IL160771A0 - Carbazole derivatives and their use as nyp5 receptor anatagonists - Google Patents

Carbazole derivatives and their use as nyp5 receptor anatagonists

Info

Publication number
IL160771A0
IL160771A0 IL16077102A IL16077102A IL160771A0 IL 160771 A0 IL160771 A0 IL 160771A0 IL 16077102 A IL16077102 A IL 16077102A IL 16077102 A IL16077102 A IL 16077102A IL 160771 A0 IL160771 A0 IL 160771A0
Authority
IL
Israel
Prior art keywords
nyp5
carbazole derivatives
receptor anatagonists
anatagonists
receptor
Prior art date
Application number
IL16077102A
Other languages
English (en)
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of IL160771A0 publication Critical patent/IL160771A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
IL16077102A 2001-09-11 2002-09-09 Carbazole derivatives and their use as nyp5 receptor anatagonists IL160771A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0121941.9A GB0121941D0 (en) 2001-09-11 2001-09-11 Chemical compounds
PCT/GB2002/004109 WO2003022849A1 (en) 2001-09-11 2002-09-09 Carbazole derivatives and their use as npy5 receptor antagonists

Publications (1)

Publication Number Publication Date
IL160771A0 true IL160771A0 (en) 2004-08-31

Family

ID=9921890

Family Applications (1)

Application Number Title Priority Date Filing Date
IL16077102A IL160771A0 (en) 2001-09-11 2002-09-09 Carbazole derivatives and their use as nyp5 receptor anatagonists

Country Status (14)

Country Link
US (1) US7408064B2 (xx)
EP (1) EP1427729A1 (xx)
JP (1) JP2005516892A (xx)
KR (1) KR20040036939A (xx)
CN (1) CN1653067A (xx)
BR (1) BR0212484A (xx)
CA (1) CA2459973A1 (xx)
GB (1) GB0121941D0 (xx)
IL (1) IL160771A0 (xx)
MX (1) MXPA04002338A (xx)
NO (1) NO20041008L (xx)
NZ (1) NZ531678A (xx)
WO (1) WO2003022849A1 (xx)
ZA (1) ZA200401956B (xx)

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WO2014139388A1 (en) 2013-03-14 2014-09-18 Merck Sharp & Dohme Corp. Novel indole derivatives useful as anti-diabetic agents
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JP6606491B2 (ja) 2013-06-05 2019-11-13 シナジー ファーマシューティカルズ インコーポレイテッド グアニル酸シクラーゼｃの超高純度アゴニスト、その作成および使用方法
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EP3551176A4 (en) 2016-12-06 2020-06-24 Merck Sharp & Dohme Corp. ANTIDIABETIC HETEROCYCLIC COMPOUNDS
EP3558298A4 (en) 2016-12-20 2020-08-05 Merck Sharp & Dohme Corp. ANTIDIABETIC SPIROCHROMAN COMPOUNDS

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Also Published As

Publication number Publication date
US20050065157A1 (en) 2005-03-24
ZA200401956B (en) 2005-04-15
CN1653067A (zh) 2005-08-10
NO20041008L (no) 2004-03-10
BR0212484A (pt) 2004-08-24
NZ531678A (en) 2005-09-30
EP1427729A1 (en) 2004-06-16
MXPA04002338A (es) 2004-06-29
WO2003022849A1 (en) 2003-03-20
KR20040036939A (ko) 2004-05-03
CA2459973A1 (en) 2003-03-20
JP2005516892A (ja) 2005-06-09
GB0121941D0 (en) 2001-10-31
US7408064B2 (en) 2008-08-05

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