IL83814A - 10-(cyclic)amino-9-halo-7-oxo-2,3-dihydro-7h-pyrido(3,2,1-ij)-1,3,4-benzoxadiazine-6-carboxylic acid derivatives,their manufacture and pharmaceutical compositions containing them and some intermediates therefor - Google Patents

10-(cyclic)amino-9-halo-7-oxo-2,3-dihydro-7h-pyrido(3,2,1-ij)-1,3,4-benzoxadiazine-6-carboxylic acid derivatives,their manufacture and pharmaceutical compositions containing them and some intermediates therefor

Info

Publication number
IL83814A
IL83814A IL83814A IL8381487A IL83814A IL 83814 A IL83814 A IL 83814A IL 83814 A IL83814 A IL 83814A IL 8381487 A IL8381487 A IL 8381487A IL 83814 A IL83814 A IL 83814A
Authority
IL
Israel
Prior art keywords
benzoxadiazine
pyrido
dihydro
halo
oxo
Prior art date
Application number
IL83814A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of IL83814A publication Critical patent/IL83814A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/06Peri-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/58Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems with hetero atoms directly attached to the ring nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Quinoline Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL83814A 1986-09-12 1987-09-07 10-(cyclic)amino-9-halo-7-oxo-2,3-dihydro-7h-pyrido(3,2,1-ij)-1,3,4-benzoxadiazine-6-carboxylic acid derivatives,their manufacture and pharmaceutical compositions containing them and some intermediates therefor IL83814A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP86112619 1986-09-12

Publications (1)

Publication Number Publication Date
IL83814A true IL83814A (en) 1991-09-16

Family

ID=8195410

Family Applications (1)

Application Number Title Priority Date Filing Date
IL83814A IL83814A (en) 1986-09-12 1987-09-07 10-(cyclic)amino-9-halo-7-oxo-2,3-dihydro-7h-pyrido(3,2,1-ij)-1,3,4-benzoxadiazine-6-carboxylic acid derivatives,their manufacture and pharmaceutical compositions containing them and some intermediates therefor

Country Status (22)

Country Link
JP (3) JPH0696578B2 (fi)
KR (1) KR960002857B1 (fi)
CN (1) CN1017800B (fi)
AT (1) AT389119B (fi)
AU (1) AU602534B2 (fi)
CA (1) CA1336905C (fi)
CZ (1) CZ281195B6 (fi)
DK (1) DK173330B1 (fi)
DZ (1) DZ1124A1 (fi)
FI (1) FI86428C (fi)
HU (1) HU199481B (fi)
IE (1) IE61624B1 (fi)
IL (1) IL83814A (fi)
MC (1) MC1850A1 (fi)
MX (1) MX8302A (fi)
NO (1) NO169125C (fi)
NZ (1) NZ221681A (fi)
PH (1) PH23930A (fi)
PT (1) PT85686B (fi)
SK (1) SK278990B6 (fi)
ZA (1) ZA876636B (fi)
ZW (1) ZW16387A1 (fi)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZW16387A1 (en) * 1986-09-12 1988-05-25 Hoffmann La Roche Tricyclic compounds
EP1757598A4 (en) 2004-05-13 2010-07-21 Daiichi Seiyaku Co SUBSTITUTED PYRROLIDINE DERIVATIVE
US7563805B2 (en) * 2005-05-19 2009-07-21 Daiichi Pharmaceutical Co., Ltd. Tri-, tetra-substituted-3-aminopyrrolidine derivative
CN101443314B (zh) 2006-03-13 2014-04-09 杏林制药株式会社 作为gsk-3抑制剂的氨基喹诺酮类
JP5426552B2 (ja) 2007-09-11 2014-02-26 杏林製薬株式会社 Gsk−3阻害剤としてのシアノアミノキノロン及びテトラゾロアミノキノロン
MX2010002662A (es) 2007-09-12 2010-04-09 Activx Biosciences Inc Aminoquinolonas espirociclicas como inhibidores de gsk-3.
FR2928150A1 (fr) * 2008-02-29 2009-09-04 Vetoquinol Sa Sa Nouveaux derives 7-substitues de 3-carboxy-oxadiazino-quinolones, leur preparation et leur application comme anti-bacteriens
EP2145891A1 (en) * 2008-07-09 2010-01-20 Vetoquinol S.A. 9-substituted-5-carboxy-oxadiazino-quinolone derivatives, their preparation and their application as anti-bacterials
WO2010104205A1 (en) 2009-03-11 2010-09-16 Kyorin Pharmaceutical Co., Ltd. 7-cycloalkylaminoquinolones as gsk-3 inhibitors
CN107522718B (zh) * 2017-09-14 2019-11-08 浙江国邦药业有限公司 一种马波沙星的合成方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZW16387A1 (en) * 1986-09-12 1988-05-25 Hoffmann La Roche Tricyclic compounds

Also Published As

Publication number Publication date
KR960002857B1 (ko) 1996-02-27
ATA263887A (de) 1989-03-15
SK660487A3 (en) 1998-05-06
DK173330B1 (da) 2000-07-24
NO169125B (no) 1992-02-03
FI86428C (fi) 1992-08-25
MC1850A1 (fr) 1988-09-30
IE872444L (en) 1988-03-12
CN87106838A (zh) 1988-05-11
HUT47294A (en) 1989-02-28
DK477287A (da) 1988-03-13
JPH07138262A (ja) 1995-05-30
FI86428B (fi) 1992-05-15
JPH0826030B2 (ja) 1996-03-13
NO873816L (no) 1988-03-14
PT85686B (pt) 1990-05-31
KR880003954A (ko) 1988-06-01
NO873816D0 (no) 1987-09-11
HU199481B (en) 1990-02-28
SK278990B6 (sk) 1998-05-06
JPS63132891A (ja) 1988-06-04
AU602534B2 (en) 1990-10-18
CN1017800B (zh) 1992-08-12
AU7811487A (en) 1988-03-17
ZA876636B (en) 1988-07-27
CZ660487A3 (en) 1996-04-17
CA1336905C (en) 1995-09-05
IE61624B1 (en) 1994-11-16
JPH07138256A (ja) 1995-05-30
ZW16387A1 (en) 1988-05-25
DK477287D0 (da) 1987-09-11
FI873940A (fi) 1988-03-13
CZ281195B6 (cs) 1996-07-17
PH23930A (en) 1990-01-23
JPH0819120B2 (ja) 1996-02-28
PT85686A (en) 1987-10-01
NO169125C (no) 1992-05-13
AT389119B (de) 1989-10-25
FI873940A0 (fi) 1987-09-11
JPH0696578B2 (ja) 1994-11-30
NZ221681A (en) 1990-12-21
DZ1124A1 (fr) 2004-09-13
MX8302A (es) 1993-12-01

Similar Documents

Publication Publication Date Title
PT84407A (en) Process for the preparation of aromatic 2-aminoalkyl-1,2-benzoisothiazol-3 (2h)one-1,1-dioxide derivatives and of pharmaceutical compositions containing the same
IL81790A0 (en) Hydroxylamine derivatives,their manufacture and pharmaceutical compositions containing them
IL82448A0 (en) Tetrahydronaphthalene derivatives,their manufacture and pharmaceutical compositions containing them
IL84766A0 (en) Phosphinic acid derivatives,their manufacture and pharmaceutical compositions containing them
IL81791A0 (en) 3,5-disubstituted pyrocatechol derivatives,their manufacture and pharmaceutical compositions containing them
IL84522A0 (en) Imidazopyridine derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same
ZA877530B (en) Imidazopyridine derivatives and pharmaceutical compositions containing the same as well as processes for production thereof
PT85071A (en) Process for the preparation of derivatives of fused cyclic azepin-2-ones and of pharmaceutical compositions containing the same
IL76133A (en) Mercaptomethyl-octahydro-oxo-pyridazino(1,2-a)(1,2)diazepine-,diazocine-and(1,2,5)triazepinecarboxylic acid derivatives,their preparation and pharmaceutical compositions containing them and certain intermediates therefor
NZ222349A (en) Hexahydro-8-hydroxy-2,6-methano-2h-quinolizine-3(4h)-one compounds, esters thereof, and pharmaceutical compositions containing such
IL87714A0 (en) 3,7-diazabicyclo(3,3,1)nonane derivatives,their preparation and pharmaceutical compositions containing them
IL84765A0 (en) Pyridazodiazepine derivatives,their manufacture and pharmaceutical compositions containing them
IL83814A (en) 10-(cyclic)amino-9-halo-7-oxo-2,3-dihydro-7h-pyrido(3,2,1-ij)-1,3,4-benzoxadiazine-6-carboxylic acid derivatives,their manufacture and pharmaceutical compositions containing them and some intermediates therefor
IL76546A (en) 9-(heteroarylalkyl)-6-purine(thi)one derivatives,their preparation and pharmaceutical compositions containing them
IL83049A (en) 4-quinolinone-3-carboxylic acid derivatives,their manufacture and pharmaceutical compositions containing them
IL81410A (en) Pharmaceutical compositions containing substituted n-arylmethylamine derivatives,certain such novel compounds and their preparation
NZ218880A (en) Pyrido(2,3-b)indole-3-carboxylic acid derivatives and pharmaceutical compositions thereof
IL84636A0 (en) Lactam derivatives,their preparation and pharmaceutical compositions containing them
HUT45256A (en) Process for producing 1,3,4,9-tetrahydropyrano/3,4-b/indol-1-acetic acid derivatives and pharmaceutical composition containing them
IL84808A (en) Furanuronic acid derivatives,their preparation and pharmaceutical compositions containing them
IL84728A (en) Bicyclic v-triazine-4-one derivatives,their manufacture and pharmaceutical compositions containing them
PT81954A (en) Process for the preparation of pharmaceutical compositions containing 9,10-dihydro alkalloids of ergot
DE3573428D1 (en) Novel delta4- and delta5- androstene derivatives, processes for their preparation and pharmaceutical compositions containing these derivatives
IL82477A0 (en) Fungicidal compositions containing benzothiazinone derivatives,certain such novel derivatives and their preparation
IL84916A (en) Tricyclic 1h-imidazole-5-carboxylic acid derivatives,their preparation and herbicidal compositions containing them

Legal Events

Date Code Title Description
KB Patent renewed
KB Patent renewed
EXP Patent expired