FI103970B1 - Menetelmä kivun lievittämiseen sekä ihotautien ja muistin toimintahäiriöiden hoitoon tarkoitettujen 3-(1,2-bentsisoksatsol-3-yyli)-4-pyridiiniamiinien ja näiden johdannaisten valmistamiseksi - Google Patents

Menetelmä kivun lievittämiseen sekä ihotautien ja muistin toimintahäiriöiden hoitoon tarkoitettujen 3-(1,2-bentsisoksatsol-3-yyli)-4-pyridiiniamiinien ja näiden johdannaisten valmistamiseksi

Info

Publication number
FI103970B1
FI103970B1 FI913800A FI913800A FI103970B1 FI 103970 B1 FI103970 B1 FI 103970B1 FI 913800 A FI913800 A FI 913800A FI 913800 A FI913800 A FI 913800A FI 103970 B1 FI103970 B1 FI 103970B1
Authority
FI
Finland
Prior art keywords
treatment
benzisoxazol
derivatives
hydrogen
pyridinamine
Prior art date
Application number
FI913800A
Other languages
English (en)
Swedish (sv)
Other versions
FI913800A0 (fi
FI913800A (fi
FI103970B (fi
Inventor
Joseph Thomas Klein
Richard Charles Effland
Original Assignee
Hoechst Marion Roussel Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Marion Roussel Inc filed Critical Hoechst Marion Roussel Inc
Publication of FI913800A0 publication Critical patent/FI913800A0/fi
Publication of FI913800A publication Critical patent/FI913800A/fi
Application granted granted Critical
Publication of FI103970B1 publication Critical patent/FI103970B1/fi
Publication of FI103970B publication Critical patent/FI103970B/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
FI913800A 1990-08-13 1991-08-09 Menetelmä kivun lievittämiseen sekä ihotautien ja muistin toimintahäiriöiden hoitoon tarkoitettujen 3-(1,2-bentsisoksatsol-3-yyli)-4-pyridiiniamiinien ja näiden johdannaisten valmistamiseksi FI103970B (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US56693290 1990-08-13
US07/566,932 US5055476A (en) 1990-08-13 1990-08-13 3-(1,2-benzisoxazol-3-yl)-4-pyridinamines and derivatives

Publications (4)

Publication Number Publication Date
FI913800A0 FI913800A0 (fi) 1991-08-09
FI913800A FI913800A (fi) 1992-02-14
FI103970B1 true FI103970B1 (fi) 1999-10-29
FI103970B FI103970B (fi) 1999-10-29

Family

ID=24265033

Family Applications (1)

Application Number Title Priority Date Filing Date
FI913800A FI103970B (fi) 1990-08-13 1991-08-09 Menetelmä kivun lievittämiseen sekä ihotautien ja muistin toimintahäiriöiden hoitoon tarkoitettujen 3-(1,2-bentsisoksatsol-3-yyli)-4-pyridiiniamiinien ja näiden johdannaisten valmistamiseksi

Country Status (24)

Country Link
US (1) US5055476A (fi)
EP (1) EP0471297B1 (fi)
JP (1) JP3057829B2 (fi)
KR (1) KR100191386B1 (fi)
AT (1) ATE130004T1 (fi)
AU (1) AU633791B2 (fi)
CA (1) CA2048959C (fi)
CZ (1) CZ280568B6 (fi)
DE (1) DE69114405T2 (fi)
DK (1) DK0471297T3 (fi)
ES (1) ES2079531T3 (fi)
FI (1) FI103970B (fi)
GR (1) GR3018184T3 (fi)
HU (1) HU213201B (fi)
IE (1) IE70597B1 (fi)
IL (1) IL99166A (fi)
MX (1) MX9100639A (fi)
NO (1) NO179519C (fi)
NZ (1) NZ239326A (fi)
PT (1) PT98645B (fi)
RU (1) RU2012561C1 (fi)
TW (1) TW202446B (fi)
YU (1) YU140991A (fi)
ZA (1) ZA916342B (fi)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5308826A (en) * 1993-04-22 1994-05-03 Zeneca Limited Herbicidal 4-substituted pyridyl-3-carbinols
EP0758323A1 (en) * 1994-05-02 1997-02-19 Zeneca Limited Herbicidal hydroxybenzyl-substituted heteroaryl compounds and derivatives thereof
US5595958A (en) * 1994-05-02 1997-01-21 Zeneca Limited 3-substituted pyridine compounds and derivatives thereof
SG194219A1 (en) 2011-06-10 2013-11-29 Merck Patent Gmbh Compositions and methods for the production of pyrimidine and pyridine compounds with btk inhibitory activity
RU2626650C2 (ru) * 2015-08-31 2017-07-31 Федеральное государственное бюджетное образовательное учреждение высшего образования "Пермский государственный национальный исследовательский университет" 2-Арил-2,4-дигидрокси-2,5-дигидро-3-гетерил-5-оксо-1Н-пиррол-1-ил-4-метилбелзолсульфаниламиды, обладающие анальгетической активностью
WO2023083445A1 (en) 2021-11-10 2023-05-19 Symrise Ag Compositions comprising trpm8 agonistic cooling agents

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4355037A (en) * 1981-11-12 1982-10-19 Hoechst-Roussel Pharmaceuticals 3-(4-Piperidyl)-1,2-benzisoxales
IL66866A (en) * 1982-04-09 1987-08-31 Hoechst Roussel Pharma 1-(3-(6-fluoro-1,2-benzisoxazol-3-yl)propyl)-4-(substituted)-piperazines and-piperidines,a process for the preparation thereof,and pharmaceutical compositions containing them
CA1335289C (en) * 1987-10-26 1995-04-18 Fujio Antoku Piperidinyl benzisoxazole derivatives, their production and pharmaceutical use
IE74711B1 (en) * 1990-07-27 1997-07-30 Ici Plc Fungicides

Also Published As

Publication number Publication date
HU213201B (en) 1997-03-28
FI913800A0 (fi) 1991-08-09
RU2012561C1 (ru) 1994-05-15
NO179519C (no) 1996-10-23
US5055476A (en) 1991-10-08
ES2079531T3 (es) 1996-01-16
AU633791B2 (en) 1993-02-04
NO179519B (no) 1996-07-15
AU8176591A (en) 1992-02-20
FI913800A (fi) 1992-02-14
IE912851A1 (en) 1992-02-26
IL99166A (en) 1995-12-08
YU140991A (sh) 1995-01-31
PT98645B (pt) 1999-01-29
GR3018184T3 (en) 1996-02-29
CA2048959C (en) 2003-07-29
HU912673D0 (en) 1992-01-28
EP0471297B1 (en) 1995-11-08
JPH05112562A (ja) 1993-05-07
NO913142L (no) 1992-02-14
CZ280568B6 (cs) 1996-02-14
HUT61755A (en) 1993-03-01
EP0471297A1 (en) 1992-02-19
TW202446B (fi) 1993-03-21
NO913142D0 (no) 1991-08-12
DK0471297T3 (da) 1996-03-04
NZ239326A (en) 1994-04-27
DE69114405T2 (de) 1996-05-02
KR920004383A (ko) 1992-03-27
ATE130004T1 (de) 1995-11-15
KR100191386B1 (ko) 1999-06-15
JP3057829B2 (ja) 2000-07-04
IE70597B1 (en) 1996-12-11
MX9100639A (es) 1992-04-01
CA2048959A1 (en) 1992-02-14
CS248991A3 (en) 1992-03-18
DE69114405D1 (de) 1995-12-14
FI103970B (fi) 1999-10-29
ZA916342B (en) 1992-04-29
IL99166A0 (en) 1992-07-15
PT98645A (pt) 1992-06-30

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Legal Events

Date Code Title Description
GB Transfer or assigment of application

Owner name: HOECHST MARION ROUSSEL, INC.