JP2002507576A5 - - Google Patents
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- Publication number
- JP2002507576A5 JP2002507576A5 JP2000537561A JP2000537561A JP2002507576A5 JP 2002507576 A5 JP2002507576 A5 JP 2002507576A5 JP 2000537561 A JP2000537561 A JP 2000537561A JP 2000537561 A JP2000537561 A JP 2000537561A JP 2002507576 A5 JP2002507576 A5 JP 2002507576A5
- Authority
- JP
- Japan
- Prior art keywords
- seq
- formula
- peptide
- fmoc
- side chain
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/045,920 US6281331B1 (en) | 1998-03-23 | 1998-03-23 | Methods and compositions for peptide synthesis |
| US09/045,920 | 1998-03-23 | ||
| US09/071,877 US6015881A (en) | 1998-03-23 | 1998-05-01 | Methods and compositions for peptide synthesis |
| US09/071,877 | 1998-05-01 | ||
| PCT/US1999/006230 WO1999048513A1 (en) | 1998-03-23 | 1999-03-22 | Methods and compositions for peptide synthesis |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009247579A Division JP4755713B2 (ja) | 1998-03-23 | 2009-10-28 | ペプチド合成のための方法および組成物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2002507576A JP2002507576A (ja) | 2002-03-12 |
| JP2002507576A5 true JP2002507576A5 (https=) | 2006-06-08 |
| JP4602547B2 JP4602547B2 (ja) | 2010-12-22 |
Family
ID=26723345
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2000537561A Expired - Fee Related JP4602547B2 (ja) | 1998-03-23 | 1999-03-22 | ペプチド合成のための方法および組成物 |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP1071442B9 (https=) |
| JP (1) | JP4602547B2 (https=) |
| CN (1) | CN100383158C (https=) |
| AT (1) | ATE299029T1 (https=) |
| AU (1) | AU751358B2 (https=) |
| BR (1) | BR9909018A (https=) |
| CA (1) | CA2324348C (https=) |
| DE (1) | DE69926061T2 (https=) |
| DK (1) | DK1071442T3 (https=) |
| ES (1) | ES2245505T3 (https=) |
| NZ (1) | NZ507083A (https=) |
| TW (1) | TWI233931B (https=) |
| WO (1) | WO1999048513A1 (https=) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6281331B1 (en) * | 1998-03-23 | 2001-08-28 | Trimeris, Inc. | Methods and compositions for peptide synthesis |
| US6469136B1 (en) | 1999-07-07 | 2002-10-22 | Trimeris, Inc. | Methods and composition for peptide synthesis |
| KR100614714B1 (ko) | 2001-06-15 | 2006-08-21 | 에프. 호프만-라 로슈 아게 | ｇｐ41 단편의 아세틸화 |
| HRP20050024A2 (en) * | 2002-07-24 | 2006-02-28 | F. Hoffmann - La Roche Ag | Pegylated t20 polypeptide |
| ATE410437T1 (de) | 2003-12-31 | 2008-10-15 | Hoffmann La Roche | Verfahren und systeme zur rückgewinnung von peptiden |
| ATE376556T1 (de) | 2003-12-31 | 2007-11-15 | Hoffmann La Roche | Verfahren zur peptidsynthese unter verwendung einer reduzierten menge an entschützungsmittel |
| EP1701976A2 (en) * | 2003-12-31 | 2006-09-20 | F.Hoffmann-La Roche Ag | Peptide synthesis and deprotection with co-solvent |
| JP4886702B2 (ja) * | 2004-12-30 | 2012-02-29 | エフ．ホフマン−ラ ロシュ アーゲー | ペプチド中間体断片を使用するペプチドｔ−２０の合成 |
| CA2651070A1 (en) | 2006-05-03 | 2007-11-15 | Mallinckrodt Inc. | Composition and method for the release of protected peptides from a resin |
| EP2181983A4 (en) * | 2007-07-25 | 2013-01-02 | Ajinomoto Kk | METHOD FOR THE SELECTIVE REMOVAL OF A DIBENZOFULVENE DERIVATIVE |
| CN101835794A (zh) * | 2007-10-27 | 2010-09-15 | 霍夫曼-拉罗奇有限公司 | 使用固相和溶液相组合技术的促胰岛素肽合成法 |
| EP2222695A2 (en) * | 2007-12-11 | 2010-09-01 | F. Hoffmann-La Roche AG | Insulinotropic peptide synthesis using solid and solution phase combination techniques |
| JP5445456B2 (ja) * | 2008-08-06 | 2014-03-19 | 味の素株式会社 | ジベンゾフルベンの除去方法 |
| US20100081788A1 (en) * | 2008-09-03 | 2010-04-01 | Scinopharm Taiwan Ltd. | Process for the Preparation of Pramlintide |
| US20110288235A1 (en) * | 2008-09-03 | 2011-11-24 | Scinopharm Taiwan Ltd. | Process for the Preparation of Pramlintide |
| WO2011095989A2 (en) * | 2010-02-04 | 2011-08-11 | Matrix Laboratories Ltd | An improved process for the preparation of enfuvirtide |
| PL219569B1 (pl) * | 2010-02-19 | 2015-05-29 | Peptaderm Spółka Z Ograniczoną Odpowiedzialnością | Cykliczne tetrapeptydy i ich zastosowanie |
| CN103374054B (zh) * | 2012-04-28 | 2014-12-24 | 上海第一生化药业有限公司 | 一步法固相合成多肽的方法 |
| GB201315335D0 (en) | 2013-08-29 | 2013-10-09 | Of Singapore | Amino diacids containing peptide modifiers |
| CN115298193B (zh) * | 2020-02-05 | 2026-03-31 | 伊莱利利公司 | 串联树脂反应器的肽合成仪 |
| CN114315957B (zh) * | 2021-12-30 | 2023-07-07 | 深圳瑞德林生物技术有限公司 | 一种多肽的制备方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1987007616A1 (en) * | 1986-06-12 | 1987-12-17 | Biogen N.V. | Peptides involved in the pathogenesis of hiv infection |
| US4787222A (en) * | 1986-11-24 | 1988-11-29 | Novatek Medical Inc. | Combination lock for blood identification system |
| US5444044A (en) * | 1992-03-26 | 1995-08-22 | New York Blood Center | Synthetic polypeptides as inhibitors of HIV-1 |
| WO1994028929A1 (en) * | 1993-06-07 | 1994-12-22 | Genentech, Inc. | Hiv envelope polypeptides |
| US6479055B1 (en) * | 1993-06-07 | 2002-11-12 | Trimeris, Inc. | Methods for inhibition of membrane fusion-associated events, including respiratory syncytial virus transmission |
| US5464933A (en) * | 1993-06-07 | 1995-11-07 | Duke University | Synthetic peptide inhibitors of HIV transmission |
| DE69426725T2 (de) * | 1993-09-11 | 2001-09-06 | Polimun Scientific Immunbiologische Forschungsgesellschaft Mbh, Wien | Peptide, die neutralisierende antikörper gegen genetisch divergierende hiv-1 stämme, induzieren |
| CN1186355C (zh) * | 1996-02-09 | 2005-01-26 | 霍夫曼-拉罗奇有限公司 | 血管活性肠肽类似物的合成 |
-
1999
- 1999-03-22 WO PCT/US1999/006230 patent/WO1999048513A1/en not_active Ceased
- 1999-03-22 DE DE69926061T patent/DE69926061T2/de not_active Expired - Lifetime
- 1999-03-22 DK DK99912802T patent/DK1071442T3/da active
- 1999-03-22 AU AU31097/99A patent/AU751358B2/en not_active Expired
- 1999-03-22 CN CNB998064319A patent/CN100383158C/zh not_active Expired - Fee Related
- 1999-03-22 JP JP2000537561A patent/JP4602547B2/ja not_active Expired - Fee Related
- 1999-03-22 BR BR9909018-0A patent/BR9909018A/pt not_active IP Right Cessation
- 1999-03-22 AT AT99912802T patent/ATE299029T1/de active
- 1999-03-22 NZ NZ507083A patent/NZ507083A/en not_active IP Right Cessation
- 1999-03-22 ES ES99912802T patent/ES2245505T3/es not_active Expired - Lifetime
- 1999-03-22 CA CA002324348A patent/CA2324348C/en not_active Expired - Lifetime
- 1999-03-22 EP EP99912802A patent/EP1071442B9/en not_active Expired - Lifetime
- 1999-03-23 TW TW088104562A patent/TWI233931B/zh not_active IP Right Cessation
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