JP2001510195A - 縮合化１，２，４−チアジアジン誘導体、その調製及び使用 - Google Patents

縮合化１，２，４−チアジアジン誘導体、その調製及び使用

Info

Publication number
JP2001510195A
JP2001510195A JP2000503085A JP2000503085A JP2001510195A JP 2001510195 A JP2001510195 A JP 2001510195A JP 2000503085 A JP2000503085 A JP 2000503085A JP 2000503085 A JP2000503085 A JP 2000503085A JP 2001510195 A JP2001510195 A JP 2001510195A
Authority
JP
Japan
Prior art keywords
alkyl
thiadiazine
dioxide
thieno
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2000503085A
Other languages
English (en)
Japanese (ja)
Inventor
エルメルン ニールセン，フレミン
ボンドー ハンセン，ヨーン
クラウス ハンセン，ホルゲー
メラー タグモセ，ティナ
パトリック モーゲンセン，ヨーン
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novo Nordisk AS
Original Assignee
Novo Nordisk AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk AS filed Critical Novo Nordisk AS
Publication of JP2001510195A publication Critical patent/JP2001510195A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
JP2000503085A 1997-07-16 1998-06-30 縮合化１，２，４−チアジアジン誘導体、その調製及び使用 Pending JP2001510195A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
DK0872/97 1997-07-16
DK87297 1997-07-16
DK0368/98 1998-03-17
DK36898 1998-03-17
PCT/DK1998/000288 WO1999003861A1 (en) 1997-07-16 1998-06-30 Fused 1,2,4-thiadiazine derivatives, their preparation and use

Publications (1)

Publication Number Publication Date
JP2001510195A true JP2001510195A (ja) 2001-07-31

Family

ID=26063863

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2000503085A Pending JP2001510195A (ja) 1997-07-16 1998-06-30 縮合化１，２，４−チアジアジン誘導体、その調製及び使用

Country Status (13)

Country Link
EP (1) EP1000066A1 (ko)
JP (1) JP2001510195A (ko)
KR (1) KR20010021936A (ko)
CN (1) CN1264384A (ko)
AU (1) AU757693B2 (ko)
BR (1) BR9810592A (ko)
CA (1) CA2294830A1 (ko)
HU (1) HUP0003999A3 (ko)
IL (1) IL133604A0 (ko)
NO (1) NO315470B1 (ko)
PL (1) PL338013A1 (ko)
RU (1) RU2215004C2 (ko)
WO (1) WO1999003861A1 (ko)

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* Cited by examiner, † Cited by third party
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