IL299730A - Production method of 1,3-benzodioxole derivative - Google Patents

Production method of 1,3-benzodioxole derivative

Info

Publication number
IL299730A
IL299730A IL299730A IL29973023A IL299730A IL 299730 A IL299730 A IL 299730A IL 299730 A IL299730 A IL 299730A IL 29973023 A IL29973023 A IL 29973023A IL 299730 A IL299730 A IL 299730A
Authority
IL
Israel
Prior art keywords
formula
production method
compound represented
solvent
iii
Prior art date
Application number
IL299730A
Other languages
English (en)
Hebrew (he)
Original Assignee
Daiichi Sankyo Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Sankyo Co Ltd filed Critical Daiichi Sankyo Co Ltd
Publication of IL299730A publication Critical patent/IL299730A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00Preparation of carboxylic acid esters
    • C07C67/30Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
    • C07C67/307Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by introduction of halogen; by substitution of halogen atoms by other halogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/76Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring
    • C07C69/84Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring of monocyclic hydroxy carboxylic acids, the hydroxy groups and the carboxyl groups of which are bound to carbon atoms of a six-membered aromatic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D317/00Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Light Receiving Elements (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL299730A 2020-07-08 2021-07-07 Production method of 1,3-benzodioxole derivative IL299730A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2020117639 2020-07-08
PCT/JP2021/025537 WO2022009911A1 (ja) 2020-07-08 2021-07-07 1,3-ベンゾジオキソール誘導体の製造方法

Publications (1)

Publication Number Publication Date
IL299730A true IL299730A (en) 2023-03-01

Family

ID=79553255

Family Applications (1)

Application Number Title Priority Date Filing Date
IL299730A IL299730A (en) 2020-07-08 2021-07-07 Production method of 1,3-benzodioxole derivative

Country Status (9)

Country Link
US (1) US20230257368A1 (https=)
EP (1) EP4180426A4 (https=)
JP (1) JP7720846B2 (https=)
KR (1) KR20230037488A (https=)
CN (1) CN116018335B (https=)
BR (1) BR112022026641A2 (https=)
IL (1) IL299730A (https=)
TW (1) TW202216654A (https=)
WO (1) WO2022009911A1 (https=)

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7208630B2 (en) * 2004-10-27 2007-04-24 University Of Kansas Heat shock protein 90 inhibitors
JP2007161674A (ja) * 2005-12-16 2007-06-28 Tanabe Seiyaku Co Ltd ピペリジン化合物およびその製法
WO2008071646A1 (en) * 2006-12-11 2008-06-19 Boehringer Ingelheim International Gmbh New pyridazine derivatives with mch antagonistic activity and medicaments comprising these compounds
LT3121175T (lt) * 2014-03-17 2020-03-10 Daiichi Sankyo Company, Limited 1,3-benzodioksazolo dariniai, kaip ezh1 ir (arba) ezh2 inhibitoriai
BR112018001688B1 (pt) * 2015-07-30 2023-05-02 Daiichi Sankyo Company, Limited Uso de um composto
CN106883125A (zh) * 2017-03-07 2017-06-23 怀化金鑫新材料有限公司 感光材料稳定剂4‑十六烷氧羰基氧基‑3,5‑二氯苯甲酸乙酯的合成方法
HRP20240793T1 (hr) * 2018-04-18 2024-09-13 Constellation Pharmaceuticals, Inc. Modulatori enzima koji modificiraju metil, njihovi pripravci i upotreba
EP3797108B1 (en) * 2018-05-21 2022-07-20 Constellation Pharmaceuticals, Inc. Modulators of methyl modifying enzymes, compositions and uses thereof
JP2020045306A (ja) * 2018-09-18 2020-03-26 第一三共株式会社 ヘテロシクロアルキル環を含むアミド誘導体

Also Published As

Publication number Publication date
JP7720846B2 (ja) 2025-08-08
EP4180426A1 (en) 2023-05-17
TW202216654A (zh) 2022-05-01
KR20230037488A (ko) 2023-03-16
BR112022026641A2 (pt) 2023-02-07
CA3185274A1 (en) 2022-01-13
EP4180426A4 (en) 2024-08-07
US20230257368A1 (en) 2023-08-17
WO2022009911A1 (ja) 2022-01-13
CN116018335A (zh) 2023-04-25
JPWO2022009911A1 (https=) 2022-01-13
CN116018335B (zh) 2025-10-10

Similar Documents

Publication Publication Date Title
KR20200087670A (ko) L-글루포시네이트 제조 방법
CA2491472C (en) Process for the preparation of n-monosubstituted .beta.-amino alcohols
WO2020094434A1 (en) Process for preparation of optically enriched isoxazolines
IL299730A (en) Production method of 1,3-benzodioxole derivative
EP1758855B1 (en) Process for preparing 2-oxo-1-pyrrolidine derivatives by intramolecular allylation
Jung et al. Facile chemical synthesis of S, S-isodityrosine, a naturally-occurring cross-linking amino acid
CN104557583B (zh) 一种合成γ-氨基丁酸类手性化合物的方法
KR100360139B1 (ko) 사이클로프로판 유도체 및 이의 제조방법
DE60031299T2 (de) Verfahren zur industriellen Herstellung von (Aminomethyl)trifluormethlcarbinol-Derivaten
NZ502786A (en) Preparation of gabapentin analogues comprised of adding cyclohexanone to sodium hydride and finally heating the formed lactam in HCl and dioxan
IL299619A (en) METHOD FOR THE PREPARATION OF AN INTERMEDIATE COMPOUND OF URACIL CONTAINING ISOXAZOLINE
CN117015542B (zh) 吡咯并吡啶衍生物的制备方法
Nguyen et al. Practical asymmetric access to carboxy-differentiated aspartate derivatives via 1, 3-dipolar cycloaddition of a nitrone with (R)-4-ethyl-N-vinyloxazolidin-2-one
CA3058183A1 (en) Synthetic processes and synthetic intermediates towardthe production of txa709
US9067868B2 (en) Chemical process for opening ring compounds
EP2426116B1 (de) Verfahren zur Herstellung von (S)-3-N-Methylamino-1-(2-thienyl)-1-propanol
JPH05194380A (ja) 置換されたピロリジン
EP1991524A1 (en) A process for the preparation of phenylcarbamates
KR101859586B1 (ko) 라코사마이드 또는 이의 유사체의 제조방법
EP0726897A1 (en) Process for the preparation of n-4- (substituted phenyl)alkylthienyl]-, and n-4- (substituted phenyl)alkylfuryl]but-3-yn-2-yl]-n-hydroxyurea compounds
US6433170B1 (en) Method for producing 4-[2',5'-diamino-6'-halopyrimidine-4'-yl)amino]- cyclopent-2-enylmethanols
Chandra Babu et al. Asymmetric synthesis of chiral amines by highly diastereoselective 1, 2-additions of organometallic reagents to N-tert-butanesulfinyl imines
JPH09227471A (ja) N−アルキル−n−(ヒドロキシアルキル)アミンの製法
KR20010108170A (ko) O-티오카바모일-아미노알카놀 화합물, 이의 약학적 허용염 및 제조방법
MXPA99011865A (es) Proceso para la preparacion de 5-hidroximetiltiazoles