IL154590A0 - Fused pyrrolocarbozoles against inflammation - Google Patents
Fused pyrrolocarbozoles against inflammationInfo
- Publication number
- IL154590A0 IL154590A0 IL15459001A IL15459001A IL154590A0 IL 154590 A0 IL154590 A0 IL 154590A0 IL 15459001 A IL15459001 A IL 15459001A IL 15459001 A IL15459001 A IL 15459001A IL 154590 A0 IL154590 A0 IL 154590A0
- Authority
- IL
- Israel
- Prior art keywords
- pyrrolocarbozoles
- fused
- against inflammation
- inflammation
- pyrrolocarbozoles against
- Prior art date
Links
- 206010061218 Inflammation Diseases 0.000 title 1
- 230000004054 inflammatory process Effects 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Virology (AREA)
- Urology & Nephrology (AREA)
- Obesity (AREA)
- Epidemiology (AREA)
- Dermatology (AREA)
- Psychology (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Endocrinology (AREA)
- Communicable Diseases (AREA)
- Molecular Biology (AREA)
- Vascular Medicine (AREA)
- Tropical Medicine & Parasitology (AREA)
- AIDS & HIV (AREA)
- Ophthalmology & Optometry (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US22780300P | 2000-08-25 | 2000-08-25 | |
| US27845501P | 2001-03-23 | 2001-03-23 | |
| US09/935,285 US6630500B2 (en) | 2000-08-25 | 2001-08-22 | Selected fused pyrrolocarbazoles |
| PCT/US2001/026266 WO2002017914A2 (en) | 2000-08-25 | 2001-08-23 | Fused pyrrolocarbazoles against inflammation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL154590A0 true IL154590A0 (en) | 2003-09-17 |
Family
ID=27397767
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL15459001A IL154590A0 (en) | 2000-08-25 | 2001-08-23 | Fused pyrrolocarbozoles against inflammation |
| IL191104A IL191104A0 (en) | 2000-08-25 | 2008-04-27 | Fused pyrrolocarbazoles against inflammation |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL191104A IL191104A0 (en) | 2000-08-25 | 2008-04-27 | Fused pyrrolocarbazoles against inflammation |
Country Status (25)
| Country | Link |
|---|---|
| US (3) | US6630500B2 (da) |
| EP (1) | EP1311263B1 (da) |
| JP (1) | JP5399598B2 (da) |
| KR (1) | KR100810190B1 (da) |
| CN (1) | CN1298323C (da) |
| AR (1) | AR034143A1 (da) |
| AT (1) | ATE306920T1 (da) |
| AU (1) | AU8520501A (da) |
| BG (1) | BG66103B1 (da) |
| BR (1) | BR0113776A (da) |
| CA (1) | CA2420592C (da) |
| CZ (1) | CZ303707B6 (da) |
| DE (1) | DE60114215T2 (da) |
| DK (1) | DK1311263T3 (da) |
| EA (1) | EA006371B1 (da) |
| ES (1) | ES2250463T3 (da) |
| HU (1) | HU230128B1 (da) |
| IL (2) | IL154590A0 (da) |
| MX (1) | MXPA03001562A (da) |
| NO (1) | NO325689B1 (da) |
| NZ (1) | NZ524288A (da) |
| PL (1) | PL212956B1 (da) |
| SK (1) | SK287498B6 (da) |
| TW (1) | TWI299731B (da) |
| WO (1) | WO2002017914A2 (da) |
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| US9498530B2 (en) | 2002-12-24 | 2016-11-22 | Rinat Neuroscience Corp. | Methods for treating osteoarthritis pain by administering a nerve growth factor antagonist and compositions containing the same |
| US7569364B2 (en) | 2002-12-24 | 2009-08-04 | Pfizer Inc. | Anti-NGF antibodies and methods using same |
| BRPI0407375A (pt) | 2003-02-19 | 2006-02-07 | Rinat Neuroscience Corp | Métodos para tratar dor por meio da administração de um antagonista do fator de crescimento neural e u nsaid e composições contendo os mesmos |
| TW201319088A (zh) | 2003-07-18 | 2013-05-16 | Amgen Inc | 對肝細胞生長因子具專一性之結合劑 |
| US7241779B2 (en) * | 2003-12-23 | 2007-07-10 | Cephalon, Inc. | Fused pyrrolocarbazoles |
| US7169802B2 (en) * | 2003-12-23 | 2007-01-30 | Cephalon, Inc. | Fused pyrrolocarbazoles |
| PT2206728T (pt) | 2004-04-07 | 2018-04-17 | Rinat Neuroscience Corp | Métodos de tratamento da dor associada ao cancro ósseo através da administração de um anticorpo antagonista do fator de crescimento nervoso |
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| US20060134176A1 (en) * | 2004-12-22 | 2006-06-22 | Bausch & Lomb Incorporated | Pharmaceutical delivery system and method of use |
| US20060134175A1 (en) * | 2004-12-22 | 2006-06-22 | Stephen Bartels | Drug eluting pharmaceutical delivery system for treatment of ocular disease and method of use |
| US20060134174A1 (en) * | 2004-12-22 | 2006-06-22 | Bausch & Lomb Incorporated | Pharmaceutical delivery system and method of use |
| US20060216288A1 (en) * | 2005-03-22 | 2006-09-28 | Amgen Inc | Combinations for the treatment of cancer |
| US20060293378A1 (en) * | 2005-06-28 | 2006-12-28 | Mcintire Gregory | Method of lowering intraocular pressure |
| AR059066A1 (es) | 2006-01-27 | 2008-03-12 | Amgen Inc | Combinaciones del inhibidor de la angiopoyetina -2 (ang2) y el inhibidor del factor de crecimiento endotelial vascular (vegf) |
| PE20121506A1 (es) | 2006-07-14 | 2012-11-26 | Amgen Inc | Compuestos triazolopiridinas como inhibidores de c-met |
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| US9061009B2 (en) * | 2007-06-08 | 2015-06-23 | University Of Massachusetts | Mixed lineage kinases and metabolic disorders |
| CN101802008B (zh) | 2007-08-21 | 2015-04-01 | 安美基公司 | 人类c-fms抗原结合蛋白 |
| CN104016992B (zh) * | 2008-11-19 | 2017-04-12 | 赛福伦公司 | 吲唑并[5,4‑a]吡咯并[3,4‑c]咔唑化合物的形式 |
| EP2192121A1 (en) | 2008-11-27 | 2010-06-02 | Cephalon France | Regioselective reduction of fused pyrrolocarbazoles-5,7-diones |
| KR101038055B1 (ko) * | 2010-06-10 | 2011-06-01 | 송광섭 | 수중 마사지장치 |
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| DK2688887T3 (da) | 2011-03-23 | 2015-06-29 | Amgen Inc | Kondenserede tricykliske dualinhibitorer af cdk 4/6 og flt3 |
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| HK1247955A1 (zh) | 2015-01-08 | 2018-10-05 | 小利兰.斯坦福大学托管委员会 | 提供骨、骨髓及软骨的诱导的因子和细胞 |
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-
2001
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- 2001-08-23 SK SK219-2003A patent/SK287498B6/sk not_active IP Right Cessation
- 2001-08-23 AR ARP010104016A patent/AR034143A1/es not_active Application Discontinuation
- 2001-08-23 DE DE60114215T patent/DE60114215T2/de not_active Expired - Lifetime
- 2001-08-23 PL PL365683A patent/PL212956B1/pl unknown
- 2001-08-23 JP JP2002522887A patent/JP5399598B2/ja not_active Expired - Fee Related
- 2001-08-23 DK DK01964340T patent/DK1311263T3/da active
- 2001-08-23 BR BR0113776-0A patent/BR0113776A/pt not_active Application Discontinuation
- 2001-08-23 MX MXPA03001562A patent/MXPA03001562A/es active IP Right Grant
- 2001-08-23 AT AT01964340T patent/ATE306920T1/de active
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- 2001-08-23 CZ CZ20030539A patent/CZ303707B6/cs not_active IP Right Cessation
- 2001-08-23 EA EA200300293A patent/EA006371B1/ru not_active IP Right Cessation
- 2001-08-23 TW TW090120678A patent/TWI299731B/zh not_active IP Right Cessation
- 2001-08-23 AU AU8520501A patent/AU8520501A/xx active Pending
- 2001-08-23 ES ES01964340T patent/ES2250463T3/es not_active Expired - Lifetime
- 2001-08-23 WO PCT/US2001/026266 patent/WO2002017914A2/en not_active Ceased
- 2001-08-23 KR KR1020037002676A patent/KR100810190B1/ko not_active Expired - Fee Related
- 2001-08-23 NZ NZ524288A patent/NZ524288A/en unknown
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2006
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