HUP0400280A3 - Modulators of peroxisome proliferator activated receptors, process for their preparation and pharmaceutical compositions containing them - Google Patents
Modulators of peroxisome proliferator activated receptors, process for their preparation and pharmaceutical compositions containing themInfo
- Publication number
- HUP0400280A3 HUP0400280A3 HU0400280A HUP0400280A HUP0400280A3 HU P0400280 A3 HUP0400280 A3 HU P0400280A3 HU 0400280 A HU0400280 A HU 0400280A HU P0400280 A HUP0400280 A HU P0400280A HU P0400280 A3 HUP0400280 A3 HU P0400280A3
- Authority
- HU
- Hungary
- Prior art keywords
- modulators
- preparation
- pharmaceutical compositions
- compositions containing
- peroxisome proliferator
- Prior art date
Links
- 102000003728 Peroxisome Proliferator-Activated Receptors Human genes 0.000 title 1
- 108090000029 Peroxisome Proliferator-Activated Receptors Proteins 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
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- C07C59/40—Unsaturated compounds
- C07C59/58—Unsaturated compounds containing ether groups, groups, groups, or groups
- C07C59/64—Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings
- C07C59/66—Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings the non-carboxylic part of the ether containing six-membered aromatic rings
- C07C59/68—Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings the non-carboxylic part of the ether containing six-membered aromatic rings the oxygen atom of the ether group being bound to a non-condensed six-membered aromatic ring
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- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
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- C07C219/04—Compounds containing amino and esterified hydroxy groups bound to the same carbon skeleton having esterified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C219/10—Compounds containing amino and esterified hydroxy groups bound to the same carbon skeleton having esterified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having at least one of the hydroxy groups esterified by a carboxylic acid having the esterifying carboxyl group bound to an acyclic carbon atom of a carbon skeleton containing rings
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HUP0400268A2 (hu) | 2001-06-07 | 2004-07-28 | Eli Lilly And Co. | Peroxiszóma proliferátorral aktivált receptorokat (PPAR) módosító hatóanyagok, alkalmazásuk és ezeket tartalmazó gyógyszerkészítmények |
US7101910B2 (en) * | 2001-06-12 | 2006-09-05 | Wellstat Therapeutics Corporation | Compounds for the treatment of metabolic disorders |
ITRM20020016A1 (it) * | 2002-01-15 | 2003-07-15 | Sigma Tau Ind Farmaceuti | Derivati di acidi fenil(alchil)carbossilici e derivati fenilalchileterociclici dionici, loro uso come medicamenti ad attivita' ipoglicemizza |
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FR2872159B1 (fr) * | 2004-06-28 | 2007-10-05 | Merck Sante Soc Par Actions Si | Nouveaux derives acides carboxyliques phenyliques et leur utilisation dans le traitement du diabete |
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MY145712A (en) * | 2004-09-15 | 2012-03-30 | Janssen Pharmaceutica Nv | 4-((phenoxyalkyl)thio)-phenoxyacetic acids and analogs |
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FR2882359A1 (fr) * | 2005-02-24 | 2006-08-25 | Negma Lerads Soc Par Actions S | Derives activateurs de ppar, procede de preparation et application en therapeutique |
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CN105037290A (zh) * | 2015-07-14 | 2015-11-11 | 佛山市赛维斯医药科技有限公司 | 一类含苯并异恶唑和腈基苯类结构化合物及其用途 |
CN104926744A (zh) * | 2015-07-14 | 2015-09-23 | 佛山市赛维斯医药科技有限公司 | 一类含苯并异恶唑和末端苄基类结构的化合物及其用途 |
CN104974103A (zh) * | 2015-07-14 | 2015-10-14 | 佛山市赛维斯医药科技有限公司 | 一类含苯并异恶唑和烷氧苯基类结构的化合物及其用途 |
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CN104926743A (zh) * | 2015-07-14 | 2015-09-23 | 佛山市赛维斯医药科技有限公司 | 含苯并异恶唑和末端苄基类结构的化合物及其用途 |
CN104926746A (zh) * | 2015-07-14 | 2015-09-23 | 佛山市赛维斯医药科技有限公司 | 含苯并异恶唑和末端胺基苄基类结构的化合物及其用途 |
CN104926745A (zh) * | 2015-07-14 | 2015-09-23 | 佛山市赛维斯医药科技有限公司 | 含苯并异恶唑和末端卤代苄基类结构的化合物及其用途 |
CN105001174A (zh) * | 2015-07-14 | 2015-10-28 | 佛山市赛维斯医药科技有限公司 | 含苯并异恶唑和末端腈基苄基类结构的化合物及其用途 |
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IL272667B (en) | 2017-10-18 | 2022-09-01 | Jubilant Epipad LLC | Imidazo-pyridine compounds as pad inhibitors |
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SE9801990D0 (sv) | 1998-06-04 | 1998-06-04 | Astra Ab | New 3-aryl propionic acid derivatives and analogs |
SE9801992D0 (sv) | 1998-06-04 | 1998-06-04 | Astra Ab | New 3-aryl-2-hydroxypropionic acid derivative I |
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JPWO2002080899A1 (ja) * | 2001-03-30 | 2005-01-06 | エーザイ株式会社 | 消化器疾患治療剤 |
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2002
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- 2002-05-30 CN CNA028115309A patent/CN1543451A/zh active Pending
- 2002-05-30 EE EEP200400001A patent/EE200400001A/xx unknown
- 2002-05-30 SK SK1491-2003A patent/SK14912003A3/sk not_active Application Discontinuation
- 2002-05-30 EP EP02739503A patent/EP1392637A2/en not_active Withdrawn
- 2002-05-30 CZ CZ20033309A patent/CZ20033309A3/cs unknown
- 2002-05-30 EA EA200400010A patent/EA200400010A1/ru unknown
- 2002-05-30 PL PL02368051A patent/PL368051A1/xx not_active Application Discontinuation
- 2002-05-30 BR BR0210190-4A patent/BR0210190A/pt not_active IP Right Cessation
- 2002-05-30 IL IL15887302A patent/IL158873A0/xx unknown
- 2002-05-30 NZ NZ529351A patent/NZ529351A/en unknown
- 2002-05-30 WO PCT/US2002/016950 patent/WO2002100813A2/en active Application Filing
- 2002-05-30 CA CA002449256A patent/CA2449256A1/en not_active Abandoned
- 2002-05-30 KR KR10-2003-7016050A patent/KR20040012905A/ko not_active Application Discontinuation
- 2002-05-30 HU HU0400280A patent/HUP0400280A3/hu unknown
- 2002-05-30 US US10/479,262 patent/US7192982B2/en not_active Expired - Fee Related
- 2002-05-30 JP JP2003503584A patent/JP2005509590A/ja active Pending
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2003
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CA2449256A1 (en) | 2002-12-19 |
CZ20033309A3 (cs) | 2004-05-12 |
NZ529351A (en) | 2006-01-27 |
PL368051A1 (en) | 2005-03-21 |
US20050020684A1 (en) | 2005-01-27 |
AR036084A1 (es) | 2004-08-11 |
JP2005509590A (ja) | 2005-04-14 |
KR20040012905A (ko) | 2004-02-11 |
EA200400010A1 (ru) | 2004-06-24 |
ZA200308863B (en) | 2005-02-14 |
PE20030099A1 (es) | 2003-04-08 |
NO20035439D0 (no) | 2003-12-05 |
WO2002100813A2 (en) | 2002-12-19 |
US20070276138A1 (en) | 2007-11-29 |
EP1392637A2 (en) | 2004-03-03 |
ECSP034877A (es) | 2004-01-28 |
EE200400001A (et) | 2004-02-16 |
SK14912003A3 (sk) | 2004-09-08 |
WO2002100813A3 (en) | 2003-11-27 |
CO5640097A2 (es) | 2006-05-31 |
HRP20031001A2 (en) | 2004-06-30 |
BR0210190A (pt) | 2004-04-06 |
US7192982B2 (en) | 2007-03-20 |
MXPA03011201A (es) | 2004-02-26 |
CN1543451A (zh) | 2004-11-03 |
HUP0400280A2 (hu) | 2005-01-28 |
IL158873A0 (en) | 2004-05-12 |
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