IL47168A - Mono or dioxo piperazino(thio)carbonylamino derivatives ofpenicillins and cephalosporins and process for producing the same - Google Patents
Mono or dioxo piperazino(thio)carbonylamino derivatives ofpenicillins and cephalosporins and process for producing the sameInfo
- Publication number
- IL47168A IL47168A IL47168A IL4716875A IL47168A IL 47168 A IL47168 A IL 47168A IL 47168 A IL47168 A IL 47168A IL 4716875 A IL4716875 A IL 4716875A IL 47168 A IL47168 A IL 47168A
- Authority
- IL
- Israel
- Prior art keywords
- ofpenicillins
- piperazino
- cephalosporins
- dioxo
- thio
- Prior art date
Links
- -1 dioxo piperazino(thio)carbonylamino Chemical class 0.000 title abstract 2
- 229930186147 Cephalosporin Natural products 0.000 title 1
- 229940124587 cephalosporin Drugs 0.000 title 1
- 150000001780 cephalosporins Chemical class 0.000 title 1
- HTSGKJQDMSTCGS-UHFFFAOYSA-N 1,4-bis(4-chlorophenyl)-2-(4-methylphenyl)sulfonylbutane-1,4-dione Chemical compound C1=CC(C)=CC=C1S(=O)(=O)C(C(=O)C=1C=CC(Cl)=CC=1)CC(=O)C1=CC=C(Cl)C=C1 HTSGKJQDMSTCGS-UHFFFAOYSA-N 0.000 abstract 1
- FKLJPTJMIBLJAV-UHFFFAOYSA-N Compound IV Chemical compound O1N=C(C)C=C1CCCCCCCOC1=CC=C(C=2OCCN=2)C=C1 FKLJPTJMIBLJAV-UHFFFAOYSA-N 0.000 abstract 1
- 125000003342 alkenyl group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000000539 amino acid group Chemical group 0.000 abstract 1
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
- 150000001768 cations Chemical class 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
- 125000000547 substituted alkyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
- C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP5066374A JPS539238B2 (enrdf_load_stackoverflow) | 1974-05-09 | 1974-05-09 | |
| JP5225474A JPS539239B2 (enrdf_load_stackoverflow) | 1974-05-13 | 1974-05-13 | |
| JP6078774A JPS539240B2 (enrdf_load_stackoverflow) | 1974-05-31 | 1974-05-31 | |
| JP9199674A JPS5123284A (en) | 1974-08-13 | 1974-08-13 | Shinkina penishirinruino seizoho |
| JP10995474A JPS5139687A (ja) | 1974-09-26 | 1974-09-26 | Shinkinapenishirinruinoseizoho |
| JP14249974A JPS5170788A (en) | 1974-12-13 | 1974-12-13 | Shinkina sefuarosuhorinruino seizoho |
| JP50037207A JPS51113890A (en) | 1975-03-27 | 1975-03-27 | Method for preparing novel cephalosporins |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL47168A0 IL47168A0 (en) | 1975-06-25 |
| IL47168A true IL47168A (en) | 1979-07-25 |
Family
ID=27564446
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL47168A IL47168A (en) | 1974-05-09 | 1975-04-24 | Mono or dioxo piperazino(thio)carbonylamino derivatives ofpenicillins and cephalosporins and process for producing the same |
| IL53485A IL53485A0 (en) | 1974-05-09 | 1977-11-29 | 2,3-dioxypiperazine derivatives |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL53485A IL53485A0 (en) | 1974-05-09 | 1977-11-29 | 2,3-dioxypiperazine derivatives |
Country Status (18)
Families Citing this family (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL49846A (en) * | 1975-06-24 | 1979-07-25 | Bayer Ag | Penicillin and cephalosporin compounds containing an imidazolidinone ring substituted by a carbocycle or heterocycletheir preparation and pharmaceutical compositions comprising them |
| DE2528079A1 (de) * | 1975-06-24 | 1977-01-20 | Bayer Ag | Penicilline, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel |
| FR2338046A2 (fr) * | 1976-01-19 | 1977-08-12 | Toyama Chemical Co Ltd | Nouvelles cephalosporines, leur procede de preparation et leur application en therapeutique |
| JPS6026800B2 (ja) * | 1976-01-22 | 1985-06-25 | 富山化学工業株式会社 | 新規な７α−メトキシセフアロスポリン類およびその製造法 |
| JPS52106883A (en) * | 1976-02-13 | 1977-09-07 | Toyama Chem Co Ltd | Novel penicillins and cephalosporins |
| JPS5331690A (en) * | 1976-09-01 | 1978-03-25 | Shionogi & Co Ltd | Oxadithiacephalosporins |
| DE2857696C2 (de) * | 1977-07-23 | 1984-08-30 | Toyama Chemical Co. Ltd., Tokio / Tokyo | Cephalosporine |
| DE2810083A1 (de) * | 1978-03-08 | 1979-09-20 | Bayer Ag | Beta-lactam-verbindungen |
| DE2813771A1 (de) * | 1978-03-30 | 1979-10-11 | Bayer Ag | Beta-lactam-verbindungen |
| DE2817228A1 (de) * | 1978-04-20 | 1979-10-31 | Bayer Ag | Verfahren zur herstellung halbsynthetischer beta-lactamantibiotika |
| EP0015240A1 (de) * | 1979-02-16 | 1980-09-03 | Ciba-Geigy Ag | Azacyclyl (thio) ureidoacetyl-Verbindungen und Verfahren zu ihrer Herstellung |
| CA1209477A (en) * | 1981-03-26 | 1986-08-12 | Bruce E. Haeger | Composition of matter comprising a lyophilized preparation of a penicillin derivative |
| CA1200239A (en) * | 1981-03-30 | 1986-02-04 | Donald C. Boop | Process for preparing 6-¬d-(-)-alpha-(4-c1-c4 alkyl- 2,3-dioxo-1-piperazinocarbonyl-amino)- phenylacetamido|penicillanic acid |
| JPS57118587A (en) * | 1981-11-26 | 1982-07-23 | Toyama Chem Co Ltd | Novel penicillin |
| BG46664A1 (en) * | 1985-08-16 | 1990-02-15 | Druzhestven N Izsledovatelski | Method for preparing of 6- /d (-)- alpha- (4- ethyl- 2, 3- dioxo- 1- piperazine carbonylamino)- phenylacetamido/- penicillanic acid |
| DE3619562A1 (de) * | 1986-06-11 | 1987-12-17 | Basf Ag | Verfahren zur herstellung von 2,3-dioxo-4-oxicarbonylpiperazinderivaten, neue 2,3-dioxo-4-oxicarbonylpiperazinderivate und deren verwendung |
| US5859012A (en) * | 1996-04-03 | 1999-01-12 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| USRE39921E1 (en) | 1999-10-07 | 2007-11-13 | Smithkline Beecham Corporation | Chemical compounds |
| GB9923748D0 (en) | 1999-10-07 | 1999-12-08 | Glaxo Group Ltd | Chemical compounds |
| GB0025354D0 (en) | 2000-10-17 | 2000-11-29 | Glaxo Group Ltd | Chemical compounds |
| AU2002332640B2 (en) * | 2001-08-24 | 2007-11-08 | University Of South Florida | Piperazinone compounds as anti-tumor and anti-cancer agents and methods of treatment |
| JP2005522436A (ja) | 2002-02-08 | 2005-07-28 | グラクソ グループ リミテッド | ピペリジルカルボキシアミド誘導体またはそのタキキニン介在疾患の治療における使用 |
| GB0203020D0 (en) | 2002-02-08 | 2002-03-27 | Glaxo Group Ltd | Chemical compounds |
| GB0203022D0 (en) | 2002-02-08 | 2002-03-27 | Glaxo Group Ltd | Chemical compounds |
| JP5173842B2 (ja) * | 2007-01-31 | 2013-04-03 | 富山化学工業株式会社 | ピペラシリンナトリウムの新規な結晶 |
| PT2960244T (pt) | 2008-10-31 | 2016-11-02 | Shionogi & Co | Cefalosporina contendo grupo catecol |
| CA2795322A1 (en) | 2010-04-05 | 2011-10-13 | Shionogi & Co., Ltd. | Cephem compound having catechol group |
| US8883773B2 (en) | 2010-04-05 | 2014-11-11 | Shionogi & Co., Ltd. | Cephem compound having pseudo-catechol group |
| WO2011136268A1 (ja) | 2010-04-28 | 2011-11-03 | 塩野義製薬株式会社 | 新規なセフェム誘導体 |
| JP6006201B2 (ja) | 2011-04-28 | 2016-10-12 | 塩野義製薬株式会社 | カテコールまたは擬似カテコール構造を有する新規セフェム化合物 |
| US9242999B2 (en) | 2011-06-27 | 2016-01-26 | Shionogi & Co., Ltd. | Cephem compound having pyridinium group |
| CN110746445B (zh) * | 2019-10-16 | 2021-03-16 | 深圳海关食品检验检疫技术中心 | 一种头孢哌酮氘代内标物的制备方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1770620A1 (de) * | 1968-06-12 | 1971-11-11 | Bayer Ag | Neue Penicilline |
| DE2104580C3 (de) * | 1971-02-01 | 1981-04-02 | Bayer Ag, 5090 Leverkusen | Acylureidopenicilline |
| DE2025415C3 (de) * | 1970-05-25 | 1981-01-22 | Bayer Ag, 5090 Leverkusen | Verfahren zur Herstellung von cyclischen Acylureido-Penicillinen |
| BE790440A (enrdf_load_stackoverflow) * | 1971-10-23 | 1973-04-24 | Bayer Ag | |
| BE794886A (fr) * | 1972-02-22 | 1973-08-02 | Pfizer | Acides 6-(alpha-(omega-guanidinoalcanoylamino)acylamino)-penicillaniques |
| CH570407A5 (enrdf_load_stackoverflow) * | 1972-03-29 | 1975-12-15 | Ciba Geigy Ag | |
| AR204162A1 (es) * | 1972-05-08 | 1975-11-28 | Yamanouchi Pharma Co Ltd | Proceso para la preparacion de derivados de ampicilina |
-
1975
- 1975-04-24 IL IL47168A patent/IL47168A/xx unknown
- 1975-04-28 CY CY1026A patent/CY1026A/xx unknown
- 1975-04-28 GB GB15360/77A patent/GB1508064A/en not_active Expired
- 1975-04-28 GB GB17557/75A patent/GB1508062A/en not_active Expired
- 1975-04-30 DE DE2560239A patent/DE2560239C2/de not_active Expired
- 1975-04-30 DE DE2519400A patent/DE2519400C3/de not_active Expired
- 1975-05-02 BE BE156035A patent/BE828692A/xx not_active IP Right Cessation
- 1975-05-05 PH PH17137A patent/PH21545A/en unknown
- 1975-05-06 CH CH584775A patent/CH605995A5/xx not_active IP Right Cessation
- 1975-05-06 AR AR258658A patent/AR209607A1/es active
- 1975-05-06 FR FR7514159A patent/FR2269937B1/fr not_active Expired
- 1975-05-07 NL NL7505375.A patent/NL162386C/xx not_active IP Right Cessation
- 1975-05-07 FI FI751340A patent/FI63760C/fi not_active IP Right Cessation
- 1975-05-07 DK DK201975A patent/DK151338C/da not_active IP Right Cessation
- 1975-05-08 HU HUTO1002A patent/HU169633B/hu unknown
- 1975-05-08 DD DD185922A patent/DD117882A5/xx unknown
- 1975-05-09 SE SE7505392A patent/SE431457B/xx not_active IP Right Cessation
-
1976
- 1976-02-10 PH PH18076A patent/PH20534A/en unknown
- 1976-10-22 FR FR7631895A patent/FR2320295A1/fr active Granted
- 1976-11-08 AT AT828976A patent/AT344906B/de not_active IP Right Cessation
- 1976-11-15 PH PH19128A patent/PH22346A/en unknown
- 1976-11-15 PH PH19129A patent/PH22336A/en unknown
-
1977
- 1977-05-25 PH PH19814A patent/PH21987A/en unknown
- 1977-11-29 IL IL53485A patent/IL53485A0/xx not_active IP Right Cessation
-
1978
- 1978-07-27 SE SE7808204A patent/SE435062B/sv not_active IP Right Cessation
-
1979
- 1979-03-01 KE KE2923A patent/KE2923A/xx unknown
- 1979-04-26 HK HK262/79A patent/HK26279A/xx unknown
Also Published As
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