JP2003529592A - 結晶性医薬 - Google Patents

結晶性医薬

Info

Publication number
JP2003529592A
JP2003529592A JP2001572482A JP2001572482A JP2003529592A JP 2003529592 A JP2003529592 A JP 2003529592A JP 2001572482 A JP2001572482 A JP 2001572482A JP 2001572482 A JP2001572482 A JP 2001572482A JP 2003529592 A JP2003529592 A JP 2003529592A
Authority
JP
Japan
Prior art keywords
lopinavir
solid
crystalline form
infrared spectrum
peak
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2001572482A
Other languages
English (en)
Japanese (ja)
Inventor
デイツクマン，ダニエル・エイ
チエンブルカール，サンジヤイ
フオート，ジエイムズ・ジエイ
ヘンリー，ロジヤー・エフ
レチユガ−バレステロス，デイビツド
ニウ，ユイピン
ポーター，ウイリアム
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Abbott Laboratories
Original Assignee
Abbott Laboratories
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27065762&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JP2003529592(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US09/793,536 external-priority patent/US6608198B2/en
Application filed by Abbott Laboratories filed Critical Abbott Laboratories
Publication of JP2003529592A publication Critical patent/JP2003529592A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/06—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D239/08—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms directly attached in position 2
    • C07D239/10—Oxygen or sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Virology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • AIDS & HIV (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2001572482A 2000-03-30 2001-03-21 結晶性医薬 Pending JP2003529592A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US53825700A 2000-03-30 2000-03-30
US09/538,257 2000-03-30
US09/793,536 2001-02-27
US09/793,536 US6608198B2 (en) 2000-03-30 2001-02-27 Crystalline pharmaceutical
PCT/US2001/009112 WO2001074787A2 (en) 2000-03-30 2001-03-21 Crystalline pharmaceutical

Publications (1)

Publication Number Publication Date
JP2003529592A true JP2003529592A (ja) 2003-10-07

Family

ID=27065762

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2001572482A Pending JP2003529592A (ja) 2000-03-30 2001-03-21 結晶性医薬

Country Status (22)

Country Link
EP (1) EP1268442A2 (no)
JP (1) JP2003529592A (no)
KR (1) KR100773258B1 (no)
CN (2) CN1330639C (no)
AR (2) AR033360A1 (no)
AU (3) AU5092001A (no)
BG (1) BG107165A (no)
BR (1) BR0109433A (no)
CA (1) CA2403635A1 (no)
CZ (1) CZ20023529A3 (no)
HU (1) HUP0302675A3 (no)
IL (1) IL151551A0 (no)
MX (1) MXPA02009559A (no)
MY (1) MY128296A (no)
NO (1) NO325005B1 (no)
NZ (1) NZ521183A (no)
PE (1) PE20011232A1 (no)
PL (1) PL359727A1 (no)
SA (2) SA06270303B1 (no)
SK (1) SK14832002A3 (no)
TW (1) TWI284640B (no)
WO (1) WO2001074787A2 (no)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2013503176A (ja) * 2009-08-27 2013-01-31 メルク・シャープ・エンド・ドーム・コーポレイション Ｃ型肝炎ウイルスのプロテアーゼ阻害薬の調製方法

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6608198B2 (en) 2000-03-30 2003-08-19 Abbott Laboratories Crystalline pharmaceutical
US8025899B2 (en) 2003-08-28 2011-09-27 Abbott Laboratories Solid pharmaceutical dosage form
ES2459301T3 (es) * 2009-02-06 2014-05-08 Hetero Research Foundation Nuevos polimorfos de lopinavir
CN112830899A (zh) * 2021-01-18 2021-05-25 合肥华方医药科技有限公司 一种洛匹那韦新晶型及其制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5914332A (en) 1995-12-13 1999-06-22 Abbott Laboratories Retroviral protease inhibiting compounds
WO1998057648A1 (en) * 1997-06-16 1998-12-23 Vertex Pharmaceuticals Incorporated Methods of increasing the bioavailability of stable crystal polymorphs of a compound

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2013503176A (ja) * 2009-08-27 2013-01-31 メルク・シャープ・エンド・ドーム・コーポレイション Ｃ型肝炎ウイルスのプロテアーゼ阻害薬の調製方法

Also Published As

Publication number Publication date
AR049560A2 (es) 2006-08-16
CN101066952A (zh) 2007-11-07
CZ20023529A3 (cs) 2003-02-12
BR0109433A (pt) 2004-08-10
NO20024679L (no) 2002-09-30
SA01220270B1 (ar) 2006-11-14
HUP0302675A3 (en) 2004-03-29
TWI284640B (en) 2007-08-01
NZ521183A (en) 2004-03-26
WO2001074787A2 (en) 2001-10-11
CA2403635A1 (en) 2001-10-11
PE20011232A1 (es) 2001-12-08
MY128296A (en) 2007-01-31
AU2006222711A1 (en) 2006-10-19
NO325005B1 (no) 2008-01-14
WO2001074787A3 (en) 2002-02-07
SA06270303B1 (ar) 2009-08-02
IL151551A0 (en) 2003-04-10
MXPA02009559A (es) 2003-05-21
CN1422259A (zh) 2003-06-04
CN1330639C (zh) 2007-08-08
AU2001250920B2 (en) 2006-06-29
KR20030011807A (ko) 2003-02-11
EP1268442A2 (en) 2003-01-02
NO20024679D0 (no) 2002-09-30
PL359727A1 (en) 2004-09-06
KR100773258B1 (ko) 2007-11-05
BG107165A (bg) 2003-07-31
AU5092001A (en) 2001-10-15
SK14832002A3 (sk) 2003-02-04
AR033360A1 (es) 2003-12-17
HUP0302675A2 (hu) 2003-12-29

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