JP2004534057A5 - - Google Patents

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Publication number
JP2004534057A5
JP2004534057A5 JP2003503214A JP2003503214A JP2004534057A5 JP 2004534057 A5 JP2004534057 A5 JP 2004534057A5 JP 2003503214 A JP2003503214 A JP 2003503214A JP 2003503214 A JP2003503214 A JP 2003503214A JP 2004534057 A5 JP2004534057 A5 JP 2004534057A5
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JP
Japan
Prior art keywords
dosage form
prodrug
auc
gaba analog
hours
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2003503214A
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English (en)
Japanese (ja)
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JP2004534057A (ja
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Priority claimed from PCT/US2002/018701 external-priority patent/WO2002100392A1/en
Publication of JP2004534057A publication Critical patent/JP2004534057A/ja
Publication of JP2004534057A5 publication Critical patent/JP2004534057A5/ja
Pending legal-status Critical Current

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JP2003503214A 2001-06-11 2002-06-11 低毒性を示す経口投与剤形のgaba類似体プロドラッグ Pending JP2004534057A (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US29752101P 2001-06-11 2001-06-11
US29851401P 2001-06-14 2001-06-14
US36609002P 2002-03-19 2002-03-19
PCT/US2002/018701 WO2002100392A1 (en) 2001-06-11 2002-06-11 Orally administered dosage forms of gaba analog prodrugs having reduced toxicity

Publications (2)

Publication Number Publication Date
JP2004534057A JP2004534057A (ja) 2004-11-11
JP2004534057A5 true JP2004534057A5 (enExample) 2005-12-22

Family

ID=27404495

Family Applications (4)

Application Number Title Priority Date Filing Date
JP2003516067A Expired - Lifetime JP4216713B2 (ja) 2001-06-11 2002-06-11 Gaba類似体のプロドラッグ、組成物およびその使用
JP2003503214A Pending JP2004534057A (ja) 2001-06-11 2002-06-11 低毒性を示す経口投与剤形のgaba類似体プロドラッグ
JP2008171250A Withdrawn JP2009051822A (ja) 2001-06-11 2008-06-30 Gaba類似体のプロドラッグ、組成物およびその使用
JP2008171589A Expired - Lifetime JP5001227B2 (ja) 2001-06-11 2008-06-30 Gaba類似体のプロドラッグ、組成物およびその使用

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2003516067A Expired - Lifetime JP4216713B2 (ja) 2001-06-11 2002-06-11 Gaba類似体のプロドラッグ、組成物およびその使用

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2008171250A Withdrawn JP2009051822A (ja) 2001-06-11 2008-06-30 Gaba類似体のプロドラッグ、組成物およびその使用
JP2008171589A Expired - Lifetime JP5001227B2 (ja) 2001-06-11 2008-06-30 Gaba類似体のプロドラッグ、組成物およびその使用

Country Status (20)

Country Link
US (2) US6833140B2 (enExample)
EP (4) EP1404310A4 (enExample)
JP (4) JP4216713B2 (enExample)
KR (5) KR20090121404A (enExample)
CN (1) CN1533270A (enExample)
AT (2) ATE540678T1 (enExample)
AU (4) AU2002345664C1 (enExample)
CA (2) CA2449729C (enExample)
CY (1) CY1107894T1 (enExample)
DE (1) DE60223923T3 (enExample)
DK (1) DK1404324T4 (enExample)
ES (2) ES2296956T5 (enExample)
HU (2) HUP0400167A3 (enExample)
IL (5) IL159299A0 (enExample)
MX (2) MXPA03011566A (enExample)
NO (4) NO20035473D0 (enExample)
NZ (1) NZ567711A (enExample)
PT (1) PT1404324E (enExample)
WO (2) WO2002100347A2 (enExample)
ZA (1) ZA200309679B (enExample)

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