JP2005508300A5 - - Google Patents

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Publication number
JP2005508300A5
JP2005508300A5 JP2003507098A JP2003507098A JP2005508300A5 JP 2005508300 A5 JP2005508300 A5 JP 2005508300A5 JP 2003507098 A JP2003507098 A JP 2003507098A JP 2003507098 A JP2003507098 A JP 2003507098A JP 2005508300 A5 JP2005508300 A5 JP 2005508300A5
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JP
Japan
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alkyl
substituted
effective amount
pharmaceutically effective
heteroaryl
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JP2003507098A
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English (en)
Japanese (ja)
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JP4344607B2 (ja
JP2005508300A (ja
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Priority claimed from GBGB0115393.1A external-priority patent/GB0115393D0/en
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Publication of JP2005508300A publication Critical patent/JP2005508300A/ja
Publication of JP2005508300A5 publication Critical patent/JP2005508300A5/ja
Application granted granted Critical
Publication of JP4344607B2 publication Critical patent/JP4344607B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2003507098A 2001-06-23 2002-06-21 蛋白キナーゼ阻害剤としてのピロロピリミジン Expired - Fee Related JP4344607B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0115393.1A GB0115393D0 (en) 2001-06-23 2001-06-23 Chemical compounds
US30167801P 2001-06-28 2001-06-28
PCT/GB2002/002835 WO2003000695A1 (en) 2001-06-23 2002-06-21 Pyrrolopyrimidines as protein kinase inhibitors

Publications (3)

Publication Number Publication Date
JP2005508300A JP2005508300A (ja) 2005-03-31
JP2005508300A5 true JP2005508300A5 (https=) 2006-01-05
JP4344607B2 JP4344607B2 (ja) 2009-10-14

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ID=9917225

Family Applications (1)

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JP2003507098A Expired - Fee Related JP4344607B2 (ja) 2001-06-23 2002-06-21 蛋白キナーゼ阻害剤としてのピロロピリミジン

Country Status (22)

Country Link
EP (1) EP1404676A1 (https=)
JP (1) JP4344607B2 (https=)
CN (1) CN1294135C (https=)
AU (1) AU2002314325B8 (https=)
BR (1) BR0210652A (https=)
CA (1) CA2451932C (https=)
CZ (1) CZ20033443A3 (https=)
EA (1) EA007415B1 (https=)
EC (1) ECSP034922A (https=)
EE (1) EE05432B1 (https=)
GB (1) GB0115393D0 (https=)
HU (1) HUP0400300A3 (https=)
ME (1) MEP19308A (https=)
NZ (1) NZ529766A (https=)
OA (1) OA12632A (https=)
PL (1) PL374096A1 (https=)
RS (1) RS51698B (https=)
SK (1) SK15882003A3 (https=)
TN (1) TNSN03144A1 (https=)
TR (1) TR200302242T2 (https=)
UA (1) UA76760C2 (https=)
WO (1) WO2003000695A1 (https=)

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RU2711869C3 (ru) 2009-12-01 2022-02-02 Эббви Инк. Имидазопирролопиразиновые производные, полезные для лечения заболеваний, вызванных аномальной активностью протеинкиназ Jak1, Jak3 или Syk
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CN103476776B (zh) * 2011-01-07 2016-09-28 北京赛林泰医药技术有限公司 作为FAK/Pyk2抑制剂的2,4-二氨基-6,7-二氢-5H-吡咯并[2,3]嘧啶衍生物
CN102093364B (zh) * 2011-01-07 2015-01-28 北京赛林泰医药技术有限公司 作为FAK/Pyk2抑制剂的2,4-二氨基-6,7-二氢-5H-吡咯并[2,3]嘧啶衍生物
CN103797010B (zh) 2011-06-20 2016-02-24 因塞特控股公司 作为jak抑制剂的氮杂环丁烷基苯基、吡啶基或吡嗪基甲酰胺衍生物
TW201313721A (zh) 2011-08-18 2013-04-01 Incyte Corp 作為ｊａｋ抑制劑之環己基氮雜環丁烷衍生物
UA111854C2 (uk) 2011-09-07 2016-06-24 Інсайт Холдінгс Корпорейшн Способи і проміжні сполуки для отримання інгібіторів jak
JP6182593B2 (ja) 2012-04-20 2017-08-16 アドヴィーナス セラピューティクス リミテッド 置換ヘテロ二環化合物、組成物及び医薬並びにそれらの用途
TW201406761A (zh) 2012-05-18 2014-02-16 Incyte Corp 做爲ｊａｋ抑制劑之哌啶基環丁基取代之吡咯并吡啶及吡咯并嘧啶衍生物
KR101916443B1 (ko) 2012-07-26 2018-11-08 글락소 그룹 리미티드 Pad4 억제제로서의 2-(아자인돌-2-일) 벤즈이미다졸
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RS62867B1 (sr) 2013-03-06 2022-02-28 Incyte Holdings Corp Postupci i intermedijeri za dobijanje inhibitora jak
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CN104804001B9 (zh) * 2014-01-24 2022-02-08 江苏柯菲平医药股份有限公司 4-取代吡咯并[2,3-d]嘧啶化合物及其用途
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