JP2003511453A5 - - Google Patents
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- Publication number
- JP2003511453A5 JP2003511453A5 JP2001530331A JP2001530331A JP2003511453A5 JP 2003511453 A5 JP2003511453 A5 JP 2003511453A5 JP 2001530331 A JP2001530331 A JP 2001530331A JP 2001530331 A JP2001530331 A JP 2001530331A JP 2003511453 A5 JP2003511453 A5 JP 2003511453A5
- Authority
- JP
- Japan
- Prior art keywords
- ethyl
- alkyl
- ylsulfonyl
- pyrazolo
- dihydro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9924063.2A GB9924063D0 (en) | 1999-10-11 | 1999-10-11 | Pharmaceutically active compounds |
| GB9924063.2 | 1999-10-11 | ||
| GB0018656.9 | 2000-07-28 | ||
| GB0018656A GB0018656D0 (en) | 2000-07-28 | 2000-07-28 | Pharmaceutically active compounds |
| PCT/IB2000/001457 WO2001027113A2 (en) | 1999-10-11 | 2000-10-11 | PYRAZOLO `4,3-d! PYRIMIDINE DERIVATIVES |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2003511453A JP2003511453A (ja) | 2003-03-25 |
| JP2003511453A5 true JP2003511453A5 (https=) | 2006-01-05 |
| JP3834236B2 JP3834236B2 (ja) | 2006-10-18 |
Family
ID=26244757
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2001530331A Expired - Fee Related JP3834236B2 (ja) | 1999-10-11 | 2000-10-11 | ピラゾロ〔4,3−d〕ピリミジン誘導体 |
Country Status (48)
Families Citing this family (103)
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| JP3199115B2 (ja) * | 1998-12-24 | 2001-08-13 | モトローラ株式会社 | デジタル・アナログ変換回路 |
| DE19903087A1 (de) | 1999-01-27 | 2000-08-10 | Forssmann Wolf Georg | Behandlung von erektilen Dysfunktionen mit C-Typ Natriuretischem Polypeptid (CNP) als Monotherapie oder in Kombination mit Phosphodiesterasehemmern |
| WO2000053148A2 (en) | 1999-03-08 | 2000-09-14 | Merck & Co., Inc. | Methods and compositions for treating erectile dysfunction |
| IL137429A0 (en) | 1999-07-28 | 2001-07-24 | Pfizer Prod Inc | Methods and compsitions for treating diseases and conditions of the eye |
| AU5957600A (en) | 1999-07-30 | 2001-02-19 | Lakefield Minerals Ltd. | Pharmaceutical compositions for topical application to treat erectile dysfunction |
| AU779991B2 (en) | 1999-08-10 | 2005-02-24 | Board Of Regents, The University Of Texas System | Method for increasing optic nerve, choroidal and retinal blood flow to facilitate the preservation of sight |
| US6436944B1 (en) | 1999-09-30 | 2002-08-20 | Pfizer Inc. | Combination effective for the treatment of impotence |
| TWI265925B (en) | 1999-10-11 | 2006-11-11 | Pfizer | Pyrazolo[4,3-d]pyrimidin-7-ones useful in inhibiting type 5 cyclic guanosine 3',5'-monophosphate phosphodiesterases(cGMP PDE5), process and intermediates for their preparation, their uses and composition comprising them |
| YU59100A (sh) | 1999-10-11 | 2003-10-31 | Pfizer Inc. | Postupak za dobijanje pirazolo (4,3-d) pirimidin-7-ona-3-piridilsulfonil jedinjenja i njihova intermedijera |
| US6420557B1 (en) * | 2000-07-28 | 2002-07-16 | Pfizer Inc. | Crystalline therapeutic agent |
| US6407259B1 (en) * | 2000-07-28 | 2002-06-18 | Pfizer Inc. | Process for the preparation of pyrazoles |
-
2000
- 2000-09-14 TW TW089118861A patent/TWI265925B/zh not_active IP Right Cessation
- 2000-10-06 US US09/685,080 patent/US6677335B1/en not_active Expired - Fee Related
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- 2000-10-09 EG EG20001281A patent/EG24411A/xx active
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- 2000-10-11 KR KR1020027004643A patent/KR100549152B1/ko not_active Expired - Fee Related
- 2000-10-11 TR TR2002/00989T patent/TR200200989T2/xx unknown
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- 2000-10-11 JP JP2001530331A patent/JP3834236B2/ja not_active Expired - Fee Related
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- 2000-10-11 WO PCT/IB2000/001457 patent/WO2001027113A2/en not_active Ceased
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- 2000-10-11 DZ DZ003220A patent/DZ3220A1/fr active
- 2000-10-11 AU AU76784/00A patent/AU779065B2/en not_active Ceased
- 2000-10-11 SI SI200030593T patent/SI1220856T1/xx unknown
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