New! Search for patents from more than 100 countries including Australia, Brazil, Sweden and more

NL7505375A - New penicillin and cephalosporin derivatives and process for the preparation thereof. - Google Patents

New penicillin and cephalosporin derivatives and process for the preparation thereof.

Info

Publication number
NL7505375A
NL7505375A NL7505375A NL7505375A NL7505375A NL 7505375 A NL7505375 A NL 7505375A NL 7505375 A NL7505375 A NL 7505375A NL 7505375 A NL7505375 A NL 7505375A NL 7505375 A NL7505375 A NL 7505375A
Authority
NL
NETHERLANDS
Prior art keywords
sp
gt
lt
preparation
process
Prior art date
Application number
NL7505375A
Other languages
Dutch (nl)
Other versions
NL162386B (en
NL162386C (en
Inventor
I Saikawa
S Takano
C Yoshida
Takashima
K Momonoi
S Kuroda
M Komatsu
T Yasuda
Kodama
Original Assignee
Toyama Chemical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to JP5066374A priority Critical patent/JPS539238B2/ja
Priority to JP5225474A priority patent/JPS539239B2/ja
Priority to JP6078774A priority patent/JPS539240B2/ja
Priority to JP9199674A priority patent/JPS5320996B2/ja
Priority to JP10995474A priority patent/JPS5310074B2/ja
Priority to JP14249974A priority patent/JPS5310075B2/ja
Priority to JP3720775A priority patent/JPS5320518B2/ja
Application filed by Toyama Chemical Co Ltd filed Critical Toyama Chemical Co Ltd
Publication of NL7505375A publication Critical patent/NL7505375A/en
Publication of NL162386B publication Critical patent/NL162386B/en
Application granted granted Critical
Publication of NL162386C publication Critical patent/NL162386C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms

Abstract

1508064 N-Piperazinocarbonyl-amino acid derivatives TOYAMA CHEMICAL CO Ltd 28 April 1975 [13 Aug 1974 28 Oct 1974 17 Feb 1975] 15360/77 Divided out of 1508062 Heading C2C Novel compounds I and salts and carboxyl derivatives thereof (R is an amino acid residue; R<SP>2</SP> and R<SP>3</SP> are H or alkyl and R<SP>2</SP> and R<SP>3</SP> are both linked to the same carbon atom; and A is H or an optionally substituted alkyl, alkenyl, aryl or aralkyl group) are prepared by reaction of a compound II NH 2 RCOOR<SP>1</SP> (III) (R<SP>1</SP> is H or a cation) with a reactive derivative of a compound IV
NL7505375A 1974-05-09 1975-05-07 Process for the preparation of a composition having anti-bacterial effect and process for the preparation of such a formulation suitable for inclusion into compounds. NL162386C (en)

Priority Applications (7)

Application Number Priority Date Filing Date Title
JP5066374A JPS539238B2 (en) 1974-05-09 1974-05-09
JP5225474A JPS539239B2 (en) 1974-05-13 1974-05-13
JP6078774A JPS539240B2 (en) 1974-05-31 1974-05-31
JP9199674A JPS5320996B2 (en) 1974-08-13 1974-08-13
JP10995474A JPS5310074B2 (en) 1974-09-26 1974-09-26
JP14249974A JPS5310075B2 (en) 1974-12-13 1974-12-13
JP3720775A JPS5320518B2 (en) 1975-03-27 1975-03-27

Publications (3)

Publication Number Publication Date
NL7505375A true NL7505375A (en) 1975-11-11
NL162386B NL162386B (en) 1979-12-17
NL162386C NL162386C (en) 1980-05-16

Family

ID=27564446

Family Applications (1)

Application Number Title Priority Date Filing Date
NL7505375A NL162386C (en) 1974-05-09 1975-05-07 Process for the preparation of a composition having anti-bacterial effect and process for the preparation of such a formulation suitable for inclusion into compounds.

Country Status (18)

Country Link
AR (1) AR209607A1 (en)
AT (1) AT344906B (en)
BE (1) BE828692A (en)
CH (1) CH605995A5 (en)
CY (1) CY1026A (en)
DD (1) DD117882A5 (en)
DE (2) DE2560239C2 (en)
DK (1) DK151338C (en)
FI (1) FI63760C (en)
FR (2) FR2269937B1 (en)
GB (2) GB1508064A (en)
HK (1) HK26279A (en)
HU (1) HU169633B (en)
IL (2) IL47168A (en)
KE (1) KE2923A (en)
NL (1) NL162386C (en)
PH (5) PH21545A (en)
SE (3) SE7505392L (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2338046A2 (en) * 1976-01-19 1977-08-12 Toyama Chemical Co Ltd Broad-spectrum cephalosporin antibiotics resistant to beta-lactamase - 7-(alpha-(4pethyl-2,3-dioxo-piperazinocarbonylamino)-para-hydroxy- phenylacetamido)-ceph-3-em-4-carboxylic acids

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL49846A (en) * 1975-06-24 1979-07-25 Bayer Ag Penicillin and cephalosporin compounds containing an imidazolidinone ring substituted by a carbocycle or heterocycletheir preparation and pharmaceutical compositions comprising them
DE2528079A1 (en) * 1975-06-24 1977-01-20 Bayer Ag Penicillins, methods for their manufacture and their use as medicines
JPS6026800B2 (en) * 1976-01-22 1985-06-25 Toyama Chemical Co Ltd
JPS52106883A (en) * 1976-02-13 1977-09-07 Toyama Chem Co Ltd Novel penicillins and cephalosporins
JPS612672B2 (en) * 1976-09-01 1986-01-27 Shionogi & Co
DE2857696C2 (en) * 1977-07-23 1984-08-30 Toyama Chemical Co. Ltd., Tokio / Tokyo, Jp
DE2810083A1 (en) * 1978-03-08 1979-09-20 Bayer Ag Beta-lactam compounds
DE2813771A1 (en) * 1978-03-30 1979-10-11 Bayer Ag Beta-lactam compounds
DE2817228A1 (en) * 1978-04-20 1979-10-31 Bayer Ag A process for the production of semisynthetic beta-lactam antibiotics
EP0015240A1 (en) * 1979-02-16 1980-09-03 Ciba-Geigy Ag Azacyclyl (thio) ureidoacetyl compounds and their preparation
CA1209477A (en) * 1981-03-26 1986-08-12 Bruce E. Haeger Composition of matter comprising a lyophilized preparation of a penicillin derivative
CA1200239A (en) * 1981-03-30 1986-02-04 Donald C. Boop Process for preparing 6-¬d-(-)-alpha-(4-c1-c4 alkyl- 2,3-dioxo-1-piperazinocarbonyl-amino)- phenylacetamido|penicillanic acid
JPS57118587A (en) * 1981-11-26 1982-07-23 Toyama Chem Co Ltd Novel penicillin
BG46664A1 (en) * 1985-08-16 1990-02-15 Druzhestven N Izsledovatelski Method for preparing of 6- /d (-)- alpha- (4- ethyl- 2, 3- dioxo- 1- piperazine carbonylamino)- phenylacetamido/- penicillanic acid
DE3619562A1 (en) * 1986-06-11 1987-12-17 Basf Ag A process for the preparation of 2,3-dioxo-4-oxicarbonylpiperazinderivaten new 2,3-dioxo-4-oxicarbonylpiperazinderivate and their use
US5859012A (en) * 1996-04-03 1999-01-12 Merck & Co., Inc. Inhibitors of farnesyl-protein transferase
USRE39921E1 (en) 1999-10-07 2007-11-13 Smithkline Beecham Corporation Chemical compounds
GB9923748D0 (en) 1999-10-07 1999-12-08 Glaxo Group Ltd Chemical compounds
GB0025354D0 (en) 2000-10-17 2000-11-29 Glaxo Group Ltd Chemical compounds
AT530184T (en) * 2001-08-24 2011-11-15 Univ Yale Piperazinone compounds active ingredients as tumor- and cancer-fighting
GB0203020D0 (en) 2002-02-08 2002-03-27 Glaxo Group Ltd Chemical compounds
GB0203022D0 (en) 2002-02-08 2002-03-27 Glaxo Group Ltd Chemical compounds
EP1472222A1 (en) 2002-02-08 2004-11-03 Glaxo Group Limited Piperidylcarboxamide derivatives and their use in the treatment of tachykinim-mediated diseases
RU2009132516A (en) * 2007-01-31 2011-03-10 Тояма Кемикал Ко., Лтд. (Jp) The new crystalline form piperatsillinnatriya
PE00102012A1 (en) 2008-10-31 2012-02-07 Shionogi & Co Cephalosporins having a group catechol
MX2012011521A (en) 2010-04-05 2013-03-08 Shionogi & Co Cephem compound having catechol group.
WO2011125966A1 (en) 2010-04-05 2011-10-13 塩野義製薬株式会社 Cephem compound having pseudo-catechol group
JP5852562B2 (en) 2010-04-28 2016-02-03 塩野義製薬株式会社 The novel cephem derivatives
CN103635478A (en) 2011-04-28 2014-03-12 盐野义制药株式会社 Novel cephem compound having catechol or pseudo-catechol structure
CN103619853A (en) 2011-06-27 2014-03-05 盐野义制药株式会社 Cephem compound having pyridinium group

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1770620A1 (en) * 1968-06-12 1971-11-11 Bayer Ag new penicillins
DE2025415C3 (en) * 1970-05-25 1981-01-22 Bayer Ag, 5090 Leverkusen
DE2104580C3 (en) * 1971-02-01 1981-04-02 Bayer Ag, 5090 Leverkusen, De
BE790440A (en) * 1971-10-23 1973-04-24 Bayer Ag
BE794886A (en) * 1972-02-22 1973-08-02 Pfizer 6 acids (alpha (omega-guanidinoalcanoylamino) acylamino) -penicillaniques
CH570407A5 (en) * 1972-03-29 1975-12-15 Ciba Geigy Ag
AR204162A1 (en) * 1972-05-08 1975-11-28 Yamanouchi Pharma Co Ltd Process for the preparation of derivatives of ampicillin

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2338046A2 (en) * 1976-01-19 1977-08-12 Toyama Chemical Co Ltd Broad-spectrum cephalosporin antibiotics resistant to beta-lactamase - 7-(alpha-(4pethyl-2,3-dioxo-piperazinocarbonylamino)-para-hydroxy- phenylacetamido)-ceph-3-em-4-carboxylic acids

Also Published As

Publication number Publication date
HU169633B (en) 1976-12-28
PH20534A (en) 1987-02-09
SE7505392L (en) 1975-12-23
ATA828976A (en) 1977-12-15
FR2320295B1 (en) 1980-11-07
NL162386B (en) 1979-12-17
HK26279A (en) 1979-05-04
KE2923A (en) 1979-04-06
NL162386C (en) 1980-05-16
AR209607A1 (en) 1977-05-13
IL47168A (en) 1979-07-25
DE2519400B2 (en) 1981-05-21
PH22346A (en) 1988-08-12
DK151338C (en) 1988-07-18
IL53485D0 (en) 1978-01-31
PH21545A (en) 1987-12-11
SE435062B (en) 1984-09-03
AT344906B (en) 1978-08-25
FR2269937A1 (en) 1975-12-05
FI751340A (en) 1975-11-10
FI63760B (en) 1983-04-29
DK201975A (en) 1975-11-10
BE828692A (en) 1975-11-03
DK151338B (en) 1987-11-23
CH605995A5 (en) 1978-10-13
DE2519400C3 (en) 1982-02-11
AU8043175A (en) 1976-10-28
IL47168D0 (en) 1975-06-25
GB1508064A (en) 1978-04-19
BE828692A1 (en)
CY1026A (en) 1980-08-01
SE7808204A (en) 1978-07-27
DD117882A5 (en) 1976-02-05
PH22336A (en) 1988-08-12
GB1508062A (en) 1978-04-19
FR2320295A1 (en) 1977-03-04
SE431457B (en) 1984-02-06
DE2560239C2 (en) 1984-10-11
FI63760C (en) 1983-08-10
DE2519400A1 (en) 1976-03-04
FR2269937B1 (en) 1979-06-15
PH21987A (en) 1988-05-02

Similar Documents

Publication Publication Date Title
GB1398421A (en) Sulphosuccinate derivatives for use as detergent builders
GB1433920A (en) Alkanolamine derivatives
GB1053825A (en)
GB1465661A (en) Stilbene derivatives
GB1203149A (en) Piperidine derivatives
GB1425354A (en) Indole derivatives
GB1309743A (en) Dyeing keratinous fibres
JPS5265263A (en) Azetidinone compounds
GB1212174A (en) Process for the production of new 2-oxo-1,2-dihydroquinoline derivatives
GB1412546A (en) Morpholine derivatives
GB1139985A (en) Basically substituted 2-imidazolidone derivatives and their production
GB1183648A (en) Acrylic Acid Derivatives for Hardening Gelatine
GB1427139A (en) Penicillins
GB1445257A (en) Preparation
GB1269776A (en) Epoxides and halohydrins and conversion thereof to alkanolamine derivatives
GB1531963A (en) Pyrido(1,2alpha)pyrimidine derivatives
GB1436502A (en) Amide derivatives of 3-benzoylphenyl-alkanoic acids
GB1126672A (en) Sulphamylanthranilic acid amides and process for their manufacture
GB1461750A (en)
GB1513824A (en) 1,3,4,6,7,11b-hexahydro-2h-benzo(a)quinolizine derivative
GB1368074A (en) Substituted beta-lactams and their preparation
FR2414508A1 (en) Process for the production of cephalosporin
GB1434405A (en) Phenyl-benzoic acid derivatives
GB1456627A (en) Pyridobenzodiazepinones
GB1434580A (en) Disubstituted piperazines

Legal Events

Date Code Title Description
V4 Lapsed because of reaching the maxim lifetime of a patent