IL151619A0 - N-(heterocyclyl) benzene or pyridine sulphonamides as antithrombotic agents and anticoagulants - Google Patents

N-(heterocyclyl) benzene or pyridine sulphonamides as antithrombotic agents and anticoagulants

Info

Publication number
IL151619A0
IL151619A0 IL15161901A IL15161901A IL151619A0 IL 151619 A0 IL151619 A0 IL 151619A0 IL 15161901 A IL15161901 A IL 15161901A IL 15161901 A IL15161901 A IL 15161901A IL 151619 A0 IL151619 A0 IL 151619A0
Authority
IL
Israel
Prior art keywords
sulphonamides
anticoagulants
heterocyclyl
pyridine
benzene
Prior art date
Application number
IL15161901A
Other languages
English (en)
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Publication of IL151619A0 publication Critical patent/IL151619A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72Nitrogen atoms
    • C07D213/73Unsubstituted amino or imino radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
IL15161901A 2000-03-23 2001-03-22 N-(heterocyclyl) benzene or pyridine sulphonamides as antithrombotic agents and anticoagulants IL151619A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0003724A FR2806722B1 (fr) 2000-03-23 2000-03-23 Derives de n-(heterocyclylbutyl) benzene-ou pyridine sulfonamide, leur preparation et leur application en therapeutique
PCT/FR2001/000861 WO2001070736A1 (fr) 2000-03-23 2001-03-22 N-(heterocyclyl)benzene-ou pyridine sulfonamides comme agents antithrombotiques et anticoagulantes

Publications (1)

Publication Number Publication Date
IL151619A0 true IL151619A0 (en) 2003-04-10

Family

ID=8848428

Family Applications (2)

Application Number Title Priority Date Filing Date
IL15161901A IL151619A0 (en) 2000-03-23 2001-03-22 N-(heterocyclyl) benzene or pyridine sulphonamides as antithrombotic agents and anticoagulants
IL151619A IL151619A (en) 2000-03-23 2002-09-04 N - (Tirocyclil) Gasoline or pyridine sulfonamides, processes for their preparation in their pharmaceutical preparations

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL151619A IL151619A (en) 2000-03-23 2002-09-04 N - (Tirocyclil) Gasoline or pyridine sulfonamides, processes for their preparation in their pharmaceutical preparations

Country Status (35)

Country Link
US (1) US6680329B2 (no)
EP (1) EP1268469B1 (no)
JP (1) JP2003528098A (no)
KR (1) KR100791693B1 (no)
CN (1) CN1183128C (no)
AR (1) AR029900A1 (no)
AT (1) ATE269325T1 (no)
AU (2) AU2001246617B2 (no)
BG (1) BG65863B1 (no)
BR (1) BR0109385A (no)
CA (1) CA2401637C (no)
DE (1) DE60103868T2 (no)
DK (1) DK1268469T3 (no)
EA (1) EA004986B1 (no)
EE (1) EE05084B1 (no)
ES (1) ES2222358T3 (no)
FR (1) FR2806722B1 (no)
HK (1) HK1051537A1 (no)
HR (1) HRP20020762B1 (no)
HU (1) HUP0300695A2 (no)
IL (2) IL151619A0 (no)
IS (1) IS2304B (no)
ME (1) MEP17408A (no)
MX (1) MXPA02009276A (no)
NO (1) NO324835B1 (no)
PL (1) PL204660B1 (no)
PT (1) PT1268469E (no)
RS (1) RS50370B (no)
SI (1) SI1268469T1 (no)
SK (1) SK286687B6 (no)
TR (1) TR200402343T4 (no)
TW (1) TWI290141B (no)
UA (1) UA71667C2 (no)
WO (1) WO2001070736A1 (no)
ZA (1) ZA200206996B (no)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8729107B2 (en) * 2002-12-06 2014-05-20 Purdue Research Foundation Pyridines for treating injured mammalian nerve tissue
DE60329415D1 (de) * 2002-12-06 2009-11-05 Purdue Research Foundation Pyridine zur behandlung von verletztemsäugetiernervengewebe
US7750162B2 (en) 2004-04-19 2010-07-06 Daiso Co., Ltd. Process for preparation of nonnatural amino acid and intermediate thereof
EP1739077A4 (en) * 2004-04-19 2008-04-16 Daiso Co Ltd PROCESS FOR THE PRODUCTION OF NON-NATURAL AMINO ACIDS AND INTERMEDIATES THEREFOR
GB0507577D0 (en) 2005-04-14 2005-05-18 Novartis Ag Organic compounds
US8586748B2 (en) * 2008-04-09 2013-11-19 Boehringer Ingelheim International Gmbh 2-sulfonylamino-4-heteroaryl butyramide antagonists of CCR10
EP2294051B1 (en) * 2008-05-22 2014-08-13 Boehringer Ingelheim International GmbH Alpha-substituted n-sulfonyl gylcine amides antagonists of ccr10, compositions containing the same and methods for using them
ES2569983T3 (es) * 2010-01-28 2016-05-13 The Medicines Company (Leipzig) Gmbh Inhibidores de serinproteasa de tipo tripsina y su preparación y uso
FR2981071B1 (fr) * 2011-10-10 2014-02-07 Centre Nat Rech Scient Synthese versatile et stereospecifique d'acides amines gamma,delta-insatures par la reaction de wittig

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2727410B1 (fr) * 1994-11-25 1996-12-20 Synthelabo Chlorures de sulfonyles, leur preparation et leur utilisation comme intermediaires de synthese
FR2728570B1 (fr) * 1994-12-23 1997-04-11 Synthelabo Derives de 1-oxo-2-(phenylsulfonylamino)pentylpiperidine, leur preparation et leur application en therapeutique
FR2756285B1 (fr) * 1996-11-22 1998-12-18 Synthelabo Derives de n-(imidazolylbutyle)benzenesulfonamide, leur preparation et leur application en therapeutique
FR2756220B1 (fr) * 1996-11-27 1998-12-24 Lorraine Laminage Roue pour vehicule terrestre a moteur
FR2771094B1 (fr) * 1997-11-19 2000-02-04 Synthelabo Derives de piperidine-2-carboxylate, leur preparation et leur application en therapeutique

Also Published As

Publication number Publication date
JP2003528098A (ja) 2003-09-24
EE200200540A (et) 2004-04-15
ES2222358T3 (es) 2005-02-01
MEP17408A (en) 2010-06-10
HUP0300695A2 (hu) 2003-07-28
WO2001070736A1 (fr) 2001-09-27
EA004986B1 (ru) 2004-10-28
YU67002A (sh) 2005-07-19
AR029900A1 (es) 2003-07-23
IL151619A (en) 2009-05-04
EP1268469A1 (fr) 2003-01-02
BR0109385A (pt) 2003-06-03
TR200402343T4 (tr) 2004-12-21
PL364988A1 (en) 2004-12-27
NO20024496D0 (no) 2002-09-19
PL204660B1 (pl) 2010-01-29
FR2806722B1 (fr) 2002-05-17
US20030207920A1 (en) 2003-11-06
UA71667C2 (uk) 2004-12-15
CA2401637A1 (en) 2001-09-27
ATE269325T1 (de) 2004-07-15
BG65863B1 (bg) 2010-03-31
EP1268469B1 (fr) 2004-06-16
US6680329B2 (en) 2004-01-20
PT1268469E (pt) 2004-10-29
IS6535A (is) 2002-08-30
SK286687B6 (sk) 2009-03-05
HRP20020762A2 (en) 2003-12-31
KR20020081476A (ko) 2002-10-26
FR2806722A1 (fr) 2001-09-28
HK1051537A1 (en) 2003-08-08
HRP20020762B1 (en) 2005-02-28
NO324835B1 (no) 2007-12-17
DK1268469T3 (da) 2004-10-11
DE60103868D1 (de) 2004-07-22
DE60103868T2 (de) 2005-06-09
ZA200206996B (en) 2003-09-01
AU2001246617B2 (en) 2006-03-02
MXPA02009276A (es) 2003-05-23
EA200200838A1 (ru) 2003-04-24
AU4661701A (en) 2001-10-03
CN1426407A (zh) 2003-06-25
TWI290141B (en) 2007-11-21
SI1268469T1 (en) 2004-10-31
CN1183128C (zh) 2005-01-05
IS2304B (is) 2007-10-15
BG107130A (bg) 2003-06-30
SK13512002A3 (sk) 2003-03-04
RS50370B (sr) 2009-11-10
EE05084B1 (et) 2008-10-15
KR100791693B1 (ko) 2008-01-03
CA2401637C (en) 2009-11-10
NO20024496L (no) 2002-11-22

Similar Documents

Publication Publication Date Title
DK1345918T3 (da) 1,5-benzothiazepiner og deres anvendelse som antihyperlipidæmiske midler
PL349781A1 (en) Novel sulfonamide compounds and uses thereof
NO996269D0 (no) Quinolin-indol antimikrobielle midler, samt anvendelse og blandinger derav
EE9900160A (et) Elastne vaheriie
DE69937649D1 (de) Mikromechanischer schalter und dessen herstellungsverfahren
ATE303388T1 (de) Substituierte 2-pyridinyl-6,7,8,9- tetrahydropyrimidoc1,2-aöpyrimidin-4-on- und 7- pyridinyl-2,3-dihydroimidazo-c1,2-aöpyrimidin- 5(1h)onderivate
IS5295A (is) Azetidínýlprópýlpíperidín afleiður, milliefni og notkun sem mótlyf gegn kínínhröðun
DE69806010D1 (de) Mikromechanischer Beschleunigungsschalter
DE50006919D1 (de) Femurschlitten
DK1246810T3 (da) Piperidinyloxy- og pyrrolidinyloxyphenyloxazolidinoner som antibakterielle midler
AU4661701A (en) N-(heterocyclyl)benzene or pyridine sulphonamides as antithrombotic agents and anticoagulants
AU2001246617A1 (en) N-(heterocyclyl)benzene or pyridine sulphonamides as antithrombotic agents and anticoagulants
DE60036580D1 (de) Türkontaktschalter
DE69832333D1 (de) Mikroelektromechanischer Schalter
ATE461989T1 (de) Reinigungs-mittel oder -bestandteile
DE69930169D1 (de) Mikromechanischer schalter
NO20015068D0 (no) Nya 8A- og 9A-15-medlemmers laktamer
DK1054662T3 (da) Vandoplöselige öjendråber
DE50107204D1 (de) 8beta-substituierte-11beta-pentyl-und 11beta-hexyl-estra-1,3,5(10)-trienderivate
NO20025549D0 (no) Bicyklyl- eller heterocyklylmetansulfonylaminosubstituerte N- hydroksyformamider
AU2001278714A1 (en) Vascular relaxation agents
DK1235809T3 (da) Substituerede 1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazociner og deres anvendelse som lægemidler
AU6924398A (en) N-(arginyl)benzenesulphonamide derivatives and use thereof as antithrombotic agents
ITMI992193A0 (it) Guanto perfezionato da lavoro facilmente indossabile e sfilabile
DE69921863D1 (de) Verbinden von elastomeren gegenständen