IN2014DN07082A - - Google Patents

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Publication number
IN2014DN07082A
IN2014DN07082A IN7082DEN2014A IN2014DN07082A IN 2014DN07082 A IN2014DN07082 A IN 2014DN07082A IN 7082DEN2014 A IN7082DEN2014 A IN 7082DEN2014A IN 2014DN07082 A IN2014DN07082 A IN 2014DN07082A
Authority
IN
India
Prior art keywords
alkyl
dibenzoyltartrate
haloalkyl
cycloalkyl
chloride
Prior art date
Application number
Other languages
English (en)
Inventor
Alfred Fetscher
Jochen Matthias Scher
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49292482&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IN2014DN07082(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of IN2014DN07082A publication Critical patent/IN2014DN07082A/en

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
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Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pulmonology (AREA)
  • Inorganic Chemistry (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Oncology (AREA)
  • Neurology (AREA)
  • Communicable Diseases (AREA)
  • Urology & Nephrology (AREA)
  • Otolaryngology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Transplantation (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IN7082DEN2014 2012-04-04 2013-04-02 IN2014DN07082A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12163078 2012-04-04
PCT/EP2013/056867 WO2013149987A1 (fr) 2012-04-04 2013-04-02 Formulations pharmaceutiques comprenant des antagonistes de ccr3

Publications (1)

Publication Number Publication Date
IN2014DN07082A true IN2014DN07082A (fr) 2015-04-10

Family

ID=49292482

Family Applications (1)

Application Number Title Priority Date Filing Date
IN7082DEN2014 IN2014DN07082A (fr) 2012-04-04 2013-04-02

Country Status (30)

Country Link
US (3) US10213421B2 (fr)
EP (3) EP3970693A1 (fr)
JP (4) JP6320990B2 (fr)
KR (2) KR102338465B1 (fr)
CN (1) CN104203213A (fr)
AR (1) AR090596A1 (fr)
AU (1) AU2013245028B2 (fr)
BR (1) BR112014024479A8 (fr)
CA (1) CA2869058C (fr)
CL (1) CL2014002524A1 (fr)
CY (1) CY1121137T1 (fr)
DK (2) DK3524230T3 (fr)
EA (1) EA027627B1 (fr)
ES (2) ES2898179T3 (fr)
HR (1) HRP20190069T1 (fr)
HU (2) HUE056943T2 (fr)
IL (1) IL234299A (fr)
IN (1) IN2014DN07082A (fr)
LT (1) LT2833864T (fr)
MX (1) MX358307B (fr)
NZ (1) NZ628993A (fr)
PH (1) PH12014502241A1 (fr)
PL (2) PL3524230T3 (fr)
PT (2) PT2833864T (fr)
RS (1) RS58360B1 (fr)
SI (1) SI2833864T1 (fr)
TR (1) TR201821285T4 (fr)
TW (1) TW201400115A (fr)
UY (1) UY34730A (fr)
WO (1) WO2013149987A1 (fr)

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Publication number Priority date Publication date Assignee Title
US8278302B2 (en) 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
US8680280B2 (en) 2012-04-02 2014-03-25 Boehringer Ingelheim International Gmbh Process for the manufacturing of CRR inhibitors
US20130261153A1 (en) * 2012-04-03 2013-10-03 Boehringer Ingelheim International Gmbh Use of ccr3-inhibitors
US10213421B2 (en) 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists
SG11201909207VA (en) * 2017-04-05 2019-11-28 Alkahest Inc Methods and compositions for treating retina-associated disease using ccr3-inhibitors
JP2020513005A (ja) * 2017-04-05 2020-04-30 アルカヘスト，インコーポレイテッド Ｃｃｒ３阻害剤を用いて、加齢性機能障害を治療するための方法及び組成物
US20190111042A1 (en) * 2017-10-13 2019-04-18 Alkahest, Inc. Methods and Compositions for Treating Pruritus, Xerosis, and Associated Disease Using CCR-Inhibitors
EP3793602A4 (fr) 2018-05-15 2022-04-20 Alkahest, Inc. Traitement d'une maladie associée au vieillissement avec des modulateurs de la leucotriène a4 hydrolase
MA53743A (fr) * 2018-09-26 2022-01-05 Alkahest Inc Procédés et compositions pour traiter des troubles liés au vieillissement au moyen d'inhibiteurs de ccr3
JPWO2022045226A1 (fr) 2020-08-27 2022-03-03
CA3221177A1 (fr) 2021-11-01 2023-05-04 Meghan Kerrisk Campbell Modulateurs de benzodioxane de leucotriene a4 hydrolase (lta4h) pour la prevention et le traitement de maladies liees au vieillissement

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ES2324224T3 (es) 2004-02-05 2009-08-03 Schering Corporation Derivados de piperidina que se pueden utilizar como antagonistas ccr3.
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PT2833864T (pt) 2019-03-28
JP2018138557A (ja) 2018-09-06
IL234299A (en) 2017-07-31
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