JP2005507873A5 - - Google Patents
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- Publication number
- JP2005507873A5 JP2005507873A5 JP2003521208A JP2003521208A JP2005507873A5 JP 2005507873 A5 JP2005507873 A5 JP 2005507873A5 JP 2003521208 A JP2003521208 A JP 2003521208A JP 2003521208 A JP2003521208 A JP 2003521208A JP 2005507873 A5 JP2005507873 A5 JP 2005507873A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- compound
- formula
- haloalkyl
- independently
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 claims description 40
- 229910052739 hydrogen Inorganic materials 0.000 claims description 21
- 238000000034 method Methods 0.000 claims description 21
- 229910052794 bromium Inorganic materials 0.000 claims description 16
- 229910052801 chlorine Inorganic materials 0.000 claims description 16
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims description 15
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims description 10
- 229910052736 halogen Inorganic materials 0.000 claims description 10
- 150000002367 halogens Chemical class 0.000 claims description 10
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 claims description 6
- 125000004768 (C1-C4) alkylsulfinyl group Chemical group 0.000 claims description 5
- 125000004769 (C1-C4) alkylsulfonyl group Chemical group 0.000 claims description 5
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims description 5
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims description 5
- 125000006656 (C2-C4) alkenyl group Chemical group 0.000 claims description 5
- 125000006650 (C2-C4) alkynyl group Chemical group 0.000 claims description 5
- 125000006643 (C2-C6) haloalkenyl group Chemical group 0.000 claims description 5
- -1 C 1 -C 4 alkylthio Chemical group 0.000 claims description 5
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims description 5
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims description 5
- 125000000217 alkyl group Chemical group 0.000 claims description 5
- 125000006310 cycloalkyl amino group Chemical group 0.000 claims description 5
- 125000004663 dialkyl amino group Chemical group 0.000 claims description 5
- 125000004473 dialkylaminocarbonyl group Chemical group 0.000 claims description 5
- 238000004519 manufacturing process Methods 0.000 claims description 4
- 150000004703 alkoxides Chemical class 0.000 claims description 3
- 230000002152 alkylating effect Effects 0.000 claims description 3
- 239000003795 chemical substances by application Substances 0.000 claims description 3
- 239000002253 acid Substances 0.000 claims description 2
- 230000015572 biosynthetic process Effects 0.000 description 1
- 229910052731 fluorine Inorganic materials 0.000 description 1
- 229910052740 iodine Inorganic materials 0.000 description 1
- 125000001453 quaternary ammonium group Chemical group 0.000 description 1
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US31191901P | 2001-08-13 | 2001-08-13 | |
| US34189401P | 2001-12-19 | 2001-12-19 | |
| US36965902P | 2002-04-02 | 2002-04-02 | |
| PCT/US2002/025612 WO2003016282A2 (en) | 2001-08-13 | 2002-08-13 | Substituted 1h-dihydropyrazoles, their preparation and use |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005507873A JP2005507873A (ja) | 2005-03-24 |
| JP2005507873A5 true JP2005507873A5 (enExample) | 2006-01-05 |
| JP4448327B2 JP4448327B2 (ja) | 2010-04-07 |
Family
ID=27405543
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003521208A Expired - Fee Related JP4448327B2 (ja) | 2001-08-13 | 2002-08-13 | 新規置換１ｈ−ジヒドロピラゾール、それらの製造および使用 |
Country Status (8)
| Country | Link |
|---|---|
| US (3) | US7038057B2 (enExample) |
| EP (1) | EP1417200B1 (enExample) |
| JP (1) | JP4448327B2 (enExample) |
| AT (1) | ATE469892T1 (enExample) |
| AU (1) | AU2002319814A1 (enExample) |
| CA (1) | CA2454298A1 (enExample) |
| DE (1) | DE60236600D1 (enExample) |
| WO (1) | WO2003016282A2 (enExample) |
Families Citing this family (67)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI312274B (en) | 2001-08-13 | 2009-07-21 | Du Pont | Method for controlling particular insect pests by applying anthranilamide compounds |
| TWI356822B (en) | 2001-08-13 | 2012-01-21 | Du Pont | Novel substituted dihydro 3-halo-1h-pyrazole-5-car |
| EP1417200B1 (en) * | 2001-08-13 | 2010-06-02 | E.I. Du Pont De Nemours And Company | Substituted 1h-dihydropyrazoles, their preparation and use |
| AR036872A1 (es) * | 2001-08-13 | 2004-10-13 | Du Pont | Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados |
| RU2283839C2 (ru) * | 2001-08-15 | 2006-09-20 | Е.И.Дюпон Де Немур Энд Компани | Ортозамещенные ариламиды, способ борьбы с насекомыми, композиция для борьбы с насекомыми, промежуточное соединение |
| ATE417829T1 (de) * | 2001-08-16 | 2009-01-15 | Du Pont | Substituierte anthranilamide und ihre verwendung als pesticide |
| TW200724033A (en) * | 2001-09-21 | 2007-07-01 | Du Pont | Anthranilamide arthropodicide treatment |
| US20040110777A1 (en) * | 2001-12-03 | 2004-06-10 | Annis Gary David | Quinazolinones and pyridinylpyrimidinones for controlling invertebrate pests |
| KR101011837B1 (ko) * | 2002-01-22 | 2011-01-31 | 이 아이 듀폰 디 네모아 앤드 캄파니 | 무척추 해충 방제를 위한 퀴나졸린(디)온 |
| BR0311707A (pt) * | 2002-06-13 | 2005-03-15 | Du Pont | Composto, composição e método de controle de pelo menos uma praga invertebrada |
| TWI326283B (en) * | 2002-07-31 | 2010-06-21 | Du Pont | Method for preparing fused oxazinones |
| US7666882B2 (en) * | 2002-11-15 | 2010-02-23 | E.I. Du Pont De Nemours And Company | Anthranilamide insecticides |
| PT1599463E (pt) | 2003-01-28 | 2013-09-03 | Du Pont | Insecticidas à base de ciano-antranilamida |
| TWI367882B (en) * | 2003-03-26 | 2012-07-11 | Du Pont | Preparation and use of 2-substituted-5-oxo-3-pyrazolidinecarboxylates |
| EP1631564A1 (en) * | 2003-06-12 | 2006-03-08 | E.I. Dupont De Nemours And Company | Method for preparing fused oxazinones |
| DE102004021564A1 (de) | 2003-11-14 | 2005-07-07 | Bayer Cropscience Ag | Wirkstoffkombinationen mit insektiziden Eigenschaften |
| DE10353281A1 (de) | 2003-11-14 | 2005-06-16 | Bayer Cropscience Ag | Wirkstoffkombination mit insektiziden und akariziden Eigenschaften |
| DE102004006075A1 (de) | 2003-11-14 | 2005-06-16 | Bayer Cropscience Ag | Wirkstoffkombinationen mit insektiziden Eigenschaften |
| DE10356550A1 (de) | 2003-12-04 | 2005-07-07 | Bayer Cropscience Ag | Wirkstoffkombinationen mit insektiziden Eigenschaften |
| CA2547989C (en) | 2003-12-04 | 2012-10-09 | Bayer Cropscience Ag | Active substance combinations having insecticidal properties |
| WO2005118552A2 (en) * | 2004-04-13 | 2005-12-15 | E.I. Dupont De Nemours And Company | Anthranilamide insecticides |
| DE102004031100A1 (de) * | 2004-06-28 | 2006-01-12 | Bayer Cropscience Ag | Anthranilamide |
| GT200500179AA (es) * | 2004-07-01 | 2008-10-29 | Mezclas sinergistas de agentes de antranilamida para el control de plagas de invertebrados | |
| JP4920878B2 (ja) * | 2004-07-14 | 2012-04-18 | 日本電気株式会社 | 認証システム、ネットワーク集線装置及びそれらに用いる認証方法並びにそのプログラム |
| DE102004035134A1 (de) | 2004-07-20 | 2006-02-16 | Bayer Cropscience Ag | Selektive Insektizide auf Basis von Halogenalkylnicotinsäurederivaten, Anthranilsäureamiden oder Phthalsäurediamiden und Safenern |
| MY140912A (en) * | 2004-07-26 | 2010-01-29 | Du Pont | Mixtures of anthranilamide invertebrate pest control agents |
| AU2005306363B2 (en) * | 2004-11-18 | 2012-08-09 | E. I. Du Pont De Nemours And Company | Anthranilamide insecticides |
| EP1924575A1 (en) * | 2005-08-24 | 2008-05-28 | E.I.Du pont de nemours and company | Anthranilamides for controlling invertebrate pests |
| DE102005044108A1 (de) | 2005-09-15 | 2007-03-29 | Bayer Cropscience Ag | Dioxazin- und Oxdiazin-substituierte Arylamide |
| DE102006032168A1 (de) | 2006-06-13 | 2007-12-20 | Bayer Cropscience Ag | Anthranilsäurediamid-Derivate mit heteroaromatischen Substituenten |
| DE102006030710A1 (de) * | 2006-07-03 | 2008-01-10 | Bayer Cropscience Ag | Synergistische insektizide und fungizide Mischungen |
| WO2008031548A1 (en) * | 2006-09-11 | 2008-03-20 | Syngenta Participations Ag | Process for the preparation of anthranilamide derivatives |
| CN101541178A (zh) * | 2006-11-17 | 2009-09-23 | 巴斯夫欧洲公司 | 提高植物干生物量的方法 |
| JP5507045B2 (ja) * | 2006-12-15 | 2014-05-28 | 石原産業株式会社 | アントラニルアミド系化合物の製造方法 |
| JP2009001541A (ja) * | 2006-12-15 | 2009-01-08 | Ishihara Sangyo Kaisha Ltd | 新規ピラゾール化合物を中間体として用いるアントラニルアミド系化合物の製造方法 |
| CN104496901B (zh) * | 2006-12-15 | 2016-05-25 | 石原产业株式会社 | 邻氨基苯甲酰胺系化合物的制造方法 |
| TWI415827B (zh) | 2006-12-21 | 2013-11-21 | Du Pont | 製備２-胺基-５-氰基苯甲酸衍生物之方法 |
| CA2842899C (en) * | 2007-04-25 | 2015-11-17 | Syngenta Participations Ag | Fungicidal compositions comprising a 3-substituted 1-methyl-1h-pyrazole-4-carboxylic acid (9-dihalomethylidene-benzonorbornene-5-yl) amide and a second fungicide |
| US8399490B2 (en) * | 2007-07-16 | 2013-03-19 | Syngenta Crop Protection Llc | Insecticides |
| EP2100883A1 (de) * | 2008-03-10 | 2009-09-16 | Bayer CropScience AG | Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4carbonsäure-Derivaten |
| CN102317279B (zh) | 2008-12-18 | 2015-03-04 | 拜尔农作物科学股份公司 | 作为杀虫剂的被四唑取代的邻氨基苯甲酰胺 |
| EP2243777A1 (de) | 2009-04-03 | 2010-10-27 | Bayer CropScience AG | Verfahren zum Herstellen von Pyridyl-substituierten Pyrazolen |
| EP2456760B1 (de) | 2009-07-23 | 2014-05-07 | Bayer CropScience AG | Verfahren zum herstellen von aryl-substituierten pyrazolen |
| CN102753531B (zh) | 2009-12-15 | 2015-07-01 | 拜尔农作物科学股份公司 | 制备1-烷基-/1-芳基-5-吡唑羧酸衍生物的方法 |
| WO2011098408A2 (de) | 2010-02-09 | 2011-08-18 | Bayer Cropscience Ag | Hydrazin-substituierte anthranilsäurederivate |
| EP2558460B1 (de) | 2010-04-16 | 2015-03-04 | Bayer Intellectual Property GmbH | Triazolsubstituierte anthranilsäureamide als pestizide |
| EP2582695B1 (de) | 2010-06-15 | 2015-09-30 | Bayer Intellectual Property GmbH | Anthranilsäurediamid-derivate mit zyklischen seitenketten |
| CN103068814B (zh) | 2010-06-15 | 2015-11-25 | 拜耳知识产权有限责任公司 | 邻氨基苯甲酸衍生物 |
| ES2575566T3 (es) | 2010-06-15 | 2016-06-29 | Bayer Intellectual Property Gmbh | Nuevos derivados de arilamida orto-sustituidos |
| MX2012014958A (es) | 2010-06-15 | 2013-02-12 | Bayer Ip Gmbh | Derivados de diamida antranilica. |
| JP5926253B2 (ja) | 2010-07-09 | 2016-05-25 | バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ ＧｍｂＨ | 有害生物駆除剤としてのアントラニルアミド誘導体 |
| HUE025309T2 (en) | 2011-01-28 | 2016-01-28 | Du Pont | Process for the preparation of 2-aminobenzamide derivatives |
| CA2859467C (en) | 2011-12-19 | 2019-10-01 | Bayer Cropscience Ag | Use of anthranilic acid diamide derivatives for pest control in transgenic crops |
| EP2606732A1 (en) | 2011-12-19 | 2013-06-26 | Bayer CropScience AG | Use of an anthranilic diamide derivatives with heteroaromatic and heterocyclic substituents in combination with a biological control agent |
| EP3763367A1 (en) | 2012-12-06 | 2021-01-13 | Celgene Quanticel Research, Inc. | Pyridine-pyrazole derivatives as histone demethylase inhibitors |
| MX2015011423A (es) | 2013-03-06 | 2016-02-03 | Bayer Cropscience Ag | Diamidas de acido antranilico sustituidas con alcoximino como pesticidas. |
| JP2016522234A (ja) * | 2013-06-20 | 2016-07-28 | ビーエーエスエフ ソシエタス・ヨーロピアＢａｓｆ Ｓｅ | ピリジルヒドラジンからピリジルピラゾール化合物及びその誘導体を製造するための方法 |
| CN103467380B (zh) * | 2013-09-29 | 2015-06-24 | 南开大学 | 一类取代苯基吡唑酰胺衍生物及其制备方法和应用 |
| LT3828173T (lt) | 2014-03-07 | 2022-11-10 | Biocryst Pharmaceuticals, Inc. | Pakeistieji pirazolai kaip žmogaus plazmos kalikreino inhibitoriai |
| JP7044766B2 (ja) | 2016-09-21 | 2022-03-30 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | ３－フルオロアルキル－５－ピラゾールカルボキシレート類及び３－フルオロアルキル－５－ピラゾールカルボン酸類を調製する方法 |
| JP7403454B2 (ja) | 2017-12-20 | 2023-12-22 | ピーアイ インダストリーズ リミテッド | ピラゾロピリジン－ジアミド、殺虫剤としてのそれらの使用およびそれらの製造方法 |
| WO2019123194A1 (en) | 2017-12-20 | 2019-06-27 | Pi Industries Ltd. | Anthranilamides, their use as insecticide and processes for preparing the same. |
| CA3090764A1 (en) | 2018-01-30 | 2019-08-08 | Pi Industries Ltd | Novel anthranilamides, their use as insecticide and processes for preparing the same |
| KR102760014B1 (ko) | 2018-05-21 | 2025-01-24 | 피아이 인더스트리스 엘티디. | 안트라닐산 디아미드의 새로운 제조 방법 |
| IL279890B2 (en) | 2018-07-20 | 2024-02-01 | Pi Industries Ltd | A process for the preparation of enteric diamides |
| BR112022002060A2 (pt) * | 2019-08-06 | 2022-06-07 | Biocryst Pharm Inc | Síntese de escala de processo de um inibidor de calicreína de plasma |
| US12010989B2 (en) | 2019-11-07 | 2024-06-18 | S. C. Johnson & Son, Inc. | Roach gel formulations |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL121416C (enExample) | 1961-05-31 | |||
| US5091405A (en) | 1987-01-05 | 1992-02-25 | E. I. Du Pont De Nemours And Company | Insecticidal pyrazolines |
| WO1988006583A1 (en) | 1987-01-05 | 1988-09-07 | E.I. Du Pont De Nemours And Company | Insecticidal pyrazolines |
| DE3808896A1 (de) | 1988-03-17 | 1989-09-28 | Hoechst Ag | Pflanzenschuetzende mittel auf basis von pyrazolcarbonsaeurederivaten |
| NL9202078A (nl) * | 1992-11-30 | 1994-06-16 | Rijkslandbouwhogeschool | Nieuwe N-acyl-antranilzuurverbindingen en toepassing van N-acyl-antranilzuurverbindingen bij de bestrijding van insecten. |
| US5945641A (en) * | 1998-07-15 | 1999-08-31 | Shieh; Woei-Kang | Stethoscope structure |
| US7015218B1 (en) | 1999-02-10 | 2006-03-21 | Mitsubishi Pharma Corporation | Amide compounds and medicinal use thereof |
| DE19951360A1 (de) * | 1999-10-26 | 2001-05-03 | Aventis Pharma Gmbh | Substituierte Indole |
| MY138097A (en) | 2000-03-22 | 2009-04-30 | Du Pont | Insecticidal anthranilamides |
| AU2002227243A1 (en) | 2000-12-11 | 2002-06-24 | E.I. Du Pont De Nemours And Company | Quinazolinones and pyridinopyrimidinones for controlling invertebrate pests |
| JP2004515547A (ja) | 2000-12-11 | 2004-05-27 | イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー | 置換複素環式フタル酸ジアミド殺節足動物剤 |
| EP1417200B1 (en) * | 2001-08-13 | 2010-06-02 | E.I. Du Pont De Nemours And Company | Substituted 1h-dihydropyrazoles, their preparation and use |
| AR036872A1 (es) | 2001-08-13 | 2004-10-13 | Du Pont | Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados |
| TWI356822B (en) | 2001-08-13 | 2012-01-21 | Du Pont | Novel substituted dihydro 3-halo-1h-pyrazole-5-car |
| ATE417829T1 (de) | 2001-08-16 | 2009-01-15 | Du Pont | Substituierte anthranilamide und ihre verwendung als pesticide |
| US20040110777A1 (en) | 2001-12-03 | 2004-06-10 | Annis Gary David | Quinazolinones and pyridinylpyrimidinones for controlling invertebrate pests |
| US20040063738A1 (en) * | 2001-12-05 | 2004-04-01 | Lahm George Philip | Substituted heterocyclic phthalic acid diamide arthropodicides |
| TW200401641A (en) | 2002-07-18 | 2004-02-01 | Wyeth Corp | 1-Heterocyclylalkyl-3-sulfonylindole or-indazole derivatives as 5-hydroxytryptamine-6 ligands |
| TWI343376B (en) * | 2002-07-31 | 2011-06-11 | Du Pont | Method for preparing 3-halo-4, 5-dihydro-1h-pyrazoles |
| GB0409785D0 (en) | 2004-04-30 | 2004-06-09 | Resolution Chemicals Ltd | Preparation of cabergoline |
-
2002
- 2002-08-13 EP EP02750482A patent/EP1417200B1/en not_active Expired - Lifetime
- 2002-08-13 CA CA002454298A patent/CA2454298A1/en not_active Abandoned
- 2002-08-13 WO PCT/US2002/025612 patent/WO2003016282A2/en not_active Ceased
- 2002-08-13 JP JP2003521208A patent/JP4448327B2/ja not_active Expired - Fee Related
- 2002-08-13 AT AT02750482T patent/ATE469892T1/de not_active IP Right Cessation
- 2002-08-13 AU AU2002319814A patent/AU2002319814A1/en not_active Abandoned
- 2002-08-13 DE DE60236600T patent/DE60236600D1/de not_active Expired - Lifetime
- 2002-08-13 US US10/482,556 patent/US7038057B2/en not_active Expired - Fee Related
-
2006
- 2006-02-13 US US11/352,805 patent/US7622595B2/en not_active Expired - Fee Related
-
2009
- 2009-10-13 US US12/578,227 patent/US7932395B2/en not_active Expired - Fee Related
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