GB1508064A - Amino acid derivatives - Google Patents

Amino acid derivatives

Info

Publication number
GB1508064A
GB1508064A GB1536077A GB1536077A GB1508064A GB 1508064 A GB1508064 A GB 1508064A GB 1536077 A GB1536077 A GB 1536077A GB 1536077 A GB1536077 A GB 1536077A GB 1508064 A GB1508064 A GB 1508064A
Authority
GB
Grant status
Application
Patent type
Prior art keywords
lt
sp
acid
derivatives
amino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB1536077A
Inventor
I Saikawa
S Takano
C Yoshida
Takashima
K Momonoi
S Kuroda
M Komatsu
T Yasuda
Kodama
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Toyama Chemical Co Ltd
Original Assignee
Toyama Chemical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms

Abstract

1508064 N-Piperazinocarbonyl-amino acid derivatives TOYAMA CHEMICAL CO Ltd 28 April 1975 [13 Aug 1974 28 Oct 1974 17 Feb 1975] 15360/77 Divided out of 1508062 Heading C2C Novel compounds I and salts and carboxyl derivatives thereof (R is an amino acid residue; R<SP>2</SP> and R<SP>3</SP> are H or alkyl and R<SP>2</SP> and R<SP>3</SP> are both linked to the same carbon atom; and A is H or an optionally substituted alkyl, alkenyl, aryl or aralkyl group) are prepared by reaction of a compound II NH 2 RCOOR<SP>1</SP> (III) (R<SP>1</SP> is H or a cation) with a reactive derivative of a compound IV
GB1536077A 1974-05-09 1975-04-28 Amino acid derivatives Expired GB1508064A (en)

Priority Applications (7)

Application Number Priority Date Filing Date Title
JP5066374A JPS539238B2 (en) 1974-05-09 1974-05-09
JP5225474A JPS539239B2 (en) 1974-05-13 1974-05-13
JP6078774A JPS539240B2 (en) 1974-05-31 1974-05-31
JP9199674A JPS5320996B2 (en) 1974-08-13 1974-08-13
JP10995474A JPS5310074B2 (en) 1974-09-26 1974-09-26
JP14249974A JPS5310075B2 (en) 1974-12-13 1974-12-13
JP3720775A JPS5320518B2 (en) 1975-03-27 1975-03-27

Publications (1)

Publication Number Publication Date
GB1508064A true true GB1508064A (en) 1978-04-19

Family

ID=27564446

Family Applications (2)

Application Number Title Priority Date Filing Date
GB1536077A Expired GB1508064A (en) 1974-05-09 1975-04-28 Amino acid derivatives
GB1755775A Expired GB1508062A (en) 1974-05-09 1975-04-28 Penicillins and cephalosporins and process for producing the same

Family Applications After (1)

Application Number Title Priority Date Filing Date
GB1755775A Expired GB1508062A (en) 1974-05-09 1975-04-28 Penicillins and cephalosporins and process for producing the same

Country Status (7)

Country Link
BE (1) BE828692A (en)
DE (2) DE2519400C3 (en)
DK (1) DK151338C (en)
FI (1) FI63760C (en)
FR (2) FR2269937B1 (en)
GB (2) GB1508064A (en)
NL (1) NL162386C (en)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1538284A (en) * 1975-06-24 1979-01-17 Bayer Ag 2-oxo-imidazolidine(-yl-carbonyl or thiocarbonylamino)-acetamido penicillins and cephalosporins
DE2528079A1 (en) * 1975-06-24 1977-01-20 Bayer Ag Penicillins, methods for their manufacture and their use as medicines
FR2338046B2 (en) * 1976-01-19 1979-07-20 Toyama Chemical Co Ltd
JPS6026800B2 (en) * 1976-01-22 1985-06-25 Toyama Chemical Co Ltd
JPS52106883A (en) * 1976-02-13 1977-09-07 Toyama Chem Co Ltd Novel penicillins and cephalosporins
JPS612672B2 (en) * 1976-09-01 1986-01-27 Shionogi & Co
DE2857696C2 (en) * 1977-07-23 1984-08-30 Toyama Chemical Co. Ltd., Tokio / Tokyo, Jp
DE2810083A1 (en) * 1978-03-08 1979-09-20 Bayer Ag Beta-lactam compounds
DE2813771A1 (en) * 1978-03-30 1979-10-11 Bayer Ag Beta-lactam compounds
DE2817228A1 (en) * 1978-04-20 1979-10-31 Bayer Ag A process for the production of semisynthetic beta-lactam antibiotics
EP0015240A1 (en) * 1979-02-16 1980-09-03 Ciba-Geigy Ag Azacyclyl (thio) ureidoacetyl compounds and their preparation
CA1200239A (en) * 1981-03-30 1986-02-04 Donald C. Boop Process for preparing 6-¬d-(-)-alpha-(4-c1-c4 alkyl- 2,3-dioxo-1-piperazinocarbonyl-amino)- phenylacetamido|penicillanic acid
JPS57118587A (en) * 1981-11-26 1982-07-23 Toyama Chem Co Ltd Novel penicillin
GB2179348B (en) * 1985-08-16 1989-08-02 Dso Pharmachim Process for the preparation of 6-d-(a)-(4-ethyl-2,3-dioxo-1-piperazinylcarbonylamino)-d-phenylacetamido-penicillanic acid
DE3619562A1 (en) * 1986-06-11 1987-12-17 Basf Ag A process for the preparation of 2,3-dioxo-4-oxicarbonylpiperazinderivaten new 2,3-dioxo-4-oxicarbonylpiperazinderivate and their use
US5859012A (en) * 1996-04-03 1999-01-12 Merck & Co., Inc. Inhibitors of farnesyl-protein transferase
GB9923748D0 (en) 1999-10-07 1999-12-08 Glaxo Group Ltd Chemical compounds
USRE39921E1 (en) 1999-10-07 2007-11-13 Smithkline Beecham Corporation Chemical compounds
GB0025354D0 (en) 2000-10-17 2000-11-29 Glaxo Group Ltd Chemical compounds
EP1427418B1 (en) * 2001-08-24 2009-11-11 Yale University Piperazinone compounds as anti-tumor and anti-cancer agents
GB0203020D0 (en) 2002-02-08 2002-03-27 Glaxo Group Ltd Chemical compounds
GB0203022D0 (en) 2002-02-08 2002-03-27 Glaxo Group Ltd Chemical compounds
EP1472222A1 (en) 2002-02-08 2004-11-03 Glaxo Group Limited Piperidylcarboxamide derivatives and their use in the treatment of tachykinim-mediated diseases
RU2009132516A (en) * 2007-01-31 2011-03-10 Тояма Кемикал Ко., Лтд. (Jp) The new crystalline form piperatsillinnatriya
ES2564836T3 (en) 2008-10-31 2016-03-29 Shionogi & Co., Ltd. Cephalosporins having a group catechol
CA2795322A1 (en) 2010-04-05 2011-10-13 Shionogi & Co., Ltd. Cephem compound having catechol group
WO2011125966A1 (en) 2010-04-05 2011-10-13 塩野義製薬株式会社 Cephem compound having pseudo-catechol group
JP5852562B2 (en) 2010-04-28 2016-02-03 塩野義製薬株式会社 The novel cephem derivatives
CN103635478A (en) 2011-04-28 2014-03-12 盐野义制药株式会社 Novel cephem compound having catechol or pseudo-catechol structure
CN103619853A (en) 2011-06-27 2014-03-05 盐野义制药株式会社 Cephem compound having pyridinium group

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1770620A1 (en) * 1968-06-12 1971-11-11 Bayer Ag new penicillins
DE2025415C3 (en) * 1970-05-25 1981-01-22 Bayer Ag, 5090 Leverkusen
DE2104580C3 (en) * 1971-02-01 1981-04-02 Bayer Ag, 5090 Leverkusen, De
BE790440A (en) * 1971-10-23 1973-04-24 Bayer Ag
BE794886A (en) * 1972-02-22 1973-08-02 Pfizer 6 acids (alpha (omega-guanidinoalcanoylamino) acylamino) -penicillaniques
DE2313667A1 (en) * 1972-03-29 1973-10-11 Ciba Geigy Ag New derivatives of penam-3-carboxylic acid and cephem-4-carboxylic acid and process for their manufacture
CA1050971A (en) * 1972-05-08 1979-03-20 Yamanouchi Pharmaceutical Co. Process for the preparation of ampicillin derivatives substituted by heterocyclic acyl group

Also Published As

Publication number Publication date Type
FR2320295B1 (en) 1980-11-07 grant
NL162386B (en) 1979-12-17 application
NL162386C (en) 1980-05-16 grant
DE2519400B2 (en) 1981-05-21 application
DK151338C (en) 1988-07-18 grant
FR2269937A1 (en) 1975-12-05 application
FI751340A (en) 1975-11-10 application
FI63760B (en) 1983-04-29 application
DK201975A (en) 1975-11-10 application
BE828692A (en) 1975-11-03 grant
DK151338B (en) 1987-11-23 grant
DE2519400C3 (en) 1982-02-11 grant
NL7505375A (en) 1975-11-11 application
BE828692A1 (en) grant
GB1508062A (en) 1978-04-19 application
FR2320295A1 (en) 1977-03-04 application
DE2560239C2 (en) 1984-10-11 grant
FI63760C (en) 1983-08-10 grant
DE2519400A1 (en) 1976-03-04 application
FR2269937B1 (en) 1979-06-15 grant

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Legal Events

Date Code Title Description
PS Patent sealed
704A Declaration that licence is not available as of right for an excepted use (par. 4a/1977)
PE20 Patent expired after termination of 20 years

Effective date: 19950427