JP2005509590A5 - - Google Patents

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Publication number
JP2005509590A5
JP2005509590A5 JP2003503584A JP2003503584A JP2005509590A5 JP 2005509590 A5 JP2005509590 A5 JP 2005509590A5 JP 2003503584 A JP2003503584 A JP 2003503584A JP 2003503584 A JP2003503584 A JP 2003503584A JP 2005509590 A5 JP2005509590 A5 JP 2005509590A5
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JP
Japan
Prior art keywords
phenyl
methoxy
phenoxy
compound
group
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
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JP2003503584A
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English (en)
Japanese (ja)
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JP2005509590A6 (ja
JP2005509590A (ja
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Priority claimed from PCT/US2002/016950 external-priority patent/WO2002100813A2/en
Publication of JP2005509590A publication Critical patent/JP2005509590A/ja
Publication of JP2005509590A6 publication Critical patent/JP2005509590A6/ja
Publication of JP2005509590A5 publication Critical patent/JP2005509590A5/ja
Pending legal-status Critical Current

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JP2003503584A 2001-06-07 2002-05-30 ペルオキシソーム増殖因子活性化受容体の調節物質 Pending JP2005509590A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US29714401P 2001-06-07 2001-06-07
US60/297,144 2001-06-07
PCT/US2002/016950 WO2002100813A2 (en) 2001-06-07 2002-05-30 Modulators of peroxisome proliferator activated receptors

Publications (3)

Publication Number Publication Date
JP2005509590A JP2005509590A (ja) 2005-04-14
JP2005509590A6 JP2005509590A6 (ja) 2005-08-04
JP2005509590A5 true JP2005509590A5 (enExample) 2006-01-05

Family

ID=23145037

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003503584A Pending JP2005509590A (ja) 2001-06-07 2002-05-30 ペルオキシソーム増殖因子活性化受容体の調節物質

Country Status (24)

Country Link
US (2) US7192982B2 (enExample)
EP (1) EP1392637A2 (enExample)
JP (1) JP2005509590A (enExample)
KR (1) KR20040012905A (enExample)
CN (1) CN1543451A (enExample)
AR (1) AR036084A1 (enExample)
BR (1) BR0210190A (enExample)
CA (1) CA2449256A1 (enExample)
CO (1) CO5640097A2 (enExample)
CZ (1) CZ20033309A3 (enExample)
EA (1) EA200400010A1 (enExample)
EC (1) ECSP034877A (enExample)
EE (1) EE200400001A (enExample)
HR (1) HRP20031001A2 (enExample)
HU (1) HUP0400280A3 (enExample)
IL (1) IL158873A0 (enExample)
MX (1) MXPA03011201A (enExample)
NO (1) NO20035439D0 (enExample)
NZ (1) NZ529351A (enExample)
PE (1) PE20030099A1 (enExample)
PL (1) PL368051A1 (enExample)
SK (1) SK14912003A3 (enExample)
WO (1) WO2002100813A2 (enExample)
ZA (1) ZA200308863B (enExample)

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CN102114076B (zh) * 2006-10-25 2013-04-10 中国科学院上海生命科学研究院 肉桂提取物的制备方法、肉桂提取物、其组合物以及用途
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JP2016516004A (ja) 2013-02-22 2016-06-02 メルク・シャープ・アンド・ドーム・コーポレーションＭｅｒｃｋ Ｓｈａｒｐ ＆ Ｄｏｈｍｅ Ｃｏｒｐ． 抗糖尿病二環式化合物
EP3065723B1 (en) 2013-11-05 2020-09-23 Ben Gurion University of the Negev Research and Development Authority Compounds for the treatment of diabetes and disease complications arising from same
CN104926743A (zh) * 2015-07-14 2015-09-23 佛山市赛维斯医药科技有限公司 含苯并异恶唑和末端苄基类结构的化合物及其用途
CN104945344A (zh) * 2015-07-14 2015-09-30 佛山市赛维斯医药科技有限公司 一类含苯并异恶唑和末端胺基结构化合物及其用途
CN104926742A (zh) * 2015-07-14 2015-09-23 佛山市赛维斯医药科技有限公司 一类含苯并异恶唑和硝基苯基类结构的化合物及其用途
CN104926745A (zh) * 2015-07-14 2015-09-23 佛山市赛维斯医药科技有限公司 含苯并异恶唑和末端卤代苄基类结构的化合物及其用途
CN104987314A (zh) * 2015-07-14 2015-10-21 佛山市赛维斯医药科技有限公司 含苯并异恶唑和末端硝基苄基类结构的化合物及其用途
CN105037290A (zh) * 2015-07-14 2015-11-11 佛山市赛维斯医药科技有限公司 一类含苯并异恶唑和腈基苯类结构化合物及其用途
CN104961702A (zh) * 2015-07-14 2015-10-07 佛山市赛维斯医药科技有限公司 苯并异恶唑类11β-HSD1抑制剂、制备方法及其用途
CN104926746A (zh) * 2015-07-14 2015-09-23 佛山市赛维斯医药科技有限公司 含苯并异恶唑和末端胺基苄基类结构的化合物及其用途
CN104961703A (zh) * 2015-07-14 2015-10-07 佛山市赛维斯医药科技有限公司 一类苯并异恶唑类11β-HSD1抑制剂、制备方法及其用途
CN104974103A (zh) * 2015-07-14 2015-10-14 佛山市赛维斯医药科技有限公司 一类含苯并异恶唑和烷氧苯基类结构的化合物及其用途
CN104926744A (zh) * 2015-07-14 2015-09-23 佛山市赛维斯医药科技有限公司 一类含苯并异恶唑和末端苄基类结构的化合物及其用途
CN105001174A (zh) * 2015-07-14 2015-10-28 佛山市赛维斯医药科技有限公司 含苯并异恶唑和末端腈基苄基类结构的化合物及其用途
RU2764243C2 (ru) 2017-09-22 2022-01-14 ДЖУБИЛАНТ ЭПИПЭД ЭлЭлСи Гетероциклические соединения в качестве ингибиторов PAD
CN111225915B (zh) 2017-10-18 2023-03-07 朱比兰特埃皮帕德有限公司 作为pad抑制剂的咪唑并吡啶化合物
US11629135B2 (en) 2017-11-06 2023-04-18 Jubilant Prodell Llc Pyrimidine derivatives as inhibitors of PD1/PD-L1 activation
RS65576B1 (sr) 2017-11-24 2024-06-28 Jubilant Episcribe Llc Heterociklična jedinjenja kao inhibitori prmt5
CN112105610B (zh) 2018-03-13 2024-01-26 朱比连特普罗德尔有限责任公司 作为pd1/pd-l1相互作用/活化的抑制剂的双环化合物
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