JP2005507873A5 - - Google Patents
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- Publication number
- JP2005507873A5 JP2005507873A5 JP2003521208A JP2003521208A JP2005507873A5 JP 2005507873 A5 JP2005507873 A5 JP 2005507873A5 JP 2003521208 A JP2003521208 A JP 2003521208A JP 2003521208 A JP2003521208 A JP 2003521208A JP 2005507873 A5 JP2005507873 A5 JP 2005507873A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- compound
- formula
- haloalkyl
- independently
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 claims description 40
- 229910052739 hydrogen Inorganic materials 0.000 claims description 21
- 238000000034 method Methods 0.000 claims description 21
- 229910052794 bromium Inorganic materials 0.000 claims description 16
- 229910052801 chlorine Inorganic materials 0.000 claims description 16
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 15
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 10
- 229910052736 halogen Inorganic materials 0.000 claims description 10
- 150000002367 halogens Chemical class 0.000 claims description 10
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 claims description 6
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims description 5
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims description 5
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims description 5
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 5
- 125000006656 (C2-C4) alkenyl group Chemical group 0.000 claims description 5
- 125000006650 (C2-C4) alkynyl group Chemical group 0.000 claims description 5
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims description 5
- -1 C 1 -C 4 alkylthio Chemical group 0.000 claims description 5
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 5
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims description 5
- 125000000217 alkyl group Chemical group 0.000 claims description 5
- 125000006310 cycloalkyl amino group Chemical group 0.000 claims description 5
- 125000004663 dialkyl amino group Chemical group 0.000 claims description 5
- 125000004473 dialkylaminocarbonyl group Chemical group 0.000 claims description 5
- 238000004519 manufacturing process Methods 0.000 claims description 4
- 150000004703 alkoxides Chemical class 0.000 claims description 3
- 230000002152 alkylating effect Effects 0.000 claims description 3
- 239000003795 chemical substances by application Substances 0.000 claims description 3
- 239000002253 acid Substances 0.000 claims description 2
- 230000015572 biosynthetic process Effects 0.000 description 1
- 229910052731 fluorine Inorganic materials 0.000 description 1
- 229910052740 iodine Inorganic materials 0.000 description 1
- 125000001453 quaternary ammonium group Chemical group 0.000 description 1
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US31191901P | 2001-08-13 | 2001-08-13 | |
| US34189401P | 2001-12-19 | 2001-12-19 | |
| US36965902P | 2002-04-02 | 2002-04-02 | |
| PCT/US2002/025612 WO2003016282A2 (en) | 2001-08-13 | 2002-08-13 | Substituted 1h-dihydropyrazoles, their preparation and use |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005507873A JP2005507873A (ja) | 2005-03-24 |
| JP2005507873A5 true JP2005507873A5 (enExample) | 2006-01-05 |
| JP4448327B2 JP4448327B2 (ja) | 2010-04-07 |
Family
ID=27405543
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003521208A Expired - Fee Related JP4448327B2 (ja) | 2001-08-13 | 2002-08-13 | 新規置換１ｈ−ジヒドロピラゾール、それらの製造および使用 |
Country Status (8)
| Country | Link |
|---|---|
| US (3) | US7038057B2 (enExample) |
| EP (1) | EP1417200B1 (enExample) |
| JP (1) | JP4448327B2 (enExample) |
| AT (1) | ATE469892T1 (enExample) |
| AU (1) | AU2002319814A1 (enExample) |
| CA (1) | CA2454298A1 (enExample) |
| DE (1) | DE60236600D1 (enExample) |
| WO (1) | WO2003016282A2 (enExample) |
Families Citing this family (67)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI325302B (en) * | 2001-08-13 | 2010-06-01 | Du Pont | Benzoxazinone compounds |
| US7038057B2 (en) * | 2001-08-13 | 2006-05-02 | E.I. Du Pont De Nemours And Company | Substituted 1H-dihydropyrazoles, their preparation and use |
| TWI356822B (en) | 2001-08-13 | 2012-01-21 | Du Pont | Novel substituted dihydro 3-halo-1h-pyrazole-5-car |
| AR036872A1 (es) * | 2001-08-13 | 2004-10-13 | Du Pont | Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados |
| DE60226875D1 (de) * | 2001-08-15 | 2008-07-10 | Du Pont | Orthosubstituierte arylamide zur bekämpfung von wirbellosen schädlingen |
| ES2319743T3 (es) * | 2001-08-16 | 2009-05-12 | E.I. Du Pont De Nemours And Company | Antranilamidas sustituidas para controlar plagas de invertebrados. |
| TWI283164B (en) * | 2001-09-21 | 2007-07-01 | Du Pont | Anthranilamide arthropodicide treatment |
| US20040110777A1 (en) * | 2001-12-03 | 2004-06-10 | Annis Gary David | Quinazolinones and pyridinylpyrimidinones for controlling invertebrate pests |
| EP1467988B1 (en) * | 2002-01-22 | 2013-07-17 | E.I. Du Pont De Nemours And Company | Quinazoline(di)ones for invertebrate pest control |
| JP4287816B2 (ja) * | 2002-06-13 | 2009-07-01 | イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー | ピラゾールカルボキサミド殺虫剤 |
| TWI326283B (en) * | 2002-07-31 | 2010-06-21 | Du Pont | Method for preparing fused oxazinones |
| KR20050075001A (ko) * | 2002-11-15 | 2005-07-19 | 이 아이 듀폰 디 네모아 앤드 캄파니 | 신규 안트라닐아미드 살충제 |
| VN23181A1 (en) * | 2003-01-28 | 2010-07-26 | Du Pont | Cyano anthranilamide insecticides |
| TWI367882B (en) * | 2003-03-26 | 2012-07-11 | Du Pont | Preparation and use of 2-substituted-5-oxo-3-pyrazolidinecarboxylates |
| US7276601B2 (en) * | 2003-06-12 | 2007-10-02 | E.I. Du Pont De Nemours And Company | Method and preparing fused oxazinones |
| DE102004021564A1 (de) | 2003-11-14 | 2005-07-07 | Bayer Cropscience Ag | Wirkstoffkombinationen mit insektiziden Eigenschaften |
| DE102004006075A1 (de) | 2003-11-14 | 2005-06-16 | Bayer Cropscience Ag | Wirkstoffkombinationen mit insektiziden Eigenschaften |
| DE10353281A1 (de) | 2003-11-14 | 2005-06-16 | Bayer Cropscience Ag | Wirkstoffkombination mit insektiziden und akariziden Eigenschaften |
| EP1691611A1 (de) | 2003-12-04 | 2006-08-23 | Bayer CropScience Aktiengesellschaft | Wirkstoffkombinationen mit insektiziden eigenschaften |
| DE10356550A1 (de) | 2003-12-04 | 2005-07-07 | Bayer Cropscience Ag | Wirkstoffkombinationen mit insektiziden Eigenschaften |
| RU2006139953A (ru) * | 2004-04-13 | 2008-05-20 | Е.И. Дюпон Де Немур Энд Компани (Us) | Антраниламидные инсектициды |
| DE102004031100A1 (de) * | 2004-06-28 | 2006-01-12 | Bayer Cropscience Ag | Anthranilamide |
| GT200500179A (es) * | 2004-07-01 | 2006-02-23 | Mezclas sinergistas de agentes de antranilamida para el control de plagas de invertebrados | |
| JP4920878B2 (ja) * | 2004-07-14 | 2012-04-18 | 日本電気株式会社 | 認証システム、ネットワーク集線装置及びそれらに用いる認証方法並びにそのプログラム |
| DE102004035134A1 (de) | 2004-07-20 | 2006-02-16 | Bayer Cropscience Ag | Selektive Insektizide auf Basis von Halogenalkylnicotinsäurederivaten, Anthranilsäureamiden oder Phthalsäurediamiden und Safenern |
| MY140912A (en) * | 2004-07-26 | 2010-01-29 | Du Pont | Mixtures of anthranilamide invertebrate pest control agents |
| BRPI0516781A (pt) * | 2004-11-18 | 2008-09-23 | Du Pont | compostos, composições para o controle de pragas invertebradas, dispositivo de armadilha e composições spray e de isca para o controle de pragas invertebradas e métodos para o controle de pragas invertebradas |
| CN101243067A (zh) * | 2005-08-24 | 2008-08-13 | 杜邦公司 | 用于防治无脊椎害虫的新的邻氨基苯甲酰胺 |
| DE102005044108A1 (de) | 2005-09-15 | 2007-03-29 | Bayer Cropscience Ag | Dioxazin- und Oxdiazin-substituierte Arylamide |
| DE102006032168A1 (de) | 2006-06-13 | 2007-12-20 | Bayer Cropscience Ag | Anthranilsäurediamid-Derivate mit heteroaromatischen Substituenten |
| DE102006030710A1 (de) * | 2006-07-03 | 2008-01-10 | Bayer Cropscience Ag | Synergistische insektizide und fungizide Mischungen |
| WO2008031548A1 (en) * | 2006-09-11 | 2008-03-20 | Syngenta Participations Ag | Process for the preparation of anthranilamide derivatives |
| EP2083630A2 (en) * | 2006-11-17 | 2009-08-05 | Basf Se | Method for increasing the dry biomass of plants |
| CN104496901B (zh) * | 2006-12-15 | 2016-05-25 | 石原产业株式会社 | 邻氨基苯甲酰胺系化合物的制造方法 |
| JP5507045B2 (ja) * | 2006-12-15 | 2014-05-28 | 石原産業株式会社 | アントラニルアミド系化合物の製造方法 |
| JP2009001541A (ja) * | 2006-12-15 | 2009-01-08 | Ishihara Sangyo Kaisha Ltd | 新規ピラゾール化合物を中間体として用いるアントラニルアミド系化合物の製造方法 |
| TWI415827B (zh) | 2006-12-21 | 2013-11-21 | Du Pont | 製備２-胺基-５-氰基苯甲酸衍生物之方法 |
| PL2193714T3 (pl) * | 2007-04-25 | 2012-01-31 | Syngenta Participations Ag | Kompozycje grzybobójcze |
| ES2377588T3 (es) * | 2007-07-16 | 2012-03-29 | Syngenta Participations Ag | Insecticidas de antranilamida condensada |
| EP2100883A1 (de) * | 2008-03-10 | 2009-09-16 | Bayer CropScience AG | Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4carbonsäure-Derivaten |
| KR101687743B1 (ko) | 2008-12-18 | 2016-12-19 | 바이엘 인텔렉쳐 프로퍼티 게엠베하 | 살해충제로서의 테트라졸 치환된 안트라닐산 아미드 |
| EP2243777A1 (de) | 2009-04-03 | 2010-10-27 | Bayer CropScience AG | Verfahren zum Herstellen von Pyridyl-substituierten Pyrazolen |
| KR101701335B1 (ko) | 2009-07-23 | 2017-02-01 | 바이엘 인텔렉쳐 프로퍼티 게엠베하 | 아릴 치환된 피라졸의 제조방법 |
| BR112012014683B1 (pt) * | 2009-12-15 | 2017-11-07 | Bayer Cropscience Ag | Process for the production of 5-pyrazolcarboxylic acid derivatives 1-alkyl- / 1-aryl-substituted and compound acid |
| EP2533641B1 (de) | 2010-02-09 | 2016-07-13 | Bayer CropScience AG | Hydrazin-substituierte anthranilsäurederivate |
| EP2558460B1 (de) | 2010-04-16 | 2015-03-04 | Bayer Intellectual Property GmbH | Triazolsubstituierte anthranilsäureamide als pestizide |
| BR112012032247A2 (pt) | 2010-06-15 | 2015-09-15 | Bayer Ip Gmbh | derivados de ácido antranílico |
| BR112012032238A2 (pt) | 2010-06-15 | 2015-09-15 | Bayer Ip Gmbh | derivados de diamida antranílica que têm cadeias laterais cíclicas |
| WO2011157663A1 (de) | 2010-06-15 | 2011-12-22 | Bayer Cropscience Ag | Neue ortho-substituierte arylamid-derivate |
| WO2011157654A1 (de) | 2010-06-15 | 2011-12-22 | Bayer Cropscience Ag | Anthranilsäurediamid-derivate |
| KR20130093086A (ko) | 2010-07-09 | 2013-08-21 | 바이엘 인텔렉쳐 프로퍼티 게엠베하 | 농약으로서의 안트라닐산 디아미드 유도체 |
| EP2668153B1 (en) | 2011-01-28 | 2015-03-04 | E.I. Du Pont De Nemours And Company | Method for preparing 2-aminobenzamide derivatives |
| EP2606732A1 (en) | 2011-12-19 | 2013-06-26 | Bayer CropScience AG | Use of an anthranilic diamide derivatives with heteroaromatic and heterocyclic substituents in combination with a biological control agent |
| IN2014CN04325A (enExample) | 2011-12-19 | 2015-09-04 | Bayer Cropscience Ag | |
| WO2014089364A1 (en) | 2012-12-06 | 2014-06-12 | Quanticel Pharmaceuticals, Inc | Histone demethylase inhibitors |
| BR112015020830A2 (pt) | 2013-03-06 | 2017-07-18 | Bayer Cropscience Ag | diamidas de ácido antranílico substituídas com alcoximino como pesticidas |
| US20160137624A1 (en) * | 2013-06-20 | 2016-05-19 | Basf Se | Process for preparing pyridylpyrazole compounds and derivatives thereof from pyridylhydrazine |
| CN103467380B (zh) * | 2013-09-29 | 2015-06-24 | 南开大学 | 一类取代苯基吡唑酰胺衍生物及其制备方法和应用 |
| LT3113772T (lt) | 2014-03-07 | 2020-12-28 | Biocryst Pharmaceuticals, Inc. | Trifluormetilo pakeistieji pirazolai kaip žmogaus plazmos kalikreino inhibitoriai |
| WO2018054807A1 (en) * | 2016-09-21 | 2018-03-29 | Bayer Cropscience Aktiengesellschaft | Process for preparing 3-fluoroalkyl-5-pyrazolecarboxylates and 3-fluoroalkyl-5-pyrazolecarboxylic acids |
| WO2019123194A1 (en) | 2017-12-20 | 2019-06-27 | Pi Industries Ltd. | Anthranilamides, their use as insecticide and processes for preparing the same. |
| US12024510B2 (en) | 2017-12-20 | 2024-07-02 | Pi Industries Ltd. | Pyrazolopyridine-diamides, their use as insecticide and processes for preparing the same |
| US12221436B2 (en) | 2018-01-30 | 2025-02-11 | Pi Industries Ltd. | Anthranilamides, their use as insecticide and processes for preparing the same |
| CN112119071B (zh) | 2018-05-21 | 2024-08-02 | Pi工业有限公司 | 制备邻甲酰氨基苯甲酰胺类化合物的方法 |
| IL279890B2 (en) | 2018-07-20 | 2024-02-01 | Pi Industries Ltd | A process for the preparation of enteric diamides |
| EP4010320A4 (en) | 2019-08-06 | 2023-08-16 | Biocryst Pharmaceuticals, Inc. | Process-scale synthesis of a plasma kallikrein inhibitor |
| US12010989B2 (en) | 2019-11-07 | 2024-06-18 | S. C. Johnson & Son, Inc. | Roach gel formulations |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL279140A (enExample) | 1961-05-31 | |||
| ATE57690T1 (de) | 1987-01-05 | 1990-11-15 | Du Pont | Pyrazolin mit insektizidischer aktivitaet. |
| US5091405A (en) | 1987-01-05 | 1992-02-25 | E. I. Du Pont De Nemours And Company | Insecticidal pyrazolines |
| DE3808896A1 (de) | 1988-03-17 | 1989-09-28 | Hoechst Ag | Pflanzenschuetzende mittel auf basis von pyrazolcarbonsaeurederivaten |
| NL9202078A (nl) * | 1992-11-30 | 1994-06-16 | Rijkslandbouwhogeschool | Nieuwe N-acyl-antranilzuurverbindingen en toepassing van N-acyl-antranilzuurverbindingen bij de bestrijding van insecten. |
| US5945641A (en) * | 1998-07-15 | 1999-08-31 | Shieh; Woei-Kang | Stethoscope structure |
| KR100659007B1 (ko) | 1999-02-10 | 2007-02-28 | 미츠비시 웰파마 가부시키가이샤 | 아미드 화합물 및 그 의약으로서의 용도 |
| DE19951360A1 (de) * | 1999-10-26 | 2001-05-03 | Aventis Pharma Gmbh | Substituierte Indole |
| MY138097A (en) * | 2000-03-22 | 2009-04-30 | Du Pont | Insecticidal anthranilamides |
| JP2004515543A (ja) | 2000-12-11 | 2004-05-27 | イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー | 有害無脊椎動物を防除するためのキナゾリノン類およびピリジニルピリミジノン類 |
| EP1341780A2 (en) | 2000-12-11 | 2003-09-10 | E. I. du Pont de Nemours and Company | Substituted heterocyclic phthalic acid diamide arthropodicides |
| TWI356822B (en) | 2001-08-13 | 2012-01-21 | Du Pont | Novel substituted dihydro 3-halo-1h-pyrazole-5-car |
| AR036872A1 (es) | 2001-08-13 | 2004-10-13 | Du Pont | Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados |
| US7038057B2 (en) * | 2001-08-13 | 2006-05-02 | E.I. Du Pont De Nemours And Company | Substituted 1H-dihydropyrazoles, their preparation and use |
| ES2319743T3 (es) | 2001-08-16 | 2009-05-12 | E.I. Du Pont De Nemours And Company | Antranilamidas sustituidas para controlar plagas de invertebrados. |
| US20040110777A1 (en) | 2001-12-03 | 2004-06-10 | Annis Gary David | Quinazolinones and pyridinylpyrimidinones for controlling invertebrate pests |
| US20040063738A1 (en) * | 2001-12-05 | 2004-04-01 | Lahm George Philip | Substituted heterocyclic phthalic acid diamide arthropodicides |
| TW200401641A (en) * | 2002-07-18 | 2004-02-01 | Wyeth Corp | 1-Heterocyclylalkyl-3-sulfonylindole or-indazole derivatives as 5-hydroxytryptamine-6 ligands |
| TWI343376B (en) * | 2002-07-31 | 2011-06-11 | Du Pont | Method for preparing 3-halo-4, 5-dihydro-1h-pyrazoles |
| GB0409785D0 (en) | 2004-04-30 | 2004-06-09 | Resolution Chemicals Ltd | Preparation of cabergoline |
-
2002
- 2002-08-13 US US10/482,556 patent/US7038057B2/en not_active Expired - Fee Related
- 2002-08-13 AT AT02750482T patent/ATE469892T1/de not_active IP Right Cessation
- 2002-08-13 JP JP2003521208A patent/JP4448327B2/ja not_active Expired - Fee Related
- 2002-08-13 CA CA002454298A patent/CA2454298A1/en not_active Abandoned
- 2002-08-13 AU AU2002319814A patent/AU2002319814A1/en not_active Abandoned
- 2002-08-13 WO PCT/US2002/025612 patent/WO2003016282A2/en not_active Ceased
- 2002-08-13 EP EP02750482A patent/EP1417200B1/en not_active Expired - Lifetime
- 2002-08-13 DE DE60236600T patent/DE60236600D1/de not_active Expired - Lifetime
-
2006
- 2006-02-13 US US11/352,805 patent/US7622595B2/en not_active Expired - Fee Related
-
2009
- 2009-10-13 US US12/578,227 patent/US7932395B2/en not_active Expired - Fee Related
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