IL159304A0 - Process for the production of piperidine derivatives - Google Patents

Process for the production of piperidine derivatives

Info

Publication number
IL159304A0
IL159304A0 IL15930402A IL15930402A IL159304A0 IL 159304 A0 IL159304 A0 IL 159304A0 IL 15930402 A IL15930402 A IL 15930402A IL 15930402 A IL15930402 A IL 15930402A IL 159304 A0 IL159304 A0 IL 159304A0
Authority
IL
Israel
Prior art keywords
production
piperidine derivatives
piperidine
derivatives
Prior art date
Application number
IL15930402A
Other languages
English (en)
Original Assignee
Aventis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh
Publication of IL159304A0 publication Critical patent/IL159304A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/66—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
    • C07C69/73—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of unsaturated acids
    • C07C69/738—Esters of keto-carboxylic acids or aldehydo-carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL15930402A 2001-06-15 2002-06-12 Process for the production of piperidine derivatives IL159304A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US29839701P 2001-06-15 2001-06-15
PCT/EP2002/006424 WO2002102776A1 (en) 2001-06-15 2002-06-12 Process for the production of the piperidine derivative fexofenadine

Publications (1)

Publication Number Publication Date
IL159304A0 true IL159304A0 (en) 2004-06-01

Family

ID=23150325

Family Applications (2)

Application Number Title Priority Date Filing Date
IL15930402A IL159304A0 (en) 2001-06-15 2002-06-12 Process for the production of piperidine derivatives
IL159304A IL159304A (en) 2001-06-15 2003-12-10 Process for the production of piperidine derivatives

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL159304A IL159304A (en) 2001-06-15 2003-12-10 Process for the production of piperidine derivatives

Country Status (22)

Country Link
US (2) US6743941B2 (enExample)
EP (1) EP1401816B1 (enExample)
JP (1) JP4344230B2 (enExample)
KR (1) KR100903285B1 (enExample)
CN (1) CN1229347C (enExample)
AR (1) AR037005A1 (enExample)
AT (1) ATE386021T1 (enExample)
AU (1) AU2002320847B2 (enExample)
BR (1) BR0210410A (enExample)
CA (1) CA2450313C (enExample)
DE (1) DE60225008T2 (enExample)
DK (1) DK1401816T3 (enExample)
ES (1) ES2298384T3 (enExample)
HU (1) HUP0401125A2 (enExample)
IL (2) IL159304A0 (enExample)
MX (1) MXPA03010960A (enExample)
NO (1) NO20035572L (enExample)
NZ (1) NZ530153A (enExample)
PL (1) PL364369A1 (enExample)
PT (1) PT1401816E (enExample)
WO (1) WO2002102776A1 (enExample)
ZA (1) ZA200308697B (enExample)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7498443B2 (en) * 2004-09-17 2009-03-03 Albany Molecular Research, Inc. Process for production of carebastine
US7498345B2 (en) * 2004-09-17 2009-03-03 Albany Molecular Research, Inc. Process for production of piperidine derivatives
CN100453522C (zh) * 2005-01-26 2009-01-21 中国科学技术大学 4-[4-(1-乙氧基酰基-1-甲基乙基苯)]-4-氧代丁酸的制备方法
WO2007135693A2 (en) * 2006-05-18 2007-11-29 Ind-Swift Laboratories Limited Intermediates useful for the preparation of antihistaminic piperidine derivative
ITMI20061491A1 (it) * 2006-07-27 2008-01-28 Archimica Srl Processo per la preparazione di fexofenadina.
ITMI20061492A1 (it) * 2006-07-27 2008-01-28 Archimica Srl Processo per la preparazione di fexofenadina.
CN102070490B (zh) * 2009-11-21 2014-07-30 浙江华海药业股份有限公司 一种非索非那定中间体2-(4-(4-羟基丁酰基)苯基)-2-甲基丙氰的制备方法
CN102070570A (zh) * 2009-11-21 2011-05-25 浙江华海药业股份有限公司 一种非索非那定中间体2-甲基-2(4-(2-氧代四氢呋喃-3-羰基)苯基)丙氰及其盐的制备方法
CA2986587C (en) 2015-06-15 2024-03-12 Asana Biosciences, Llc Heterocyclic inhibitors of erk1 and erk2 and their use in the treatment of cancer
CN104876853B (zh) * 2015-06-17 2017-06-16 苏州卫生职业技术学院 盐酸非索非那定的合成方法
CN109071438B (zh) 2015-10-22 2023-02-21 赛诺菲-安万特德国有限公司 用于制备非索非那定和其中使用的中间体的方法
EP3600302A4 (en) 2017-03-29 2020-12-30 United States Government as Represented by The Department of Veterans Affairs METHODS AND COMPOSITIONS FOR THE TREATMENT OF CANCER
US20230027072A1 (en) 2019-10-28 2023-01-26 Asana Biosciences, Llc Improved methods, kits, compositions and dosing regimens for the use of heterocyclic inhibitors of erk1 and erk2

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2946809A1 (de) * 1979-11-20 1981-06-11 A. Nattermann & Cie GmbH, 5000 Köln 4-phenyl-4-oxo-buttersaeuren, deren salze und ester, verfahren zu deren herstellung und diese enthaltende arzneimittel
IT1200123B (it) 1985-09-27 1989-01-05 Ind Chimica Srl Procedimento per la preparazione di alfa-(p-terbutilfenil)-4-(idrossidifenilmetil)-1-piperidinobutanolo
EP0347123A3 (en) 1988-06-17 1991-07-03 Fisons Corporation Dibenzo-cycloheptenyl, -cycloheptyl and -oxepinyl amines having antihistaminic properties
IT1249684B (it) 1991-07-19 1995-03-09 Sorin Biomedica Spa Epitopi della proteina env del virus dell'epatite c.
MX9302076A (es) * 1992-04-10 1994-03-31 Merrell Dow Pharma Proceso novedoso para preparar derivados de piperidina.
DK0703902T3 (da) 1993-06-24 1999-08-23 Albany Molecular Res Inc Fremgangsmåde til fremstilling af piperidinderivater

Also Published As

Publication number Publication date
KR20040010720A (ko) 2004-01-31
HK1063795A1 (en) 2005-01-14
DE60225008D1 (de) 2008-03-27
US20030105329A1 (en) 2003-06-05
BR0210410A (pt) 2004-08-17
NO20035572L (no) 2004-02-16
MXPA03010960A (es) 2004-02-27
EP1401816A1 (en) 2004-03-31
ATE386021T1 (de) 2008-03-15
US20040198983A1 (en) 2004-10-07
ZA200308697B (en) 2004-09-03
JP2005502603A (ja) 2005-01-27
JP4344230B2 (ja) 2009-10-14
CN1229347C (zh) 2005-11-30
PL364369A1 (en) 2004-12-13
CA2450313A1 (en) 2002-12-27
IL159304A (en) 2010-02-17
CN1516689A (zh) 2004-07-28
HUP0401125A2 (hu) 2004-09-28
PT1401816E (pt) 2008-04-08
US7235665B2 (en) 2007-06-26
EP1401816B1 (en) 2008-02-13
CA2450313C (en) 2010-08-10
US6743941B2 (en) 2004-06-01
NZ530153A (en) 2005-07-29
ES2298384T3 (es) 2008-05-16
WO2002102776A1 (en) 2002-12-27
DK1401816T3 (da) 2008-06-09
NO20035572D0 (no) 2003-12-12
DE60225008T2 (de) 2009-01-29
AR037005A1 (es) 2004-10-20
AU2002320847B2 (en) 2007-09-20
KR100903285B1 (ko) 2009-06-17

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