IL99166A - History 3-) 1,3-Benziazoxazole-3-Il-4-pyridiamine, their preparation and pharmaceutical preparations containing them - Google Patents

History 3-) 1,3-Benziazoxazole-3-Il-4-pyridiamine, their preparation and pharmaceutical preparations containing them

Info

Publication number
IL99166A
IL99166A IL9916691A IL9916691A IL99166A IL 99166 A IL99166 A IL 99166A IL 9916691 A IL9916691 A IL 9916691A IL 9916691 A IL9916691 A IL 9916691A IL 99166 A IL99166 A IL 99166A
Authority
IL
Israel
Prior art keywords
compound
hydrogen
benzisoxazol
loweralkyl
arylalkyl
Prior art date
Application number
IL9916691A
Other languages
English (en)
Hebrew (he)
Other versions
IL99166A0 (en
Original Assignee
Hoechst Roussel Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharma filed Critical Hoechst Roussel Pharma
Publication of IL99166A0 publication Critical patent/IL99166A0/xx
Publication of IL99166A publication Critical patent/IL99166A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
IL9916691A 1990-08-13 1991-08-12 History 3-) 1,3-Benziazoxazole-3-Il-4-pyridiamine, their preparation and pharmaceutical preparations containing them IL99166A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/566,932 US5055476A (en) 1990-08-13 1990-08-13 3-(1,2-benzisoxazol-3-yl)-4-pyridinamines and derivatives

Publications (2)

Publication Number Publication Date
IL99166A0 IL99166A0 (en) 1992-07-15
IL99166A true IL99166A (en) 1995-12-08

Family

ID=24265033

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9916691A IL99166A (en) 1990-08-13 1991-08-12 History 3-) 1,3-Benziazoxazole-3-Il-4-pyridiamine, their preparation and pharmaceutical preparations containing them

Country Status (24)

Country Link
US (1) US5055476A (cs)
EP (1) EP0471297B1 (cs)
JP (1) JP3057829B2 (cs)
KR (1) KR100191386B1 (cs)
AT (1) ATE130004T1 (cs)
AU (1) AU633791B2 (cs)
CA (1) CA2048959C (cs)
CZ (1) CZ280568B6 (cs)
DE (1) DE69114405T2 (cs)
DK (1) DK0471297T3 (cs)
ES (1) ES2079531T3 (cs)
FI (1) FI103970B (cs)
GR (1) GR3018184T3 (cs)
HU (1) HU213201B (cs)
IE (1) IE70597B1 (cs)
IL (1) IL99166A (cs)
MX (1) MX9100639A (cs)
NO (1) NO179519C (cs)
NZ (1) NZ239326A (cs)
PT (1) PT98645B (cs)
RU (1) RU2012561C1 (cs)
TW (1) TW202446B (cs)
YU (1) YU140991A (cs)
ZA (1) ZA916342B (cs)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5308826A (en) * 1993-04-22 1994-05-03 Zeneca Limited Herbicidal 4-substituted pyridyl-3-carbinols
US5595958A (en) * 1994-05-02 1997-01-21 Zeneca Limited 3-substituted pyridine compounds and derivatives thereof
AU2313995A (en) * 1994-05-02 1995-11-29 Zeneca Limited Herbicidal hydroxybenzyl-substituted heteroaryl compounds and derivatives thereof
DK2718270T3 (da) 2011-06-10 2022-08-01 Merck Patent Gmbh Sammensætninger og fremgangsmåder til fremstillingen af pyrimidin- og pyridinforbindelser med btk-hæmmende aktivitet
RU2626650C2 (ru) * 2015-08-31 2017-07-31 Федеральное государственное бюджетное образовательное учреждение высшего образования "Пермский государственный национальный исследовательский университет" 2-Арил-2,4-дигидрокси-2,5-дигидро-3-гетерил-5-оксо-1Н-пиррол-1-ил-4-метилбелзолсульфаниламиды, обладающие анальгетической активностью
WO2023083445A1 (en) 2021-11-10 2023-05-19 Symrise Ag Compositions comprising trpm8 agonistic cooling agents

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4355037A (en) * 1981-11-12 1982-10-19 Hoechst-Roussel Pharmaceuticals 3-(4-Piperidyl)-1,2-benzisoxales
IL66866A (en) * 1982-04-09 1987-08-31 Hoechst Roussel Pharma 1-(3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl)-4-(substituted)-piperazines and-piperidines,a process for the preparation thereof,and pharmaceutical compositions containing them
CA1335289C (en) * 1987-10-26 1995-04-18 Fujio Antoku Piperidinyl benzisoxazole derivatives, their production and pharmaceutical use
IE74711B1 (en) * 1990-07-27 1997-07-30 Ici Plc Fungicides

Also Published As

Publication number Publication date
NO913142L (no) 1992-02-14
FI103970B1 (fi) 1999-10-29
PT98645B (pt) 1999-01-29
EP0471297A1 (en) 1992-02-19
CZ280568B6 (cs) 1996-02-14
MX9100639A (es) 1992-04-01
GR3018184T3 (en) 1996-02-29
NO913142D0 (no) 1991-08-12
JPH05112562A (ja) 1993-05-07
NO179519C (no) 1996-10-23
JP3057829B2 (ja) 2000-07-04
EP0471297B1 (en) 1995-11-08
DE69114405T2 (de) 1996-05-02
HU213201B (en) 1997-03-28
CS248991A3 (en) 1992-03-18
US5055476A (en) 1991-10-08
IE912851A1 (en) 1992-02-26
IL99166A0 (en) 1992-07-15
ES2079531T3 (es) 1996-01-16
DK0471297T3 (da) 1996-03-04
RU2012561C1 (ru) 1994-05-15
TW202446B (cs) 1993-03-21
NZ239326A (en) 1994-04-27
FI913800A0 (fi) 1991-08-09
IE70597B1 (en) 1996-12-11
PT98645A (pt) 1992-06-30
YU140991A (sh) 1995-01-31
CA2048959C (en) 2003-07-29
AU8176591A (en) 1992-02-20
ZA916342B (en) 1992-04-29
DE69114405D1 (de) 1995-12-14
ATE130004T1 (de) 1995-11-15
KR100191386B1 (ko) 1999-06-15
CA2048959A1 (en) 1992-02-14
NO179519B (no) 1996-07-15
KR920004383A (ko) 1992-03-27
HU912673D0 (en) 1992-01-28
FI913800A (fi) 1992-02-14
HUT61755A (en) 1993-03-01
AU633791B2 (en) 1993-02-04
FI103970B (fi) 1999-10-29

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Legal Events

Date Code Title Description
FF Patent granted
HC Change of name of proprietor(s)
KB Patent renewed
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees