JP2005506292A5 - - Google Patents

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Publication number
JP2005506292A5
JP2005506292A5 JP2002571458A JP2002571458A JP2005506292A5 JP 2005506292 A5 JP2005506292 A5 JP 2005506292A5 JP 2002571458 A JP2002571458 A JP 2002571458A JP 2002571458 A JP2002571458 A JP 2002571458A JP 2005506292 A5 JP2005506292 A5 JP 2005506292A5
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JP
Japan
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lower alkyl
group
independently
alkyl
aryl
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JP2002571458A
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English (en)
Japanese (ja)
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JP2005506292A (ja
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Priority claimed from PCT/US2002/007033 external-priority patent/WO2002072542A2/en
Publication of JP2005506292A publication Critical patent/JP2005506292A/ja
Publication of JP2005506292A5 publication Critical patent/JP2005506292A5/ja
Pending legal-status Critical Current

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JP2002571458A 2001-03-08 2002-03-08 ｐＨに依存するＮＭＤＡレセプターアンタゴニスト Pending JP2005506292A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US27420501P 2001-03-08 2001-03-08
PCT/US2002/007033 WO2002072542A2 (en) 2001-03-08 2002-03-08 Ph-dependent nmda receptor antagonists

Publications (2)

Publication Number Publication Date
JP2005506292A JP2005506292A (ja) 2005-03-03
JP2005506292A5 true JP2005506292A5 (https=) 2007-12-20

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Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002571458A Pending JP2005506292A (ja) 2001-03-08 2002-03-08 ｐＨに依存するＮＭＤＡレセプターアンタゴニスト

Country Status (6)

Country Link
US (2) US7375136B2 (https=)
EP (1) EP1436258A4 (https=)
JP (1) JP2005506292A (https=)
AU (1) AU2002250256B2 (https=)
CA (1) CA2440284A1 (https=)
WO (1) WO2002072542A2 (https=)

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JP5934645B2 (ja) 2009-09-11 2016-06-15 プロビオドルグ エージー グルタミニルシクラーゼ阻害剤としてのヘテロ環式誘導体
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WO2011107530A2 (en) 2010-03-03 2011-09-09 Probiodrug Ag Novel inhibitors
JP5688745B2 (ja) 2010-03-10 2015-03-25 プロビオドルグ エージー グルタミニルシクラーゼ（ｑｃ、ｅｃ２．３．２．５）の複素環阻害剤
WO2011131748A2 (en) 2010-04-21 2011-10-27 Probiodrug Ag Novel inhibitors
EP2686313B1 (en) 2011-03-16 2016-02-03 Probiodrug AG Benzimidazole derivatives as inhibitors of glutaminyl cyclase
CN104490872A (zh) * 2014-12-11 2015-04-08 温州医科大学附属第一医院 2-(2-苯并呋喃基)-2-咪唑啉治疗神经系统线粒体损伤疾病中的用途
EP3383429B1 (en) 2015-11-30 2020-10-14 INSERM - Institut National de la Santé et de la Recherche Médicale Nmdar antagonists for the treatment of tumor angiogenesis
ES2812698T3 (es) 2017-09-29 2021-03-18 Probiodrug Ag Inhibidores de glutaminil ciclasa
CN114616230A (zh) 2019-07-31 2022-06-10 海洋生物技术与海洋资源有限公司 黄烷类似物化合物及其在治疗慢性和急性疼痛中的用途
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CN118019541A (zh) 2021-09-02 2024-05-10 埃默里大学 在酸性pH下具有增强的效力的N-甲基-D-天冬氨酸受体的GLUN2B-亚基选择性拮抗剂

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