IL263996B2 - Solid forms of an sgc stimulator - Google Patents

Solid forms of an sgc stimulator

Info

Publication number
IL263996B2
IL263996B2 IL263996A IL26399618A IL263996B2 IL 263996 B2 IL263996 B2 IL 263996B2 IL 263996 A IL263996 A IL 263996A IL 26399618 A IL26399618 A IL 26399618A IL 263996 B2 IL263996 B2 IL 263996B2
Authority
IL
Israel
Prior art keywords
compound
crystalline free
disease
free form
diseases
Prior art date
Application number
IL263996A
Other languages
English (en)
Hebrew (he)
Other versions
IL263996A (en
IL263996B1 (en
Original Assignee
Ironwood Pharmaceuticals Inc
Cyclerion Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ironwood Pharmaceuticals Inc, Cyclerion Therapeutics Inc filed Critical Ironwood Pharmaceuticals Inc
Publication of IL263996A publication Critical patent/IL263996A/en
Publication of IL263996B1 publication Critical patent/IL263996B1/en
Publication of IL263996B2 publication Critical patent/IL263996B2/en

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
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    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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IL263996A 2016-07-07 2017-07-06 Solid forms of an sgc stimulator IL263996B2 (en)

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