IL268501A - Sulfoxyamine glycosidase inhibitors - Google Patents

Sulfoxyamine glycosidase inhibitors

Info

Publication number
IL268501A
IL268501A IL268501A IL26850119A IL268501A IL 268501 A IL268501 A IL 268501A IL 268501 A IL268501 A IL 268501A IL 26850119 A IL26850119 A IL 26850119A IL 268501 A IL268501 A IL 268501A
Authority
IL
Israel
Prior art keywords
sulfoximine
glycosidase inhibitors
glycosidase
inhibitors
sulfoximine glycosidase
Prior art date
Application number
IL268501A
Other languages
English (en)
Hebrew (he)
Original Assignee
Asceneuron Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/EP2017/054268 external-priority patent/WO2017144633A1/en
Priority claimed from PCT/EP2017/071385 external-priority patent/WO2018153508A2/en
Application filed by Asceneuron Sa filed Critical Asceneuron Sa
Publication of IL268501A publication Critical patent/IL268501A/en

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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
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CA3053200A1 (en) 2018-08-30
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US10556902B2 (en) 2020-02-11
MA47573A (fr) 2021-04-28
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US20190388415A1 (en) 2019-12-26
AU2017222964A1 (en) 2018-08-02
KR20230026541A (ko) 2023-02-24
KR20190118184A (ko) 2019-10-17
MA47574A (fr) 2020-01-01
US20190055239A1 (en) 2019-02-21
JP2019506430A (ja) 2019-03-07
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EP3419972B1 (en) 2023-07-26
BR112019017514A2 (pt) 2020-03-31

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