IL61733A - Heterocyclic carbonylaminoalkyl benzenesulfonyl ureas,their preparation and pharmaceutical compositions comprising them - Google Patents
Heterocyclic carbonylaminoalkyl benzenesulfonyl ureas,their preparation and pharmaceutical compositions comprising themInfo
- Publication number
- IL61733A IL61733A IL61733A IL6173380A IL61733A IL 61733 A IL61733 A IL 61733A IL 61733 A IL61733 A IL 61733A IL 6173380 A IL6173380 A IL 6173380A IL 61733 A IL61733 A IL 61733A
- Authority
- IL
- Israel
- Prior art keywords
- carbonylaminoalkyl
- heterocyclic
- preparation
- pharmaceutical compositions
- benzenesulfonyl ureas
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/24—Oxygen or sulfur atoms
- C07D207/26—2-Pyrrolidones
- C07D207/263—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms
- C07D207/27—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/36—Oxygen or sulfur atoms
- C07D207/38—2-Pyrrolones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/46—Iso-indoles; Hydrogenated iso-indoles with an oxygen atom in position 1
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/72—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D211/74—Oxygen atoms
- C07D211/76—Oxygen atoms attached in position 2 or 6
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/24—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/02—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D223/06—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D223/08—Oxygen atoms
- C07D223/10—Oxygen atoms attached in position 2
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Diabetes (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Hydrogenated Pyridines (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19792951135 DE2951135A1 (de) | 1979-12-19 | 1979-12-19 | Sulfonylharnstoffe, verfahren zu ihrer herstellung, pharmazeutische praeparate auf basis dieser verbindungen und ihre verwendung |
Publications (2)
Publication Number | Publication Date |
---|---|
IL61733A0 IL61733A0 (en) | 1981-01-30 |
IL61733A true IL61733A (en) | 1985-05-31 |
Family
ID=6088937
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL61733A IL61733A (en) | 1979-12-19 | 1980-12-17 | Heterocyclic carbonylaminoalkyl benzenesulfonyl ureas,their preparation and pharmaceutical compositions comprising them |
Country Status (21)
Country | Link |
---|---|
US (1) | US4379785A (es) |
EP (1) | EP0031058B1 (es) |
JP (1) | JPS56108762A (es) |
AR (3) | AR230989A1 (es) |
AT (1) | ATE6934T1 (es) |
AU (1) | AU538129B2 (es) |
CA (1) | CA1167033A (es) |
DE (2) | DE2951135A1 (es) |
DK (1) | DK156434C (es) |
ES (6) | ES497661A0 (es) |
FI (1) | FI75338C (es) |
GR (1) | GR72534B (es) |
HU (1) | HU184943B (es) |
IE (1) | IE50635B1 (es) |
IL (1) | IL61733A (es) |
LU (1) | LU90244I2 (es) |
MX (4) | MX174496B (es) |
NL (1) | NL950026I2 (es) |
NO (2) | NO155290C (es) |
PT (1) | PT72226B (es) |
ZA (1) | ZA807911B (es) |
Families Citing this family (108)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3134780A1 (de) * | 1981-09-02 | 1983-03-10 | Hoechst Ag, 6000 Frankfurt | "sulfonylharnstoffe, verfahren zu ihrer herstellung, pharmazeutische praeparate auf basis dieser verbindungen und ihre verwendung" |
US4985417A (en) * | 1989-05-02 | 1991-01-15 | Trager Seymour F | Treatment of glaucoma |
JP3465247B2 (ja) * | 1992-12-28 | 2003-11-10 | アベンティス ファーマ株式会社 | 動脈硬化症の予防および治療剤 |
DE4344957A1 (de) * | 1993-12-30 | 1995-07-06 | Hoechst Ag | Substituierte Benzolsulfonylharnstoffe und -thioharnstoffe, Herstellungsverfahren und Verwendungsmöglichkeiten pharmazeutischer Präparate auf Basis dieser Verbindungen |
US5631275A (en) * | 1993-12-30 | 1997-05-20 | Hoechst Aktiengesellschaft | Substituted benzenesulfonylureas and -thioureas, preparation processes and possible uses of pharmaceutical preparations based on these compounds |
EA003101B1 (ru) | 1998-03-19 | 2002-12-26 | Бристол-Майерз Сквибб Компани | Двухфазная система доставки с регулируемым высвобождением для фармацевтических средств с высокой растворимостью и способ лечения диабета с помощью этой системы |
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HUP0302700A3 (en) | 2000-08-07 | 2005-05-30 | Ranbaxy Signature Llc Princeto | Liquid formulation of metformin and its use |
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BRPI0416444B8 (pt) | 2003-11-12 | 2021-05-25 | Chiesi Farm Spa | composto de ácido borônico heterocíclico, composição farmacêutica, e, combinação farmacêutica compreendendo o mesmo |
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DE2238870C3 (de) * | 1972-08-07 | 1978-09-28 | Hoechst Ag, 6000 Frankfurt | Benzolsulfonylharnstoffe |
DE2621958A1 (de) * | 1976-05-18 | 1977-12-08 | Hoechst Ag | Benzolsulfonylharnstoffe und verfahren zu ihrer herstellung |
MTP848B (en) * | 1978-06-27 | 1980-06-24 | Hoechst Ag | Sulfonyl ureas process for their manufacture pharmaceutical preparation on the basis of there compounds and their use |
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1979
- 1979-12-19 DE DE19792951135 patent/DE2951135A1/de not_active Withdrawn
-
1980
- 1980-12-04 DE DE8080107588T patent/DE3067390D1/de not_active Expired
- 1980-12-04 EP EP80107588A patent/EP0031058B1/de not_active Expired
- 1980-12-04 AT AT80107588T patent/ATE6934T1/de active
- 1980-12-12 ES ES497661A patent/ES497661A0/es active Granted
- 1980-12-16 MX MX008352A patent/MX174496B/es unknown
- 1980-12-16 MX MX809232U patent/MX6926E/es unknown
- 1980-12-17 GR GR63671A patent/GR72534B/el unknown
- 1980-12-17 FI FI803937A patent/FI75338C/fi not_active IP Right Cessation
- 1980-12-17 HU HU803027A patent/HU184943B/hu unknown
- 1980-12-17 IL IL61733A patent/IL61733A/xx not_active IP Right Cessation
- 1980-12-17 US US06/217,524 patent/US4379785A/en not_active Expired - Lifetime
- 1980-12-18 IE IE2676/80A patent/IE50635B1/en not_active IP Right Cessation
- 1980-12-18 AU AU65523/80A patent/AU538129B2/en not_active Expired
- 1980-12-18 DK DK540280A patent/DK156434C/da not_active IP Right Cessation
- 1980-12-18 ZA ZA00807911A patent/ZA807911B/xx unknown
- 1980-12-18 CA CA000367123A patent/CA1167033A/en not_active Expired
- 1980-12-18 NO NO803855A patent/NO155290C/no not_active IP Right Cessation
- 1980-12-18 PT PT72226A patent/PT72226B/pt unknown
- 1980-12-19 JP JP18117980A patent/JPS56108762A/ja active Granted
- 1980-12-30 ES ES498228A patent/ES8202543A1/es not_active Expired
- 1980-12-30 ES ES498226A patent/ES8202799A1/es not_active Expired
- 1980-12-30 ES ES498225A patent/ES8202798A1/es not_active Expired
- 1980-12-30 ES ES498224A patent/ES498224A0/es active Granted
- 1980-12-30 ES ES498227A patent/ES498227A0/es active Granted
-
1982
- 1982-02-24 AR AR288546A patent/AR230989A1/es active
- 1982-02-24 AR AR288547A patent/AR240922A1/es active
- 1982-02-24 AR AR288545A patent/AR231131A1/es active
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1985
- 1985-03-12 MX MX825485A patent/MX8254A/es unknown
- 1985-03-12 MX MX835285A patent/MX8352A/es unknown
-
1995
- 1995-11-07 NL NL950026C patent/NL950026I2/nl unknown
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1996
- 1996-07-30 NO NO1996009C patent/NO1996009I1/no unknown
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1998
- 1998-05-20 LU LU90244C patent/LU90244I2/fr unknown
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