JP7720846B2 - １，３－ベンゾジオキソール誘導体の製造方法 - Google Patents
１，３－ベンゾジオキソール誘導体の製造方法Info
- Publication number
- JP7720846B2 JP7720846B2 JP2022535364A JP2022535364A JP7720846B2 JP 7720846 B2 JP7720846 B2 JP 7720846B2 JP 2022535364 A JP2022535364 A JP 2022535364A JP 2022535364 A JP2022535364 A JP 2022535364A JP 7720846 B2 JP7720846 B2 JP 7720846B2
- Authority
- JP
- Japan
- Prior art keywords
- formula
- added
- mixture
- mol
- stirred
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C67/00—Preparation of carboxylic acid esters
- C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
- C07C67/307—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by introduction of halogen; by substitution of halogen atoms by other halogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/76—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring
- C07C69/84—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring of monocyclic hydroxy carboxylic acids, the hydroxy groups and the carboxyl groups of which are bound to carbon atoms of a six-membered aromatic ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/56—Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Light Receiving Elements (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2020117639 | 2020-07-08 | ||
| JP2020117639 | 2020-07-08 | ||
| PCT/JP2021/025537 WO2022009911A1 (ja) | 2020-07-08 | 2021-07-07 | １，３－ベンゾジオキソール誘導体の製造方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPWO2022009911A1 JPWO2022009911A1 (https=) | 2022-01-13 |
| JP7720846B2 true JP7720846B2 (ja) | 2025-08-08 |
Family
ID=79553255
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022535364A Active JP7720846B2 (ja) | 2020-07-08 | 2021-07-07 | １，３－ベンゾジオキソール誘導体の製造方法 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20230257368A1 (https=) |
| EP (1) | EP4180426A4 (https=) |
| JP (1) | JP7720846B2 (https=) |
| KR (1) | KR20230037488A (https=) |
| CN (1) | CN116018335B (https=) |
| BR (1) | BR112022026641A2 (https=) |
| IL (1) | IL299730A (https=) |
| TW (1) | TW202216654A (https=) |
| WO (1) | WO2022009911A1 (https=) |
Citations (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2007161674A (ja) | 2005-12-16 | 2007-06-28 | Tanabe Seiyaku Co Ltd | ピペリジン化合物およびその製法 |
| JP2010512366A (ja) | 2006-12-11 | 2010-04-22 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Ｍｃｈ拮抗活性を有する新規ピリダジン誘導体及びこれらの化合物を含む薬物 |
| WO2015141616A1 (ja) | 2014-03-17 | 2015-09-24 | 第一三共株式会社 | １，３－ベンゾジオキソール誘導体 |
| JP6009135B1 (ja) | 2015-07-30 | 2016-10-19 | 第一三共株式会社 | 成人ｔ細胞白血病リンパ腫の治療及び／又は予防剤 |
| WO2019204490A1 (en) | 2018-04-18 | 2019-10-24 | Constellation Pharmaceuticals, Inc. | Modulators of methyl modifying enzymes, compositions and uses thereof |
| WO2019226491A1 (en) | 2018-05-21 | 2019-11-28 | Constellation Pharmaceuticals, Inc. | Modulators of methyl modifying enzymes, compositions and uses thereof |
| JP2020045306A (ja) | 2018-09-18 | 2020-03-26 | 第一三共株式会社 | ヘテロシクロアルキル環を含むアミド誘導体 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7208630B2 (en) * | 2004-10-27 | 2007-04-24 | University Of Kansas | Heat shock protein 90 inhibitors |
| CN106883125A (zh) * | 2017-03-07 | 2017-06-23 | 怀化金鑫新材料有限公司 | 感光材料稳定剂4‑十六烷氧羰基氧基‑3，5‑二氯苯甲酸乙酯的合成方法 |
-
2021
- 2021-07-07 CN CN202180046125.6A patent/CN116018335B/zh active Active
- 2021-07-07 US US18/012,090 patent/US20230257368A1/en active Pending
- 2021-07-07 TW TW110124923A patent/TW202216654A/zh unknown
- 2021-07-07 WO PCT/JP2021/025537 patent/WO2022009911A1/ja not_active Ceased
- 2021-07-07 KR KR1020227040350A patent/KR20230037488A/ko active Pending
- 2021-07-07 EP EP21836791.0A patent/EP4180426A4/en active Pending
- 2021-07-07 BR BR112022026641A patent/BR112022026641A2/pt unknown
- 2021-07-07 JP JP2022535364A patent/JP7720846B2/ja active Active
- 2021-07-07 IL IL299730A patent/IL299730A/en unknown
Patent Citations (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2007161674A (ja) | 2005-12-16 | 2007-06-28 | Tanabe Seiyaku Co Ltd | ピペリジン化合物およびその製法 |
| JP2010512366A (ja) | 2006-12-11 | 2010-04-22 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Ｍｃｈ拮抗活性を有する新規ピリダジン誘導体及びこれらの化合物を含む薬物 |
| WO2015141616A1 (ja) | 2014-03-17 | 2015-09-24 | 第一三共株式会社 | １，３－ベンゾジオキソール誘導体 |
| US20170073335A1 (en) | 2014-03-17 | 2017-03-16 | Daiichi Sankyo Company, Limited | 1,3-benzodioxole derivative |
| JP6009135B1 (ja) | 2015-07-30 | 2016-10-19 | 第一三共株式会社 | 成人ｔ細胞白血病リンパ腫の治療及び／又は予防剤 |
| WO2019204490A1 (en) | 2018-04-18 | 2019-10-24 | Constellation Pharmaceuticals, Inc. | Modulators of methyl modifying enzymes, compositions and uses thereof |
| WO2019226491A1 (en) | 2018-05-21 | 2019-11-28 | Constellation Pharmaceuticals, Inc. | Modulators of methyl modifying enzymes, compositions and uses thereof |
| JP2020045306A (ja) | 2018-09-18 | 2020-03-26 | 第一三共株式会社 | ヘテロシクロアルキル環を含むアミド誘導体 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP4180426A1 (en) | 2023-05-17 |
| TW202216654A (zh) | 2022-05-01 |
| KR20230037488A (ko) | 2023-03-16 |
| BR112022026641A2 (pt) | 2023-02-07 |
| IL299730A (en) | 2023-03-01 |
| CA3185274A1 (en) | 2022-01-13 |
| EP4180426A4 (en) | 2024-08-07 |
| US20230257368A1 (en) | 2023-08-17 |
| WO2022009911A1 (ja) | 2022-01-13 |
| CN116018335A (zh) | 2023-04-25 |
| JPWO2022009911A1 (https=) | 2022-01-13 |
| CN116018335B (zh) | 2025-10-10 |
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