BR9810742A - Derivados de 5-naftalen -1il-1,3-dioxana, preparação dos mesmos e aplicação em terapia - Google Patents
Derivados de 5-naftalen -1il-1,3-dioxana, preparação dos mesmos e aplicação em terapiaInfo
- Publication number
- BR9810742A BR9810742A BR9810742-9A BR9810742A BR9810742A BR 9810742 A BR9810742 A BR 9810742A BR 9810742 A BR9810742 A BR 9810742A BR 9810742 A BR9810742 A BR 9810742A
- Authority
- BR
- Brazil
- Prior art keywords
- group
- therapy
- application
- nitrogen
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D319/04—1,3-Dioxanes; Hydrogenated 1,3-dioxanes
- C07D319/06—1,3-Dioxanes; Hydrogenated 1,3-dioxanes not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Psychology (AREA)
- Ophthalmology & Optometry (AREA)
- Pain & Pain Management (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Patente de Invenção: <B>"DERIVADOS DE 5-NAFTALEN-1-IL-1,3-DIOXANA, PREPARAçãO DOS MESMOS E APLICAçãO EM TERAPIA"<D>. Compostos de fórmula geral (I) na qual R~ 1~ representa um grupo alquila, V representa um átomo de hidrogênio ou um grupo alquila linear ou ramificado, cicloalquila, cicloalquilmetila, fenilalquila eventualmente substituído sobre o núcleo fenila, carboximetila, alcoxicarbonilmetila, carbamoilmetila eventualmente substituído sobre o nitrogênio, W representa um grupo carboximetila, alcoxicarbonilmetila, carbamoilmetila eventualmente substituído sobre o nitrogênio, um grupo cíclico que tem de 4 a 7 ângulos e que contém eventualmente um átomo de oxigênio ou de enxofre ou um grupo piridinilmetila, 1-metilpirrolilmetila, furanilmetila, tienilmetila ou 1,3-tiazolilmetila ou então V e W formam juntos e com o átomo de nitrogênio, um grupo pirrolidinila, piperidinila ou 1,2,3,4-tetrahidroisoquinoleína. Aplicação em terapia.
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9706944A FR2764287B1 (fr) | 1997-06-05 | 1997-06-05 | Derives de 5-naphtalen-1-yl-1,3-dioxanes, leur preparation et leur application en therapeutique |
FR9706947A FR2764291B1 (fr) | 1997-06-05 | 1997-06-05 | Derives de 5-naphtalen-1-yl-1,3-dioxane, leur preparation et leur application en therapeutique |
FR9706945A FR2764288B1 (fr) | 1997-06-05 | 1997-06-05 | Derives de 5-naphtalen-1-yl-1,3-dioxane, leur preparation et leur application en therapeutique |
FR9706946A FR2764289B1 (fr) | 1997-06-05 | 1997-06-05 | Derives de 5-naphtalen-1-yl-1,3-dioxane, leur preparation et leur application en therapeutique |
PCT/FR1998/001113 WO1998055474A1 (fr) | 1997-06-05 | 1998-06-03 | Derives de 5-naphtalen-1-yl-1,3-dioxane, leur preparation et leur application en therapeutique |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9810742A true BR9810742A (pt) | 2000-09-12 |
Family
ID=27447000
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9810742-9A BR9810742A (pt) | 1997-06-05 | 1998-06-03 | Derivados de 5-naftalen -1il-1,3-dioxana, preparação dos mesmos e aplicação em terapia |
Country Status (18)
Country | Link |
---|---|
EP (1) | EP0986552A1 (pt) |
JP (1) | JP2002502412A (pt) |
KR (1) | KR20010013435A (pt) |
CN (1) | CN1265658A (pt) |
AR (1) | AR012908A1 (pt) |
AU (1) | AU8025198A (pt) |
BG (1) | BG103937A (pt) |
BR (1) | BR9810742A (pt) |
CA (1) | CA2290695A1 (pt) |
CO (1) | CO4940480A1 (pt) |
EE (1) | EE9900560A (pt) |
HU (1) | HUP0002166A3 (pt) |
IL (1) | IL133242A0 (pt) |
NO (1) | NO995966L (pt) |
PL (1) | PL337234A1 (pt) |
SK (1) | SK166199A3 (pt) |
TR (1) | TR199903022T2 (pt) |
WO (1) | WO1998055474A1 (pt) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20020107283A1 (en) * | 2000-07-21 | 2002-08-08 | Codd Ellen E. | Carbamate compounds for use in preventing or treating neuropathic pain and cluster and migraine headache-associated pain |
FR2843964B1 (fr) * | 2002-08-29 | 2004-10-01 | Sanofi Synthelabo | Derives de dioxane-2-alkylcarbamates, leur preparation et leur application en therapeutique |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0461958B1 (fr) * | 1990-06-15 | 1994-09-14 | Synthelabo | Dérivés de 2-(aminoalkyl)-5-(arylalkyl)-1,3-dioxanes, leur préparation et leur application en thérapeutique |
FR2714055B1 (fr) * | 1993-12-22 | 1996-01-19 | Synthelabo | Dérivés de 5-(arylalkyl)-1,3-dioxane substitués en position 2, leur préparation et leur utilisation en thérapeutique. |
FR2742152B1 (fr) * | 1995-12-06 | 1998-01-16 | Synthelabo | Derives de 5-naphtalen-1-yl-1,3-dioxanes, leur preparation et leur application en therapeutique |
-
1998
- 1998-06-03 WO PCT/FR1998/001113 patent/WO1998055474A1/fr not_active Application Discontinuation
- 1998-06-03 CA CA002290695A patent/CA2290695A1/en not_active Abandoned
- 1998-06-03 EE EEP199900560A patent/EE9900560A/xx unknown
- 1998-06-03 PL PL98337234A patent/PL337234A1/xx unknown
- 1998-06-03 IL IL13324298A patent/IL133242A0/xx unknown
- 1998-06-03 EP EP98928419A patent/EP0986552A1/fr not_active Withdrawn
- 1998-06-03 SK SK1661-99A patent/SK166199A3/sk unknown
- 1998-06-03 JP JP50172399A patent/JP2002502412A/ja active Pending
- 1998-06-03 CN CN98807817A patent/CN1265658A/zh active Pending
- 1998-06-03 AR ARP980102585A patent/AR012908A1/es unknown
- 1998-06-03 TR TR1999/03022T patent/TR199903022T2/xx unknown
- 1998-06-03 KR KR1019997011436A patent/KR20010013435A/ko not_active Application Discontinuation
- 1998-06-03 AU AU80251/98A patent/AU8025198A/en not_active Abandoned
- 1998-06-03 HU HU0002166A patent/HUP0002166A3/hu unknown
- 1998-06-03 BR BR9810742-9A patent/BR9810742A/pt not_active IP Right Cessation
- 1998-06-04 CO CO98031750A patent/CO4940480A1/es unknown
-
1999
- 1999-11-30 BG BG103937A patent/BG103937A/xx unknown
- 1999-12-03 NO NO995966A patent/NO995966L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
SK166199A3 (en) | 2000-06-12 |
CA2290695A1 (en) | 1998-12-10 |
HUP0002166A2 (hu) | 2001-06-28 |
TR199903022T2 (xx) | 2000-04-21 |
EE9900560A (et) | 2000-06-15 |
EP0986552A1 (fr) | 2000-03-22 |
AU8025198A (en) | 1998-12-21 |
HUP0002166A3 (en) | 2002-12-28 |
NO995966D0 (no) | 1999-12-03 |
BG103937A (en) | 2000-07-31 |
CN1265658A (zh) | 2000-09-06 |
IL133242A0 (en) | 2001-03-19 |
NO995966L (no) | 2000-02-04 |
KR20010013435A (ko) | 2001-02-26 |
JP2002502412A (ja) | 2002-01-22 |
WO1998055474A1 (fr) | 1998-12-10 |
CO4940480A1 (es) | 2000-07-24 |
PL337234A1 (en) | 2000-08-14 |
AR012908A1 (es) | 2000-11-22 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NO20023457L (no) | Nye piperidinforbindelser og legemidler inneholdende de samme | |
DK1077927T3 (da) | Nye substituerede cykliske forbindelser, fremgangsmåde til fremstilling heraf og farmaceutiske sammensætninger indeholdende disse | |
BR9807132A (pt) | Derivados de pirrolidina tendo atividade inibitória de fosfolipase a2 | |
PT1004578E (pt) | Derivados hidroxamida do acido 5-oxo-pirrolidino-2-carboxilico | |
DK1265606T3 (da) | Celleadhæsionsinhibitorer | |
ATE438624T1 (de) | 2-pyridonderivate mit affinität für den cannabinoid-typ-2-rezeptor | |
BR9813848A (pt) | Composto heterocìclico fundido substituìdo, uso do mesmo, e, composição farmacêutica. | |
DE69416848T2 (de) | Amidino-derivate als no-synthetase inhibitoren | |
HUP0302962A2 (hu) | Béta-karbolinszármazékok, ezeket a vegyületeket tartalmazó gyógyászati készítmények és a vegyületek alkalmazása | |
BR0210297A (pt) | Derivados de n-arilfenilacetamida e composição farmacêutcia contendo os mesmos | |
BR0006823A (pt) | Composição farmacêutica estabilizada, uso de composto de polipeptìdeo cìclico, preparação de injeção e pacote comercial | |
DK1140918T3 (da) | Thrombininhibitorer | |
BR0113071A (pt) | Compostos de 1,4-dihidropiridina como antagonistas da bradiquinina | |
BR0316609A (pt) | Sinomenina e compostos de sinomenina, sìntese e uso | |
BR9810742A (pt) | Derivados de 5-naftalen -1il-1,3-dioxana, preparação dos mesmos e aplicação em terapia | |
BR0002287A (pt) | Compostos de piridina ou piperidina substituìdas, processo para preparação deles e composições farmacêuticas contendo-os | |
BR0106248A (pt) | Inibidores de metaloprotease, processo para a sua preparação e composições farmacêuticas contendo os mesmos | |
DE69941307D1 (de) | Prenyl transferasinhibitoren | |
BR9907426A (pt) | Tetrahidronaftalenos | |
BR9714007A (pt) | Novos derivados da eritromicina seu processo de preparação e sua aplicação como medicamentos | |
MY136928A (en) | New isoquinoline compounds, a process for their preparation and pharmaceutical composition containing them | |
DK0682024T3 (da) | Cyclohexan-derivater, fremgangsmåder til fremstilling og deres anvendelse som glucose-6-phosphatase inhibitorer | |
BR9811962A (pt) | Métodos para baixar as contagens de plaquetas | |
ATE311877T1 (de) | Lp(a)-mindernde mittel und inhibitoren der apoprotein (a) produktion | |
DK1312608T3 (da) | Discodermolid-analoge samt deres farmaceutiske anvendelse |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 5A, 6A, 7A, 8A E 9A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1889 DE 20/03/2007. |