IS7782A - Setin píperasín, (1,4) díassepín og 2,5-díasabísýkló (2.2.1) heptön sem histamín H1 og/eða H3 mótlyf eða histamín H3 gagnmótlyf - Google Patents

Setin píperasín, (1,4) díassepín og 2,5-díasabísýkló (2.2.1) heptön sem histamín H1 og/eða H3 mótlyf eða histamín H3 gagnmótlyf

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Publication number
IS7782A
IS7782A IS7782A IS7782A IS7782A IS 7782 A IS7782 A IS 7782A IS 7782 A IS7782 A IS 7782A IS 7782 A IS7782 A IS 7782A IS 7782 A IS7782 A IS 7782A
Authority
IS
Iceland
Prior art keywords
histamine
antagonists
diazepines
heptanes
diazabicyclo
Prior art date
Application number
IS7782A
Other languages
English (en)
Inventor
Ancliff Rachael
David Eldred Colin
C. Fogden Yvonne
Paul Hancock Ashley
Daniel Heightman Thomas
Hobbs Heather
Teanby Hodgson Simon
J. Lindon Matthew
Matthew Wilson David
Original Assignee
Glaxo Group Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Limited filed Critical Glaxo Group Limited
Publication of IS7782A publication Critical patent/IS7782A/is

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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IS7782A 2002-10-16 2005-03-31 Setin píperasín, (1,4) díassepín og 2,5-díasabísýkló (2.2.1) heptön sem histamín H1 og/eða H3 mótlyf eða histamín H3 gagnmótlyf IS7782A (is)

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ZA200603604B (en) 2007-04-25
MA27482A1 (fr) 2005-08-01
MXPA05004078A (es) 2005-06-08
BR0315283A (pt) 2005-08-30
US20100075953A1 (en) 2010-03-25
PL376477A1 (en) 2005-12-27
CN1726201A (zh) 2006-01-25
RU2005110061A (ru) 2006-01-20
US20060025404A1 (en) 2006-02-02
KR20050049553A (ko) 2005-05-25
ZA200502873B (en) 2006-07-26
CN101070309A (zh) 2007-11-14
NO20051689D0 (no) 2005-04-05
AU2003280380A1 (en) 2004-05-04
JP2006508935A (ja) 2006-03-16
RU2328494C2 (ru) 2008-07-10
US7615550B2 (en) 2009-11-10
GB0224084D0 (en) 2002-11-27
NZ539446A (en) 2006-11-30
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EP1567511A1 (en) 2005-08-31

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