NO20051689D0 - Substituerte piperaziner, (1,4) diaszepiner og 2,5-diazabicyklo(2.2.1) heptaner som histamin H1 og/eller H3 antagonister eller histamin H3 revers antagonister - Google Patents
Substituerte piperaziner, (1,4) diaszepiner og 2,5-diazabicyklo(2.2.1) heptaner som histamin H1 og/eller H3 antagonister eller histamin H3 revers antagonisterInfo
- Publication number
- NO20051689D0 NO20051689D0 NO20051689A NO20051689A NO20051689D0 NO 20051689 D0 NO20051689 D0 NO 20051689D0 NO 20051689 A NO20051689 A NO 20051689A NO 20051689 A NO20051689 A NO 20051689A NO 20051689 D0 NO20051689 D0 NO 20051689D0
- Authority
- NO
- Norway
- Prior art keywords
- histamine
- antagonists
- diaszepines
- heptanes
- diazabicyclo
- Prior art date
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
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-
- C—CHEMISTRY; METALLURGY
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
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GBGB0224084.4A GB0224084D0 (en) | 2002-10-16 | 2002-10-16 | Novel compounds |
PCT/EP2003/011423 WO2004035556A1 (en) | 2002-10-16 | 2003-10-14 | Substituted piperazines, (1,4) diaszepines, and 2,5-diazabicyclo (2.2.1) heptanes as histamine h1 and/or h3 antagonists or histamine h3 reverse antagonists |
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NO20051689A NO20051689L (no) | 2002-10-16 | 2005-04-05 | Substituerte piperaziner, (1,4) diaszepiner og 2,5-diazabicyklo(2.2.1) heptaner som histamin H1 og/eller H3 antagonister eller histamin H3 revers antagonister |
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US6620839B2 (en) * | 2000-07-13 | 2003-09-16 | Abbott Laboratories | 1,3-disubstituted and 1,3,3-trisubstituted pyrrolidines as histamine-3 receptor ligands and their therapeutic applications |
DE60130460T2 (de) | 2000-07-13 | 2008-06-05 | Abbott Laboratories, Abbott Park | 1,3-disubstituierte und 1,3,3-trisubstituierte pyrrolidine als liganden des histamin-3 rezeptors und ihre therapeutischen anwendungen |
AU2001278491A1 (en) | 2000-07-18 | 2002-01-30 | Basf Aktiengesellschaft | 1-aryl-4-alkyl halide-2(1h)-pyridones and their use as herbicides |
DE60117814T2 (de) * | 2000-08-08 | 2006-11-02 | Ortho-Mcneil Pharmaceutical, Inc. | Nicht-imidazol aryloxyalkylamine als h3 rezeptor liganden |
MXPA03001268A (es) * | 2000-08-08 | 2004-09-06 | Johnson & Johnson | Ariloxipiperidinas sin imidazol. |
JP2002173426A (ja) | 2000-12-05 | 2002-06-21 | Ss Pharmaceut Co Ltd | 血糖低下剤 |
US20040077654A1 (en) | 2001-01-15 | 2004-04-22 | Bouillot Anne Marie Jeanne | Aryl piperidine and piperazine derivatives as inducers of ldl-receptor expression |
AU2002254114A1 (en) * | 2001-03-23 | 2002-10-08 | Eli Lilly And Company | Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses |
JP4186518B2 (ja) * | 2001-06-15 | 2008-11-26 | アステラス製薬株式会社 | フェニルピリジン誘導体 |
US7459461B2 (en) | 2001-10-19 | 2008-12-02 | Ortho-Mcneil Pharmaceutical, Inc. | Phosphonic acid compounds as inhibitors of serine proteases |
EP1474401A2 (en) * | 2002-02-05 | 2004-11-10 | Novo Nordisk A/S | Novel aryl- and heteroarylpiperazines |
GB0224084D0 (en) * | 2002-10-16 | 2002-11-27 | Glaxo Group Ltd | Novel compounds |
US20060019964A1 (en) | 2002-10-16 | 2006-01-26 | Ancliff Ranchael A | Compounds |
GB0609897D0 (en) * | 2006-05-18 | 2006-06-28 | Glaxo Group Ltd | Compounds |
-
2002
- 2002-10-16 GB GBGB0224084.4A patent/GB0224084D0/en not_active Ceased
-
2003
- 2003-10-14 NZ NZ549963A patent/NZ549963A/en unknown
- 2003-10-14 PL PL03376477A patent/PL376477A1/xx unknown
- 2003-10-14 RU RU2005110061/04A patent/RU2328494C2/ru not_active IP Right Cessation
- 2003-10-14 MX MXPA05004078A patent/MXPA05004078A/es unknown
- 2003-10-14 KR KR1020057006621A patent/KR20050049553A/ko not_active Application Discontinuation
- 2003-10-14 WO PCT/EP2003/011423 patent/WO2004035556A1/en active Application Filing
- 2003-10-14 BR BR0315283-9A patent/BR0315283A/pt not_active IP Right Cessation
- 2003-10-14 CA CA002502249A patent/CA2502249A1/en not_active Abandoned
- 2003-10-14 EP EP03772221A patent/EP1567511A1/en not_active Withdrawn
- 2003-10-14 JP JP2004544241A patent/JP2006508935A/ja active Pending
- 2003-10-14 CN CNA2006101086109A patent/CN101070309A/zh active Pending
- 2003-10-14 US US10/531,758 patent/US7615550B2/en not_active Expired - Fee Related
- 2003-10-14 CN CNB2003801060141A patent/CN100400523C/zh not_active Expired - Fee Related
- 2003-10-14 NZ NZ539446A patent/NZ539446A/en unknown
- 2003-10-14 AU AU2003280380A patent/AU2003280380A1/en not_active Abandoned
-
2005
- 2005-03-31 IS IS7782A patent/IS7782A/is unknown
- 2005-04-05 NO NO20051689A patent/NO20051689L/no not_active Application Discontinuation
- 2005-04-08 ZA ZA200502873A patent/ZA200502873B/en unknown
- 2005-04-29 MA MA28246A patent/MA27482A1/fr unknown
-
2006
- 2006-05-05 ZA ZA200603604A patent/ZA200603604B/en unknown
- 2006-08-28 JP JP2006231163A patent/JP2007016041A/ja active Pending
-
2009
- 2009-09-18 US US12/562,285 patent/US20100075953A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
CN101070309A (zh) | 2007-11-14 |
WO2004035556A1 (en) | 2004-04-29 |
MA27482A1 (fr) | 2005-08-01 |
US20100075953A1 (en) | 2010-03-25 |
RU2328494C2 (ru) | 2008-07-10 |
GB0224084D0 (en) | 2002-11-27 |
PL376477A1 (en) | 2005-12-27 |
CN100400523C (zh) | 2008-07-09 |
NO20051689L (no) | 2005-07-07 |
IS7782A (is) | 2005-03-31 |
AU2003280380A1 (en) | 2004-05-04 |
JP2006508935A (ja) | 2006-03-16 |
EP1567511A1 (en) | 2005-08-31 |
NZ549963A (en) | 2008-03-28 |
BR0315283A (pt) | 2005-08-30 |
MXPA05004078A (es) | 2005-06-08 |
JP2007016041A (ja) | 2007-01-25 |
US20060025404A1 (en) | 2006-02-02 |
US7615550B2 (en) | 2009-11-10 |
RU2005110061A (ru) | 2006-01-20 |
CA2502249A1 (en) | 2004-04-29 |
ZA200502873B (en) | 2006-07-26 |
CN1726201A (zh) | 2006-01-25 |
ZA200603604B (en) | 2007-04-25 |
NZ539446A (en) | 2006-11-30 |
KR20050049553A (ko) | 2005-05-25 |
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