IN2014DN07082A - - Google Patents

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Publication number
IN2014DN07082A
IN2014DN07082A IN7082DEN2014A IN2014DN07082A IN 2014DN07082 A IN2014DN07082 A IN 2014DN07082A IN 7082DEN2014 A IN7082DEN2014 A IN 7082DEN2014A IN 2014DN07082 A IN2014DN07082 A IN 2014DN07082A
Authority
IN
India
Prior art keywords
alkyl
dibenzoyltartrate
haloalkyl
cycloalkyl
chloride
Prior art date
Application number
Other languages
English (en)
Inventor
Alfred Fetscher
Jochen Matthias Scher
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49292482&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2014DN07082(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of IN2014DN07082A publication Critical patent/IN2014DN07082A/en

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
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Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pulmonology (AREA)
  • Inorganic Chemistry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Dermatology (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Transplantation (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hematology (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IN7082DEN2014 2012-04-04 2013-04-02 IN2014DN07082A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12163078 2012-04-04
PCT/EP2013/056867 WO2013149987A1 (fr) 2012-04-04 2013-04-02 Formulations pharmaceutiques comprenant des antagonistes de ccr3

Publications (1)

Publication Number Publication Date
IN2014DN07082A true IN2014DN07082A (fr) 2015-04-10

Family

ID=49292482

Family Applications (1)

Application Number Title Priority Date Filing Date
IN7082DEN2014 IN2014DN07082A (fr) 2012-04-04 2013-04-02

Country Status (30)

Country Link
US (3) US10213421B2 (fr)
EP (3) EP2833864B1 (fr)
JP (4) JP6320990B2 (fr)
KR (2) KR102138709B1 (fr)
CN (1) CN104203213A (fr)
AR (1) AR090596A1 (fr)
AU (1) AU2013245028B2 (fr)
BR (1) BR112014024479A8 (fr)
CA (1) CA2869058C (fr)
CL (1) CL2014002524A1 (fr)
CY (1) CY1121137T1 (fr)
DK (2) DK3524230T3 (fr)
EA (1) EA027627B1 (fr)
ES (2) ES2715844T3 (fr)
HR (1) HRP20190069T1 (fr)
HU (2) HUE041519T2 (fr)
IL (1) IL234299A (fr)
IN (1) IN2014DN07082A (fr)
LT (1) LT2833864T (fr)
MX (1) MX358307B (fr)
NZ (1) NZ628993A (fr)
PH (1) PH12014502241A1 (fr)
PL (2) PL2833864T3 (fr)
PT (2) PT2833864T (fr)
RS (1) RS58360B1 (fr)
SI (1) SI2833864T1 (fr)
TR (1) TR201821285T4 (fr)
TW (1) TW201400115A (fr)
UY (1) UY34730A (fr)
WO (1) WO2013149987A1 (fr)

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Publication number Priority date Publication date Assignee Title
US8278302B2 (en) 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
AR090566A1 (es) 2012-04-02 2014-11-19 Boehringer Ingelheim Int Proceso para la produccion de inhibidores de crr
US20130261153A1 (en) * 2012-04-03 2013-10-03 Boehringer Ingelheim International Gmbh Use of ccr3-inhibitors
US10213421B2 (en) * 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists
CA3058967A1 (fr) 2017-04-05 2018-10-11 Alkahest, Inc. Methodes et compositions destinees a traiter des troubles associes au vieillissement a l'aide d'inhibiteurs de ccr3
IL269743B (en) 2017-04-05 2022-09-01 Alkahest Inc Methods and preparations for the treatment of disease related to the retina with CCR-3 inhibitor inventions
WO2019075351A1 (fr) * 2017-10-13 2019-04-18 Alkahest, Inc. Méthodes et compositions pour pour traiter un prurit, un xérosis et une maladie associée à l'aide d'inhibiteurs de ccr3
CN112469439A (zh) 2018-05-15 2021-03-09 万能溶剂有限公司 用白三烯a4水解酶调节剂治疗衰老相关性疾病
BR112021004938A2 (pt) * 2018-09-26 2021-06-01 Alkahest, Inc. métodos e composições para tratamento de danos associados com o envelhecimento usando inibidores de ccr3
CN115989200A (zh) 2020-08-27 2023-04-18 Ａｇｃ株式会社 无碱玻璃和玻璃板
AU2022376563A1 (en) 2021-11-01 2023-12-07 Alkahest, Inc. Benzodioxane modulators of leukotriene a4 hydrolase (lta4h) for prevention and treatment of aging-associated diseases

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KR20060061393A (ko) 2003-10-24 2006-06-07 에프. 호프만-라 로슈 아게 Ｃｃｒ3 수용체 길항제
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KR20140140064A (ko) 2014-12-08
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