TW202216654A - 1,3-苯并二㗁呃衍生物之製造方法 - Google Patents

1,3-苯并二㗁呃衍生物之製造方法 Download PDF

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Publication number
TW202216654A
TW202216654A TW110124923A TW110124923A TW202216654A TW 202216654 A TW202216654 A TW 202216654A TW 110124923 A TW110124923 A TW 110124923A TW 110124923 A TW110124923 A TW 110124923A TW 202216654 A TW202216654 A TW 202216654A
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TW
Taiwan
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formula
mol
added
compound
production method
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TW110124923A
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English (en)
Chinese (zh)
Inventor
上田剛
海谷雄士
內田貴久
今井誠
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日商第一三共股份有限公司
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Publication of TW202216654A publication Critical patent/TW202216654A/zh

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00—Preparation of carboxylic acid esters
    • C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
    • C07C67/307—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by introduction of halogen; by substitution of halogen atoms by other halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/76—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring
    • C07C69/84—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring of monocyclic hydroxy carboxylic acids, the hydroxy groups and the carboxyl groups of which are bound to carbon atoms of a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56—Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Light Receiving Elements (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
TW110124923A 2020-07-08 2021-07-07 1,3-苯并二㗁呃衍生物之製造方法 TW202216654A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2020117639 2020-07-08
JP2020-117639 2020-07-08

Publications (1)

Publication Number Publication Date
TW202216654A true TW202216654A (zh) 2022-05-01

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ID=79553255

Family Applications (1)

Application Number Title Priority Date Filing Date
TW110124923A TW202216654A (zh) 2020-07-08 2021-07-07 1,3-苯并二㗁呃衍生物之製造方法

Country Status (9)

Country Link
US (1) US20230257368A1 (https=)
EP (1) EP4180426A4 (https=)
JP (1) JP7720846B2 (https=)
KR (1) KR20230037488A (https=)
CN (1) CN116018335B (https=)
BR (1) BR112022026641A2 (https=)
IL (1) IL299730A (https=)
TW (1) TW202216654A (https=)
WO (1) WO2022009911A1 (https=)

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7208630B2 (en) * 2004-10-27 2007-04-24 University Of Kansas Heat shock protein 90 inhibitors
JP2007161674A (ja) * 2005-12-16 2007-06-28 Tanabe Seiyaku Co Ltd ピペリジン化合物およびその製法
WO2008071646A1 (en) * 2006-12-11 2008-06-19 Boehringer Ingelheim International Gmbh New pyridazine derivatives with mch antagonistic activity and medicaments comprising these compounds
LT3121175T (lt) * 2014-03-17 2020-03-10 Daiichi Sankyo Company, Limited 1,3-benzodioksazolo dariniai, kaip ezh1 ir (arba) ezh2 inhibitoriai
BR112018001688B1 (pt) * 2015-07-30 2023-05-02 Daiichi Sankyo Company, Limited Uso de um composto
CN106883125A (zh) * 2017-03-07 2017-06-23 怀化金鑫新材料有限公司 感光材料稳定剂4‑十六烷氧羰基氧基‑3，5‑二氯苯甲酸乙酯的合成方法
HRP20240793T1 (hr) * 2018-04-18 2024-09-13 Constellation Pharmaceuticals, Inc. Modulatori enzima koji modificiraju metil, njihovi pripravci i upotreba
EP3797108B1 (en) * 2018-05-21 2022-07-20 Constellation Pharmaceuticals, Inc. Modulators of methyl modifying enzymes, compositions and uses thereof
JP2020045306A (ja) * 2018-09-18 2020-03-26 第一三共株式会社 ヘテロシクロアルキル環を含むアミド誘導体

Also Published As

Publication number Publication date
JP7720846B2 (ja) 2025-08-08
EP4180426A1 (en) 2023-05-17
KR20230037488A (ko) 2023-03-16
BR112022026641A2 (pt) 2023-02-07
IL299730A (en) 2023-03-01
CA3185274A1 (en) 2022-01-13
EP4180426A4 (en) 2024-08-07
US20230257368A1 (en) 2023-08-17
WO2022009911A1 (ja) 2022-01-13
CN116018335A (zh) 2023-04-25
JPWO2022009911A1 (https=) 2022-01-13
CN116018335B (zh) 2025-10-10

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