,3-dioxane derivatives, preparation and therapeutic application
DE69939165D1 (de) * 1998-04-16 2008-09-04 Encysive Pharmaceuticals Inc N,n-disubstituierte amide welche die bindung von integrinen an ihre rezeptoren hemmen
FR2816938B1 (fr) * 2000-11-22 2003-01-03 Sanofi Synthelabo Derives de 3-aroylindole, leur procede de preparation et les compositions pharmaceutiques en contenant
FR2843964B1 (fr) * 2002-08-29 2004-10-01 Sanofi Synthelabo Derives de dioxane-2-alkylcarbamates, leur preparation et leur application en therapeutique

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